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1-(2-{4-[4-(3-methoxyphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-2-oxoethyl)-1,2-dihydropyrimidin-2-one
N-{[(3S,4S)-1-[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl]-3-hydroxypiperidin-4-yl]methyl}-2,2-dimethylpropanamide
3-{1-[4-(1H-1,2,4-triazol-1-yl)butanoyl]piperidin-3-yl}benzoic acid
1-[2-(2,5-dimethylphenyl)ethyl]-5-oxopyrrolidine-3-carboxylic acid
4-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-1-(1-methylpiperidin-4-yl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
N-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-1-(5-methylthiophene-2-carbonyl)piperidine-2-carboxamide
N-[3-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]-1-(2-methylfuran-3-carbonyl)piperidine-2-carboxamide
N-{3-[2-(dimethyl-1,2-oxazol-4-yl)pyrrolidin-1-yl]-3-oxopropyl}-4-fluorobenzamide
3-(1H-imidazol-2-yl)-1-[3-(5-methylthiophen-2-yl)-1H-pyrazole-5-carbonyl]piperidine
N4-[(1R,2S)-2-phenylcyclohexyl]-1H-pyrazolo[3,4-d]pyrimidine-4,6-diamine
1-methyl-4-{[1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl}piperazine-2-carboxylic acid
1'-{1-[4-(4-ethylpiperazine-1-carbonyl)phenyl]piperidin-4-yl}spiro[indene-1,4'-piperidine]
(3S,5S)-1-[(5-ethylfuran-2-yl)methyl]-5-[(6-methylpyridin-3-yl)carbamoyl]piperidine-3-carboxylic acid
5-{5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-3-carboxamide
(3aS,6aS)-2-{[2-(trifluoromethoxy)phenyl]methyl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-4-(4-fluorophenyl)-1,4-diazepane
ethyl 2-[4-(benzenesulfonyl)piperazin-1-yl]-1,3-oxazole-4-carboxylate
1-{2-[3-(4-methoxyphenoxymethyl)piperidin-1-yl]-2-oxoethyl}azepan-2-one
2-methyl-6-(2-{[4-(pyridin-2-yl)pyrimidin-2-yl]amino}ethyl)pyrimidin-4-ol
N-benzyl-N-methyl-2-(thiomorpholine-4-carbonyl)-2,3-dihydro-1H-inden-2-amine
N-(2-methyl-1-benzofuran-7-yl)-4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazine-1-carboxamide
2-(3-methoxypropyl)-9-[(4-methylphenyl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
9-[2-(adamantan-1-ylsulfanyl)acetyl]-1,4,9-triazaspiro[5.5]undecan-5-one
2-[(4-{4-[(3-fluorophenyl)methyl]-1,4-diazepane-1-carbonyl}phenyl)sulfanyl]ethan-1-ol
1-(4-acetyl-4-phenylpiperidin-1-yl)-2-[3-(dimethylamino)pyrrolidin-1-yl]ethan-1-one
N,1-dimethyl-N-[(3-methylpyridin-2-yl)methyl]-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
tert-butyl (2R,3R)-3-amino-2-(pyridin-3-ylmethoxy)-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-carboxylate
(3S,4R)-4-(3-methoxyphenyl)-1-[2-(methylsulfanyl)benzoyl]pyrrolidine-3-carboxylic acid
7-[3-(3-hydroxyquinoxalin-2-yl)propanoyl]-1-oxa-3,7-diazaspiro[4.5]decan-2-one
7-(2-hydroxyethyl)-2-[2-(3-oxo-2,3-dihydro-1H-indazol-2-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
3-(3-hydroxy-1,2-oxazol-5-yl)-N-methyl-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]propanamide
1-[(3,4-difluorophenyl)methyl]-3-hydroxy-3-({[2-methyl-1-(pyrrolidin-1-yl)propan-2-yl]amino}methyl)piperidin-2-one
N-[(2-chloro-4-fluorophenyl)methyl]-4-[(5-methyl-1H-1,2,3,4-tetrazol-1-yl)methyl]benzamide
2-{4-[1-(3-chlorophenyl)piperidin-4-yl]-1-(cyclohexylmethyl)piperazin-2-yl}ethan-1-ol
4-{[3-(2H-1,3-benzodioxol-5-ylmethyl)-3-methylpiperidin-1-yl]methyl}-N-methyl-1,3-thiazol-2-amine
3-[2-(2-fluorophenyl)ethyl]-N,N-dimethylpiperidine-1-sulfonamide
N-[2-(cyclohex-1-en-1-yl)ethyl]-2-{1-[(4-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
2-chloro-5-{1-[2-(2-methylpropanesulfonyl)ethyl]-1H-1,2,3-triazol-4-yl}pyridine
2-(4-oxo-3,4-dihydroquinazolin-3-yl)-N-(1H-1,2,3,4-tetrazol-5-ylmethyl)acetamide
2-methoxy-4-{3-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyridine
N-({5,7-dimethylimidazo[1,2-a]pyridin-2-yl}methyl)-2-(2,5-dioxoimidazolidin-4-yl)acetamide
[(2S,6S)-11-methoxy-4-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-trien-6-yl]methanol
1-{2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carbonyl}-4-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}piperidine
N-[(1-ethyl-1H-imidazol-2-yl)methyl]-2-{1-[(2-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-methylacetamide
2-(propan-2-yl)-8-(pyridin-2-yl)-2,8-diazaspiro[5.5]undecan-3-one
methyl (2S)-2-{[(2,3,4,9-tetrahydro-1H-carbazol-6-ylmethyl)carbamoyl]amino}propanoate
{2-[3-(1H-1,3-benzodiazol-2-ylmethyl)piperidin-1-yl]-1,3-thiazol-4-yl}methanol
[(2-fluorophenyl)methyl]({[1-(2-methoxyethyl)piperidin-4-yl]methyl})(oxolan-2-ylmethyl)amine
N-{1-[4-(2,4-dioxoimidazolidin-1-yl)benzoyl]piperidin-4-yl}methanesulfonamide
5-(1,4-dioxan-2-yl)-1-[2-(1H-imidazol-5-yl)ethyl]-3-[(2-methoxyphenyl)methyl]-1H-1,2,4-triazole