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N-[1-methyl-5-(4-phenylpiperidine-1-carbonyl)-2-(pyridin-4-yl)-1H-1,3-benzodiazol-7-yl]cyclobutanecarboxamide
3-{[3-cyclopentyl-1-(2-hydroxyethyl)-1H-1,2,4-triazol-5-yl]methyl}-4-(propan-2-yl)piperazin-2-one
(2R)-N-[1-methyl-4-(pyridin-3-yloxy)-1H-indazol-3-yl]oxolane-2-carboxamide
2-(dimethylamino)-2-(4-fluorophenyl)-1-[4-(pyrrolidine-1-carbonyl)piperidin-1-yl]ethan-1-one
2-[(4-methyl-1,3-thiazol-2-yl)sulfanyl]-N-{2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}acetamide
methyl (2S,4S,5R)-5-(2-chlorophenyl)-4-[(3-hydroxy-2,2-dimethylpropyl)carbamoyl]-1,2-dimethylpyrrolidine-2-carboxylate
3-{5-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)propyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanoic acid
(3R,4R)-1-[(6-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-4-(morpholin-4-yl)piperidin-3-ol
6-ethoxy-2-{4-[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl]-1,4-diazepan-1-yl}-4-methylquinazoline
2-(phenylsulfanyl)-1-[3-(pyridin-3-ylmethoxy)piperidin-1-yl]ethan-1-one
N-[(6-chloropyridin-3-yl)methyl]-5-ethyl-4-(pyrrolidin-1-ylmethyl)furan-2-carboxamide
(1S,5R)-6-[(dimethylcarbamoyl)methyl]-N-(2-methylphenyl)-7-oxo-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
1-[1'-(6-aminopyrimidin-4-yl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]propan-1-one
N-[2-(diethylamino)-2-(furan-2-yl)ethyl]-3-[(2-fluorophenyl)formamido]propanamide
3-{4-[6-amino-5-cyano-4-(furan-2-yl)pyridin-2-yl]-3,5-dimethyl-1H-pyrazol-1-yl}propanoic acid
N-{[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]methyl}-2-(1,2,3,4-tetrahydroisoquinolin-2-yl)propanamide
N-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]-6-(methoxymethyl)pyridine-2-carboxamide
8-[3-(4-hydroxyphenyl)-1H-pyrazole-5-carbonyl]-2-methyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
1-methyl-5-{[2-methyl-2-(morpholin-4-yl)propyl]amino}-N-(thiophen-2-ylmethyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
3-(2-oxo-2-{3-phenyl-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl}ethyl)-2,3-dihydro-1H-isoindol-1-one
3-[2-(7-{[(2S)-4-methyl-2-phenylpiperazin-1-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-2-oxoethyl]-1,3-thiazolidine-2,4-dione
(4aS,8aR)-1-(2-methylpropyl)-6-[3-(1,2-oxazolidin-2-yl)propanoyl]-decahydro-1,6-naphthyridin-2-one
N-{2-[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]ethyl}-1,6-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-{[8-(4-cyclopentylpyrimidin-2-yl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}acetamide
(2S,4S)-4-amino-N,N-diethyl-1-[(4-methoxypiperidin-1-yl)sulfonyl]pyrrolidine-2-carboxamide
6-[1-(2-amino-4-phenylpyrimidine-5-carbonyl)piperidin-3-yl]pyrimidin-4-ol
1-(2,3-dihydro-1H-inden-2-yl)-4-(oxolan-3-ylmethyl)-1,4-diazepane
3-hydroxy-1-[(3-methylphenyl)methyl]-3-({[(5-methylpyrazin-2-yl)methyl]amino}methyl)piperidin-2-one
N-cyclopentyl-N-[(2,5-dimethoxyphenyl)methyl]-2-(2,5-dioxoimidazolidin-4-yl)acetamide
6-[(3R,5R)-3-[(dimethylamino)methyl]-5-(hydroxymethyl)piperidine-1-carbonyl]-2-methyl-4H,7H-pyrazolo[1,5-a]pyrimidin-7-one
N-[2-(3-{[methyl(thiophen-3-ylmethyl)amino]methyl}phenoxy)propyl]-2,1,3-benzothiadiazole-4-sulfonamide
2-benzyl-N-[(1,5-dimethyl-1H-pyrazol-3-yl)methyl]-1,3-benzoxazole-5-carboxamide
3-(6-methoxynaphthalene-2-carbonyl)-1-(1,3-thiazole-5-carbonyl)piperidine
N-(1-carbamoylcycloheptyl)-5-(pyrrolidin-1-ylmethyl)furan-2-carboxamide
3-(4-methylpiperazine-1-carbonyl)-1-propyl-5-(thiomorpholin-4-yl)-4,5,6,7-tetrahydro-1H-indazole
(3S,4S)-4-methyl-1-[1-(4-methylbenzoyl)piperidine-4-carbonyl]piperidine-3,4-diol
(1S,5R)-6-(cyclopropylmethyl)-3-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}-3,6-diazabicyclo[3.2.2]nonane
methyl(1,2-oxazol-5-ylmethyl)[(2,3,4-trimethoxyphenyl)methyl]amine
3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}propanamide
{2-fluoro-5-[2-(morpholin-4-ylmethyl)phenoxy]phenyl}methanol
N-cyclopentyl-1-(2-ethoxyethyl)-2-oxo-N-propyl-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
3-hydroxy-S-(2-propanoyl-1,2,3,4-tetrahydroisoquinolin-7-yl)butane-1-sulfonamido
1'-[3-(5-methyl-1H-1,2,4-triazol-3-yl)propanoyl]-1,2-dihydrospiro[indole-3,3'-piperidine]-2-one
1-{5-[4-(4-phenylpyrimidin-2-yl)piperazine-1-carbonyl]-1H-pyrazol-3-yl}ethan-1-one
2-(cyclopropylmethyl)-9-(2-methoxy-3-methylbenzoyl)-2,9-diazaspiro[5.5]undecan-3-one
5-[4-(3-methoxyphenyl)piperazine-1-carbonyl]-1,3-benzothiazol-2-amine
2,3,5-trimethyl-N-[2-(morpholin-4-yl)butyl]pyrazolo[1,5-a]pyrimidin-7-amine
2-({3-[methyl({[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl})carbamoyl]phenyl}amino)acetic acid
2-{4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyridin-3-ol
[1-(5-fluoro-2-methylbenzenesulfonyl)-3-(3-methoxypropyl)piperidin-3-yl]methanol