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3-{1-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]piperidin-4-yl}-1-(4-phenylpiperazin-1-yl)propan-1-one
N-(3-ethyl-1,4-dimethyl-1H-pyrazol-5-yl)-4-(pyridin-3-ylmethoxy)piperidine-1-carboxamide
4-{1H-pyrrolo[2,3-b]pyridin-4-yl}phthalazin-1-ol
2-ethyl-9-{3-fluoroimidazo[1,2-a]pyridine-2-carbonyl}-2,9-diazaspiro[5.5]undecan-3-one
1-[4-(methylamino)-5H,6H,7H-cyclopenta[d]pyrimidin-2-yl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
1-[(2,6-difluorophenyl)methyl]-N-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}-1H-1,2,3-triazole-4-carboxamide
5-(2H-1,3-benzodioxol-5-ylmethyl)-1-[2-(6-hydroxy-2-methylpyrimidin-4-yl)ethyl]-5-methylpiperidin-2-one
(2S,3S)-2-{[1-(4-chlorophenyl)propan-2-yl]amino}-3-methylpentan-1-ol
(2S)-3-(4-hydroxyphenyl)-2-{[2-(1H-1,2,3,4-tetrazol-5-yl)phenyl]formamido}propanamide
2-(isoquinolin-1-yl)-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one
N-(1,3-dimethyl-1H-pyrazol-5-yl)-2-[3-(2-fluoro-4-methoxyphenyl)-1H-pyrazol-1-yl]acetamide
N-cyclooctyl-1-(2-methoxyethyl)-4-oxo-5-{1,3,3-trimethyl-6-azabicyclo[3.2.1]octane-6-carbonyl}-1,4-dihydropyridine-3-carboxamide
7-(2-phenylquinoline-4-carbonyl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
1-[5-({[2-(3-fluorophenyl)ethyl]amino}methyl)-2-methoxyphenoxy]-3-(pyrrolidin-1-yl)propan-2-ol
N4,N4-diethyl-6-[3-(2-methylpiperidin-1-yl)azetidin-1-yl]pyrimidine-2,4-diamine
N-[(3,4-difluorophenyl)methyl]-3-[1-(5-methoxyfuran-2-carbonyl)piperidin-3-yl]propanamide
3-(4-methoxy-2-methylbenzoyl)-1-{2-methylimidazo[1,2-a]pyrimidine-3-carbonyl}piperidine
3-[N-(pyridin-3-ylmethyl)-2-(2,4,7-trimethyl-1H-indol-3-yl)acetamido]propanoic acid
6-{[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]amino}pyridine-3-carboxamide
N-methyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-2-phenyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
N4-methyl-N4-(oxolan-2-ylmethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
9-ethyl-1-methyl-4-(1-methyl-3-propyl-1H-pyrazole-5-carbonyl)-1,4,9-triazaspiro[5.6]dodecan-10-one
N-{[2-(4-acetylpiperazin-1-yl)pyridin-3-yl]methyl}-4-sulfamoylbutanamide
5-[(1-benzylpiperidin-4-yl)amino]-1-(cyclohexylmethyl)-N,N-dimethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
(2R,3R)-1'-[(4-chloro-1-methyl-1H-pyrazol-3-yl)methyl]-3-(dimethylamino)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
N-[2-({[(1-methyl-1H-pyrazol-4-yl)methyl](2-methylpropyl)amino}methyl)quinolin-6-yl]acetamide
ethyl (4aR,6R,8aS)-6-(morpholin-4-yl)-2-(thiophen-2-ylmethyl)-decahydroisoquinoline-8a-carboxylate
1-ethyl-N-(furan-3-ylmethyl)-N-methyl-5-{[2-(methylsulfanyl)ethyl]amino}-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
ethyl 2-[(3R,4R)-3-hydroxy-4-{methyl[2-(pyridin-2-yl)ethyl]amino}piperidin-1-yl]-1,3-oxazole-4-carboxylate
1-(cyclopropylmethyl)-N-methyl-5-(2-phenylacetyl)-N-(1,3-thiazol-4-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
(3aS,6aS)-2-(1H-imidazol-4-ylmethyl)-5-(2-methoxypyridine-3-carbonyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-cyclopentyl-4-(1H-pyrrole-3-carbonyl)-1,4-diazepane-6-carboxylic acid
N-cyclopentyl-1-{1-[(2,5-dimethylphenyl)methyl]piperidin-3-yl}-1H-1,2,3-triazole-4-carboxamide
2-(dimethylamino)-N-({1-[2-(2-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-N-methylacetamide
3-[(3S,4R)-1-(pyridin-3-ylmethyl)-4-{4-[3-(trifluoromethyl)phenyl]piperazin-1-yl}piperidin-3-yl]-1-(thiomorpholin-4-yl)propan-1-one
4-(5-methylfuran-2-yl)-N-(pyridin-2-ylmethyl)benzamide
3-(2-fluorophenyl)-N-(2-hydroxyethyl)-N-[(2-methylphenyl)methyl]-1H-pyrazole-5-carboxamide
N-[(3R,4S)-1-(oxan-4-yl)-4-(propan-2-yl)pyrrolidin-3-yl]-4-(1H-1,2,4-triazol-1-yl)butanamide
4-(1H-imidazol-1-ylmethyl)-1-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)piperidin-4-ol
1-(2-fluorophenyl)-4-[(3-{[1-(furan-2-carbonyl)piperidin-3-yl]methoxy}phenyl)methyl]piperazine
3-[2-(2-chloro-6-fluorophenyl)-N-methylacetamido]-N-methylbutanamide
3-methyl-N-{[3-(thiophen-2-ylmethyl)-1,2,4-oxadiazol-5-yl]methyl}-1,2-oxazole-5-carboxamide
N-methyl-1-(propan-2-yl)-N-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}piperidine-4-carboxamide
N-({2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}methyl)-5-(morpholin-4-ylmethyl)furan-3-carboxamide
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-5-(3-methyl-1,2-oxazol-5-yl)furan-2-sulfonamide
(3S,4S)-1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-4-(morpholin-4-yl)pyrrolidin-3-ol
3-(3-fluorophenyl)-1-[4-(3-methylpyridin-4-yl)-1,4-diazepan-1-yl]propan-1-one
3,3-dimethyl-1-{[5-(2-phenylpropyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}urea
N-{1-[1-(2-hydroxybutyl)piperidin-4-yl]-1H-pyrazol-5-yl}benzamide
3-chloro-6-{4-[(6-methoxy-2H-chromen-3-yl)methyl]piperazin-1-yl}pyridazine