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N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-5-[(methylsulfanyl)methyl]furan-2-carboxamide
N-[(4-{2-[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]ethoxy}-3-methoxyphenyl)methyl]-2-methyl-N-[(3S)-2-oxoazepan-3-yl]-1,3-thiazole-4-carboxamide
1-ethyl-4-[3-(3-methoxyphenoxymethyl)piperidine-1-carbonyl]-1,2-dihydropyridin-2-one
2-{2-[1-(3-methylpyridin-4-yl)-3-(propan-2-yl)-1H-1,2,4-triazol-5-yl]ethyl}pyrazine
11-(1-benzyl-1H-imidazol-5-yl)-4,6,10,12-tetraazatricyclo[7.3.0.03,7]dodeca-1,3(7),8,10-tetraen-5-one
(3R,5S)-1-[(3,4-dimethoxyphenyl)methyl]-N-[2-(1-methylpyrrolidin-2-yl)ethyl]-5-[(pyridin-3-yloxy)methyl]piperidine-3-carboxamide
N-[(4-fluorophenyl)methyl]-3-[1-(isoquinolin-5-ylmethyl)piperidin-4-yl]propanamide
8-[(1-methyl-1H-indol-3-yl)methyl]-1-(2-methylpropyl)-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-(1H-pyrazol-3-yl)-1,3-benzothiazole-5-carboxamide
3-({4-[1-(propane-2-sulfonyl)pyrrolidin-3-yl]piperidin-1-yl}methyl)pyridine
[7-(4-ethyl-5-methylpyrimidin-2-yl)-5-methyl-2,3-dihydro-1-benzofuran-2-yl]methanamine
6-(2H-1,3-benzodioxol-5-yl)-N-[3-(pyridin-2-yl)propyl]pyridine-3-carboxamide
4-(5,6-dimethoxy-1-oxo-1,2-dihydroisoquinolin-2-yl)butanamide
2-{[1-(oxane-4-carbonyl)piperidin-3-yl]methyl}-1H-1,3-benzodiazole
(3R,4R)-4-{[2-(dimethylamino)-6-(trifluoromethyl)pyrimidin-4-yl]amino}piperidin-3-ol
N-[(3,5-dimethyl-2-phenyl-1H-indol-7-yl)methyl]-2-(methylamino)pyrimidine-5-carboxamide
N-[4-(ethylsulfanyl)phenyl]-4-(3-methylpyridin-4-yl)-1,4-diazepane-1-carboxamide
1-(azocan-1-yl)-3-{5-[(cyclopropylamino)methyl]-2-methoxyphenoxy}propan-2-ol
1-(1-{imidazo[1,2-a]pyrimidin-2-yl}propyl)-2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazole
N-tert-butyl-7-{[3-(dimethylamino)pyrrolidin-1-yl]sulfonyl}-1,2,3,4-tetrahydroisoquinoline-2-carboxamide
2-methyl-5-[1-(1-methylpiperidin-4-yl)-3-(phenoxymethyl)-1H-1,2,4-triazol-5-yl]pyrazine
3-(2-hydroxyphenyl)-3-(3-hydroxyphenyl)-N-methyl-N-(oxan-4-yl)propanamide
3-{2-[4-(2-cyclobutyl-5-fluoro-1H-1,3-benzodiazol-1-yl)piperidin-1-yl]-2-oxoethyl}-2,3-dihydro-1H-isoindol-1-one
2-methyl-N-[(3-methyloxetan-3-yl)methyl]-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine
4-{1-[(2-methyloxolan-2-yl)methyl]-1H-imidazol-2-yl}pyridine
1-{4-[(dimethylamino)methyl]-4-hydroxyazepan-1-yl}-2-(2-methyl-1,3-thiazol-4-yl)ethan-1-one
2-{2-[2-(1-methyl-1H-imidazol-2-yl)-1H-imidazol-1-yl]propyl}pyrazine
(3R,4R)-3-{ethyl[(4-methyl-2-oxo-2H-chromen-7-yl)methyl]amino}-4-hydroxy-1λ6-thiolane-1,1-dione
5-methoxy-3-methyl-2-({2-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidin-1-yl}methyl)-1H-indole
N-benzyl-3-cyclopropyl-N-(1,1-dioxo-1λ6-thiolan-3-yl)-1H-pyrazole-5-carboxamide
2-(3-methoxypropyl)-1-(3-methyl-1-propyl-1H-pyrazole-4-carbonyl)piperidine
4-[2-(methylsulfanyl)benzoyl]-2-(2-phenylethyl)morpholine
(3S,4R)-1-(1H-indole-2-carbonyl)-4-(3-methoxyphenyl)pyrrolidine-3-carboxylic acid
5-(2,6-difluorophenoxymethyl)-N-methyl-N-(piperidin-3-ylmethyl)-1,2-oxazole-3-carboxamide
4-[3-(carbamoylmethyl)-1-(2-hydroxybutyl)-1H-1,2,4-triazol-5-yl]-N,N-dimethylpiperidine-1-carboxamide
1-[(1-{6-[(cyclopent-3-en-1-yl)amino]pyridine-3-carbonyl}piperidin-4-yl)methyl]pyrrolidin-2-one
2-methoxyethyl (4aS,7aR)-4-[2-(dimethylamino)acetyl]-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxylate
5-{4-[(1,2-dimethyl-1H-imidazol-5-yl)methyl]piperazin-1-yl}-2-methyl-2,3-dihydropyridazin-3-one
N-[(2,2-dimethyl-1-phenylcyclopropyl)methyl]-3-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)propanamide
4-(1-{1-[(2,5-dimethylphenyl)methyl]piperidin-3-yl}-1H-1,2,3-triazole-4-carbonyl)morpholine
N-(2H-1,3-benzodioxol-5-ylmethyl)-N-methyl-5-[1-(piperidin-1-yl)ethyl]furan-2-carboxamide
N-[2-(dimethyl-1H-1,2,4-triazol-1-yl)ethyl]-8-methyl-2-propyl-2,8-diazaspiro[4.5]decane-3-carboxamide
[(1-{1-[1-(4-fluorophenyl)pyrrolidin-3-yl]piperidin-4-yl}-1H-1,2,3-triazol-4-yl)methyl]urea
N-[3-(2-amino-1,3-thiazol-4-yl)propyl]-5,6-dimethylpyrimidin-4-amine
5-[(5,6-dimethyl-1H-1,3-benzodiazol-1-yl)methyl]-N-(oxolan-2-ylmethyl)-1H-pyrazole-3-carboxamide
2-phenyl-N-[1-(1,3-thiazol-2-yl)ethyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
(3S,4R)-1-{2-[(dimethylcarbamoyl)amino]acetyl}-4-(2-methylphenyl)pyrrolidine-3-carboxylic acid
3-({[3-(3-fluorophenyl)oxolan-3-yl]methyl}amino)-4-hydroxybenzonitrile
2-{[4-(3,6-dimethylpyrazin-2-yl)piperazin-1-yl]methyl}-6-methoxyphenol
(1R,4S)-N-(2,3-dihydro-1H-inden-2-yl)-N,1,7,7-tetramethyl-3-oxo-2-oxabicyclo[2.2.1]heptane-4-carboxamide