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3-[2-(3-methoxyphenyl)ethyl]-1-[(4-methyl-1H-imidazol-5-yl)methyl]piperidine
4-(azocane-1-carbonyl)-7,8-dimethyl-2-(pyrimidin-5-yl)quinoline
N-[(1S,2S)-2-(benzyloxy)cyclohexyl]-3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)propanamide
(1S,9S)-11-{[2-(morpholin-4-yl)-1,3-thiazol-5-yl]methyl}-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-6-one
1-(adamantan-2-yl)-4-[(2S,4S)-1-[(2,5-difluorophenyl)methyl]-4-[(4-methoxyphenyl)sulfanyl]pyrrolidine-2-carbonyl]piperazine
N'-cyclopentyl-N-[(2S)-1-hydroxy-3,3-dimethylbutan-2-yl]butanediamide
3-ethyl-6-{1-methyl-1,4,9-triazaspiro[5.5]undecane-4-carbonyl}-3H-imidazo[4,5-b]pyridin-2-amine
(4aS,7aR)-1-{[3-(morpholin-4-yl)phenyl]methyl}-4-propyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-{5-[3-(4-methoxyphenyl)-3-oxopropyl]-3-methyl-1H-1,2,4-triazol-1-yl}acetic acid
1-methyl-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
N-[(1R,3S)-3-(cyclobutylcarbamoyl)cyclopentyl]-2-(1H-1,2,4-triazol-3-yl)benzamide
N-ethyl-1-[2-(furan-2-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]pyrrolidine-3-carboxamide
2-[1-(3-phenylpropyl)-4-{[1-(pyridin-3-yl)-1H-pyrrol-2-yl]methyl}piperazin-2-yl]ethan-1-ol
N-{4,5-dimethyl-3-[4-(4-methyl-4H-1,2,4-triazol-3-yl)piperidine-1-carbonyl]thiophen-2-yl}-2-methylpropanamide
N-(1H-indol-4-ylmethyl)-4-(trimethyl-1H-pyrazol-4-yl)pyrimidin-2-amine
5-(3-acetylphenoxymethyl)-N-[2-(naphthalen-2-yl)ethyl]-1,2-oxazole-3-carboxamide
N-[(3-chlorophenyl)methyl]-N-cyclopropyl-2-(2-methyl-1H-imidazol-1-yl)propanamide
2-(2,4-dimethoxy-3-methylphenyl)-4-{[2-(2-methoxyphenyl)pyrrolidin-1-yl]methyl}-5-methyl-1,3-oxazole
2-(dimethylamino)-2-(3-fluorophenyl)-1-[6-(methylsulfanyl)-1,2,3,4-tetrahydroisoquinolin-2-yl]ethan-1-one
9-[(4-methyl-1H-imidazol-2-yl)methyl]-3,9-diazaspiro[5.6]dodecane
5-methyl-1-[(2-methyl-1,3-thiazol-4-yl)methyl]-5-phenylpiperidin-2-one
2-(2H-1,3-benzodioxol-5-yl)-2-{methyl[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]amino}acetic acid
(3R,4S)-3,4-dimethyl-1-[(4-methyl-6-phenylpyrimidin-2-yl)methyl]piperidin-4-ol
(2S,4S)-1-methyl-4-(2-methylpropanamido)-N-[3-(2-oxopyrrolidin-1-yl)propyl]pyrrolidine-2-carboxamide
N-({1-[(2-ethyl-1-benzofuran-3-yl)methyl]pyrrolidin-3-yl}methyl)-2,2-difluoroacetamide
N-[(6-hydroxy-2-methylpyrimidin-4-yl)methyl]-3-(3-hydroxy-3-methylbutyl)benzamide
(4aS,7aR)-1-[3-(3-hydroxy-1,2-oxazol-5-yl)propanoyl]-4-(3-methylbut-2-en-1-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
{[2-(cyclopentylmethyl)-1H-imidazol-4-yl]methyl}(methyl)(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)amine
1-methyl-N-(3-phenylpropyl)-6-(pyridin-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
(1S,5R)-6-(2-methoxyethyl)-3-[3-(pyridin-4-yl)-1H-pyrazole-5-carbonyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
2-{1-[(5-tert-butyl-1,2,4-oxadiazol-3-yl)methyl]pyrrolidin-2-yl}-5-fluoro-1H-1,3-benzodiazole
6-[1-(3,5-dimethylphenoxy)ethyl]-3-propyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazole
N-[2-(5-chloro-1H-1,3-benzodiazol-2-yl)ethyl]-5-cyclobutyl-N-methyl-1,3,4-oxadiazol-2-amine
2-methyl-8-{[3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-2,8-diazaspiro[4.5]decane-3-carboxylic acid
(3S,4R)-3-acetamido-N-(2-phenylphenyl)-4-(propan-2-yl)pyrrolidine-1-carboxamide
(1H-1,3-benzodiazol-2-ylmethyl)(methyl)(oxolan-2-ylmethyl)amine
N-[2-(3-chlorophenyl)ethyl]-5-ethylpyrimidin-2-amine
2-[3-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)phenyl]ethan-1-amine
5-(2,3-dihydro-1H-isoindole-2-carbonyl)-1-(2-ethoxyethyl)-2,3-dihydro-1H-1,3-benzodiazol-2-one
2-(4-{2-[(3-chloro-4-fluorophenyl)carbamoyl]acetyl}morpholin-3-yl)acetic acid
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-(2-methylpyrimidin-4-yl)piperidin-3-ol
1-[2-(4-acetyl-6-hydroxy-1,4-diazepan-1-yl)-2-oxoethyl]-1,2-dihydropyridin-2-one
5-methanesulfonyl-N,2-dimethyl-N-{3-[(4-methylphenyl)sulfanyl]propyl}pyrimidin-4-amine
N-(furan-2-ylmethyl)-5-[1-(3,3,3-trifluoropropanoyl)pyrrolidin-2-yl]thiophene-2-carboxamide
3-[(3R,4S)-4-(4-methylpiperazin-1-yl)-1-(pyrazin-2-yl)piperidin-3-yl]propan-1-ol
ethyl 4-[4-(4-{[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]amino}piperidin-1-yl)benzoyl]piperazine-1-carboxylate
2-(2-hydroxyethyl)-8-(1-phenylcyclopentanecarbonyl)-2,8-diazaspiro[5.5]undecan-3-one
2-(methylamino)-N-[(5-methylthiophen-2-yl)methyl]-N-(prop-2-en-1-yl)pyridine-3-carboxamide
[(3-chloro-4,5-dimethoxyphenyl)methyl](methyl)[3-(1H-pyrazol-1-yl)propyl]amine
[5-({3-[(2H-1,3-benzodioxol-5-yl)amino]piperidin-1-yl}methyl)-2-(propan-2-yloxy)phenyl]methanol