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4-[1-(propan-2-yl)-1H-imidazol-2-yl]-1-[4-(trifluoromethyl)benzoyl]piperidine
2-(dimethylamino)-2-(4-fluorophenyl)-N-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}acetamide
1-[3-(1H-imidazol-2-yl)piperidin-1-yl]-2-(4-methyl-1,4-diazepan-1-yl)ethan-1-one
N-methyl-2-propyl-N-[1-(pyrimidin-4-yl)ethyl]-1,3-thiazole-4-carboxamide
N-[(5-methoxy-1,3-benzoxazol-2-yl)methyl]-2-(thiophen-2-yl)-1,3-thiazole-4-carboxamide
2-[4-(2-methyl-1,2,3,4-tetrahydroisoquinoline-3-carbonyl)piperazin-1-yl]pyridine-3-carbonitrile
N-(oxolan-2-ylmethyl)-3-{1-[(3-phenyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}propanamide
1-cyclopropyl-N-(3-hydroxypropyl)-N-(naphthalen-1-ylmethyl)-6-oxopiperidine-3-carboxamide
1-{[1-(2-methoxyethyl)-1H-imidazol-2-yl]methyl}-N-methylpiperidine-2-carboxamide
4-(5-methyl-1-propyl-1H-pyrazol-4-yl)-N-[2-(1-methylpyrrolidin-2-yl)ethyl]pyrimidin-2-amine
(1,4-dioxan-2-ylmethyl)({2-[(3-fluorophenyl)methoxy]-6-methylquinolin-3-yl}methyl)amine
1-(2-methoxy-5-methylphenyl)-3-[2-(propan-2-ylsulfanyl)ethyl]urea
[(2S)-1-{[3-(2H-1,3-benzodioxol-5-yl)-1-benzyl-1H-pyrazol-4-yl]methyl}pyrrolidin-2-yl]methanol
1-[2-(4-fluoro-2-methylphenyl)acetyl]-N-(6-methylpyridin-3-yl)piperazine-2-carboxamide
N-(1-cycloheptylpiperidin-3-yl)-3-{5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-6-yl}propanamide
N-cyclopropyl-3-{5-[2-(1-methyl-1H-pyrrol-2-yl)-2-oxoacetyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanamide
N-{[5-(2-methylpropyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}-2-(2-oxo-1,2-dihydropyridin-1-yl)acetamide
2-(5-fluoro-1-methyl-1H-indole-2-carbonyl)-7-methyl-2,7-diazaspiro[4.5]decan-6-one
N-(2-methylphenyl)-N'-[2-(pyridin-4-ylformamido)ethyl]propanediamide
5-[4-(2,5-dimethylphenyl)piperazine-1-carbonyl]-N-ethyl-1-(2-methylpropyl)-4-oxo-1,4-dihydropyridine-3-carboxamide
2-[benzyl(methyl)amino]-1-{5-hydroxy-1-oxa-9-azaspiro[5.5]undecan-9-yl}ethan-1-one
2,4-dimethoxy-6-[3-(pentan-2-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-1,3,5-triazine
(3S,4R)-1-(3-fluoro-4-methylbenzoyl)-4-phenylpyrrolidine-3-carboxylic acid
2-(3-methoxyphenoxymethyl)-N-methyl-N-[(2-methyl-1,3-thiazol-4-yl)methyl]-1,3-oxazole-4-carboxamide
5-chloro-N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]thiophene-2-carboxamide
1-{[3,5-dimethyl-2-(1H-pyrazol-1-yl)phenyl]methyl}-2-methyl-1,4-diazepan-5-one
N-(2,2-dimethyloxan-4-yl)-2-(4-methoxybenzamido)-7-oxo-4,5,6,7-tetrahydro-1,3-benzothiazole-5-carboxamide
5-cyclobutanecarbonyl-1'-[3-(methylsulfanyl)propyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
(4aS,8aR)-1-(4-hydroxybutyl)-6-(6-methylpyridazin-3-yl)-decahydro-1,6-naphthyridin-2-one
3-(5-{[benzyl(1,3-thiazol-2-ylmethyl)amino]methyl}thiophen-3-yl)prop-2-yn-1-ol
8-(4-carbamoylpyridin-2-yl)-2-propyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
N-[1-(1H-imidazol-1-yl)-3,3-dimethylbutan-2-yl]-1-(4,6,7-trimethylquinazolin-2-yl)piperidin-4-amine
{1-[1-(4-methoxyphenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}[(3-methylquinoxalin-2-yl)methyl]amine
2-({[4-(methylsulfanyl)phenyl]methyl}(pyridin-2-ylmethyl)amino)ethan-1-ol
3-[3-(pyrrolidin-1-yl)propyl]-1-[3-(1H-1,2,4-triazol-1-yl)phenyl]urea
N-[2-(morpholin-4-yl)ethyl]-2-(3-phenylpropyl)-1,3-benzoxazole-5-carboxamide
1-[(3R,4S)-3-amino-4-phenylpyrrolidin-1-yl]-4-(thiophen-2-yl)butan-1-one
2-[3-(3-methoxyphenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]acetic acid
1-[4-(4-chlorophenoxy)piperidin-1-yl]-3-(4-methyl-4H-1,2,4-triazol-3-yl)propan-1-one
8-(6-aminopyrimidin-4-yl)-2-[(4-chlorophenyl)methyl]-2,8-diazaspiro[4.5]decan-3-one
4-methoxy-N-{[1-(2-methoxyacetyl)piperidin-3-yl]methyl}benzene-1-sulfonamide
N-{5-[(2-methylphenyl)methyl]-1,3,4-thiadiazol-2-yl}-4-phenyl-1,4-diazepane-1-carboxamide
3-[2-(2,6-difluorophenyl)ethyl]-1-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)propyl]piperidine
1-(diethylamino)-3-[2-methoxy-5-({[2-(4-methylphenyl)ethyl]amino}methyl)phenoxy]propan-2-ol
2-{1-[(4-chloro-3-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]acetamide
2-[2-(butan-2-yl)phenoxy]-1-[4-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]ethan-1-one
1-(cyclohexylmethyl)-N-[4-(1H-pyrazol-1-yl)butan-2-yl]-1H-1,2,3-triazole-4-carboxamide
2-(methylsulfanyl)-4-{3-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyrimidine
7-chloro-N-[5-(trifluoromethyl)-1,3,4-thiadiazol-2-yl]-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carboxamide
{5-[3-(pyridin-3-ylmethoxy)piperidine-1-carbonyl]-1H-1,3-benzodiazol-2-yl}methanol