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N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-1-methyl-2-oxo-1,2-dihydroquinoline-3-carboxamide
4-ethyl-1-{[5-methyl-2-(thiophen-2-yl)-1,3-oxazol-4-yl]methyl}-3-(piperidin-4-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[(2S,4R,6S)-2-(3,5-dichloropyridin-4-yl)-6-(2-methylpropyl)oxan-4-yl]acetamide
3-(2-ethyl-7-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-N-[2-(morpholin-4-yl)-2-(pyridin-3-yl)ethyl]propanamide
1-(3,4-dimethylphenyl)-N-(thian-4-yl)-4,5,6,7-tetrahydro-1H-indazol-4-amine
1-[1'-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]propan-1-one
1-{3-[2-(pyridin-4-yl)-1H-imidazol-1-yl]propyl}-1H-1,2,3-benzotriazole
1-{4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]benzoyl}-N,N-dimethylpyrrolidin-3-amine
6-{1-[1-(2-methoxyethyl)piperidine-3-carbonyl]piperidin-4-yl}pyrimidin-4-ol
4-(3-phenyl-1,2-oxazole-5-carbonyl)-2-(1H-pyrazol-1-ylmethyl)-1,4-oxazepane
1-[2-methoxy-5-({[3-(4-methyl-1,3-thiazol-5-yl)propyl]amino}methyl)phenoxy]-3-(pyrrolidin-1-yl)propan-2-ol
9-(2-methoxypyridine-4-carbonyl)-1-oxa-9-azaspiro[5.5]undecan-5-ol
2-(5-amino-1,3,4-thiadiazol-2-yl)-1-{4-[(2E)-3-phenylprop-2-en-1-yl]piperazin-1-yl}ethan-1-one
2-chloro-4-[3-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]pyridine
3-[(3R,4S)-1-(isoquinoline-5-carbonyl)-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propan-1-ol
1-(1'-{4H-thieno[3,2-b]pyrrole-5-carbonyl}-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl)propan-1-one
(2S,4R)-4-[4-(cyclohexylmethyl)-1H-1,2,3-triazol-1-yl]-N-ethylpyrrolidine-2-carboxamide
(2R,6R)-11-methoxy-4-[3-(2-methyl-1H-imidazol-1-yl)propyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
2-[1-benzyl-4-(1-benzylpiperidin-4-yl)piperazin-2-yl]ethan-1-ol
1-{4-[4-(1,2,3,4-tetrahydroisoquinolin-2-yl)piperidine-1-carbonyl]thiophen-2-yl}ethan-1-one
4-[(3-methoxyphenyl)methyl]-1-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}piperidine-4-carboxylic acid
1-{2-[methyl({[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl})amino]ethyl}cyclopentan-1-ol
1-[(3R,4S)-3-amino-4-(3-methoxyphenyl)pyrrolidin-1-yl]-2-(7-fluoro-2-methyl-1H-indol-3-yl)ethan-1-one
3-{[(2-cyclopentylethyl)amino]methyl}-1-[(2-fluoro-5-methoxyphenyl)methyl]-3-hydroxypiperidin-2-one
N-(1-ethyl-1H-indazol-3-yl)-2-(1H-imidazol-1-yl)acetamide
1-[3-(diphenylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-2-(1H-pyrazol-1-yl)ethan-1-one
N-{[7-(4-methanesulfonylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-methoxypropanamide
N-benzyl-N,5-dimethyl-4-[(pyridin-2-ylmethyl)amino]thieno[2,3-d]pyrimidine-6-carboxamide
methyl 2-{4-[(1-cyclopentyl-1H-imidazol-5-yl)methyl]-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-2-yl}acetate
2-[4-(dimethylamino)phenyl]-N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]acetamide
2-methyl-5-{2-phenyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-1,3,4-oxadiazole
(4aS,8aS)-2-{[3-hydroxy-5-(hydroxymethyl)-2-methylpyridin-4-yl]methyl}-decahydroisoquinolin-4a-ol
N-(furan-2-ylmethyl)-N-(prop-2-en-1-yl)-4-[(pyridin-4-ylmethyl)amino]benzamide
3,6-dimethyl-N-[1-(3-methylpyridin-2-yl)propan-2-yl]-[1,2]oxazolo[5,4-d]pyrimidin-4-amine
1-[(1-methyl-1H-pyrazol-4-yl)methyl]-6-(pyridin-3-ylmethoxy)-4-{[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}-1,4-diazepan-2-one
2-{1-[1-methyl-3-(2-methylpropyl)-1H-pyrazol-5-yl]-N-(1-methylpiperidin-4-yl)formamido}acetic acid
1-{2-[7-(cyclopropylmethyl)-6-oxo-2,7-diazaspiro[4.5]decan-2-yl]-2-oxoethyl}-5,5-dimethylimidazolidine-2,4-dione
N-cyclopropyl-3-(4-methyl-1,3-thiazol-5-yl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]propanamide
4-(4-fluoro-2-methylbenzoyl)-1-(4-methoxyphenyl)piperazin-2-one
(1S,5R)-3-[(dimethyl-1,2-oxazol-4-yl)methyl]-6-[2-methyl-2-(morpholin-4-yl)propyl]-3,6-diazabicyclo[3.2.2]nonane
1-(2-methoxy-5-{[(2-methoxyethyl)(methyl)amino]methyl}phenoxy)-3-(4-methylpiperazin-1-yl)propan-2-ol
1-(furan-2-ylmethyl)-4-(2,3,4,5-tetrahydro-1-benzoxepine-4-carbonyl)piperazine
methyl 3-[({5,7-dimethylpyrazolo[1,5-a]pyrimidin-2-yl}formamido)methyl]-5-(2-methoxybenzamido)benzoate
2-cyclopentyl-8-(2-methylpyridin-4-yl)-2,8-diazaspiro[5.5]undecan-3-one
methyl 4-[(4-{4-[(propan-2-yl)carbamoyl]-1H-1,2,3-triazol-1-yl}piperidin-1-yl)methyl]benzoate
5-(3-{2-[3-(1H-pyrazol-1-yl)phenyl]-1H-imidazol-1-yl}propyl)-1H-1,2,3,4-tetrazole
4-(4-methylphenoxy)-N-{2-[(pyridin-3-yl)amino]ethyl}piperidine-4-carboxamide
1-({3-[(1-cyclohexanecarbonylpiperidin-3-yl)methoxy]phenyl}methyl)-4-(2-fluorophenyl)piperazine
5-{3-ethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}-1-(2-methoxyethyl)piperidin-2-one
[(3R,4R)-4-{[(2-methoxyethyl)(methyl)amino]methyl}-1-(2-methyl-1,3-benzothiazole-6-carbonyl)pyrrolidin-3-yl]methanol