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3-[(3S,7S,8aS)-3-[(4-hydroxyphenyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(3-chloro-2-methylphenyl)urea
N-(3-chloro-4-ethoxyphenyl)-4-(pyridin-4-ylmethyl)-1,4-diazepane-1-carboxamide
1-{4-[4-ethyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-(4H-1,2,4-triazol-4-yl)ethan-1-one
(3R)-1-{[2-(3-chlorophenyl)-5,8-dimethoxyquinolin-3-yl]methyl}pyrrolidin-3-ol
N-[(4-methoxyphenyl)(pyridin-4-yl)methyl]-2-(5-{[methyl(propan-2-yl)amino]methyl}-1H-1,2,3,4-tetrazol-1-yl)acetamide
2-[2-({[3-(dimethyl-1,2-oxazol-4-yl)propyl]carbamoyl}amino)phenyl]-N,N-dimethylacetamide
1-[(2,2-dimethyl-2,3-dihydro-1-benzofuran-5-yl)methyl]-3-(3-methyl-1H-1,2,4-triazol-5-yl)piperidine
1-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)sulfonyl]-N-methyl-N-[2-(pyridin-2-yl)ethyl]piperidin-3-amine
4-{3-[3-hydroxy-3-(hydroxymethyl)piperidin-1-yl]-3-oxopropyl}-N-methylbenzene-1-sulfonamide
N-{3-[(5-methylpyridin-2-yl)amino]propyl}-3,4-dihydro-2H-1-benzopyran-3-carboxamide
{[7-methoxy-2-(thiophen-2-yl)quinolin-3-yl]methyl}(methyl)(pyrimidin-4-ylmethyl)amine
2-(1-{[2-(2-fluoro-5-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-3-yl)-1,3-benzoxazole
methyl({[1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}){4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}amine
7-{3-[2-(2,6-difluorophenyl)ethyl]piperidine-1-carbonyl}quinolin-8-ol
4-{5-[3-(3-methylphenyl)piperidine-1-carbonyl]-1H-pyrazol-3-yl}phenol
N-[3-(3-ethylphenoxy)propyl]-N,1-dimethylazepane-2-carboxamide
N-{1-[1-(4-methoxybenzoyl)piperidin-4-yl]-1H-pyrazol-5-yl}oxolane-3-carboxamide
3-[1-(5-acetylthiophen-2-yl)-N-methylformamido]-N-methylpropanamide
1-(cyclohexylmethyl)-N-[(3-fluoro-4-methoxyphenyl)methyl]piperidin-3-amine
2-{4-[(4-chlorophenyl)methyl]-4-(hydroxymethyl)piperidin-1-yl}pyridine-3-carbonitrile
1-[3-(pyridine-3-carbonyl)piperidin-1-yl]-3-(trimethyl-1H-pyrazol-4-yl)propan-1-one
[(1R,3S,3aS,6aR)-3-[2-chloro-5-methoxy-4-(prop-2-en-1-yloxy)phenyl]-1,5-dimethyl-octahydropyrrolo[3,4-c]pyrrol-1-yl]methanol
N-[2-(1-{[2-(2,4-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-4-yl)ethyl]acetamide
3-({8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2,4,6-tetraen-3-yl}amino)azepan-2-one
2-cyclopropyl-N-(isoquinolin-5-ylmethyl)-N-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
2-(4-{[5-methyl-2-(3-phenoxyphenyl)-1,3-oxazol-4-yl]methyl}piperazin-1-yl)acetic acid
N-(2-methylpropyl)-1-[(1s,4s)-4-[2-(2-methoxyphenyl)acetamido]cyclohexyl]-1H-1,2,3-triazole-4-carboxamide
2-(3-cyanopyrazin-2-yl)-N,N-dimethylbenzamide
6-methyl-N-{[1-(2-methylpropyl)pyrrolidin-3-yl]methyl}-4-oxo-1,4-dihydropyridine-3-carboxamide
N-[1-(cyclohex-1-en-1-yl)ethyl]-3-(4-methyl-1,3-thiazol-5-yl)propanamide
3-methyl-7-({3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
3-{5-[4-(1H-pyrrol-1-ylmethyl)benzoyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanoic acid
N-[(1-hydroxycyclohexyl)methyl]-3-(1H-imidazol-2-yl)benzamide
1-[3-({[2-(dimethylamino)ethyl](methyl)amino}methyl)phenoxy]-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-ol
7-[(2,3-difluorophenyl)methyl]-2-[(2-methoxypyrimidin-5-yl)methyl]-2,7-diazaspiro[4.5]decane
propan-2-yl 4-chloro-3-{2-[4-(dimethylamino)-6-oxo-1,6-dihydropyridazin-1-yl]acetamido}benzoate
1-{4-[4-(4-methoxyphenoxy)piperidine-1-carbonyl]thiophen-2-yl}ethan-1-one
N-(2-hydroxyethyl)-2-(propan-2-yl)-N-propylpyrimidine-5-carboxamide
5-methyl-2-(3-methylthiophen-2-yl)-4-{2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-ylmethyl}-1,3-oxazole
4-(dimethyl-1,2-oxazol-4-yl)-3-(1H-indol-3-ylmethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
3-(4-methyl-1,3-thiazol-5-yl)-N-(5-oxo-1-phenylpyrrolidin-3-yl)propanamide
ethyl({[5-methyl-2-(naphthalen-1-yl)-1,3-oxazol-4-yl]methyl})[2-(1H-pyrazol-1-yl)ethyl]amine
1-{3-[2-(2,4-difluorophenyl)ethyl]piperidin-1-yl}-3-(1H-1,2,4-triazol-1-yl)propan-1-one
2-(4-{[2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl}-1-(thiophen-3-ylmethyl)piperazin-2-yl)ethan-1-ol
(2-{4-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-1,3-thiazol-4-yl)methanol
methyl(oxolan-2-ylmethyl){[1-(piperidin-4-yl)-1H-1,2,3-triazol-4-yl]methyl}amine
8-[(2,6-difluorophenyl)methyl]-1-oxa-8-azaspiro[4.6]undecan-9-one
1-benzoyl-N-[1-(pyrrolidin-1-ylmethyl)cyclohexyl]piperidin-4-amine
N-[(2-benzyl-1,3-thiazol-4-yl)methyl]-4-[(3-methoxypropyl)amino]-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
4-[(1E)-3-[3-(3-chlorobenzoyl)piperidin-1-yl]prop-1-en-1-yl]-2-methoxyphenol