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2-{[1-(2-chlorophenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}pyridine
5-{1-[2-(2-chlorophenyl)acetyl]piperidin-4-yl}-3-(oxolan-2-ylmethyl)-5-(pyridin-2-yl)imidazolidine-2,4-dione
5-[3-(2-methoxyphenoxy)azetidine-1-carbonyl]-3-methyl-1H-pyrazole
N-[(3,5-difluoro-4-methoxyphenyl)methyl]-7-fluoro-2-methylquinoline-4-carboxamide
(2S,4S)-4-(cycloheptylamino)-N,N-diethyl-1-(pyridin-4-ylmethyl)pyrrolidine-2-carboxamide
(4aS,7aR)-1-({3-[2-(dimethylamino)ethoxy]phenyl}methyl)-4-methyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-{2-oxo-2-[4-(2-phenoxyethyl)piperazin-1-yl]ethyl}-1λ6-thiolane-1,1-dione
3-[3-({[(2-amino-1,3-thiazol-4-yl)methyl]amino}methyl)-1H-indol-1-yl]propanamide
N-[(2-ethylpyrimidin-4-yl)methyl]-N-methyl-2,3-dihydro-1H-inden-2-amine
6-methyl-N4-{[1-(4-methylpiperazin-1-yl)cyclohexyl]methyl}pyrimidine-2,4-diamine
4-(3-methyl-1,2,4-oxadiazol-5-yl)-2-[2-(piperidin-1-ylmethyl)phenoxy]pyridine
(4aR,7aS)-1-{2-[(3-methoxypropyl)(methyl)amino]pyrimidin-4-yl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[1-(1,3-benzothiazol-2-yl)piperidin-3-yl]-4-(1H-pyrazol-4-yl)butanamide
7-(2H-1,3-benzodioxole-5-carbonyl)-2-methyl-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
ethyl 1-[4-(1H-pyrazol-1-yl)butan-2-yl]-4-{[2-(trifluoromethyl)phenyl]methyl}piperidine-4-carboxylate
1-(4-{[({1-[2-(2-methoxyphenyl)ethyl]piperidin-3-yl}methyl)(methyl)amino]methyl}thiophen-2-yl)ethan-1-one
5-[4-(2-methoxyphenyl)-2-methylpiperazine-1-carbonyl]-4-methyl-2-(propan-2-yl)pyrimidine
4-cyano-N-({5-cyclohexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)benzamide
(benzylsulfamoyl)[2-(4-methyl-1,3-thiazol-5-yl)ethyl]amine
(1R,7S)-N-methyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-4-oxo-3-(pentan-3-yl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
[(4-ethyl-4H-1,2,4-triazol-3-yl)methyl](methyl){[2-(morpholin-4-yl)-1,3-thiazol-5-yl]methyl}amine
N-[(3,5-dichlorophenyl)methyl]-2,8-diazaspiro[4.5]decane-3-carboxamide
N-[(1-hydroxycyclohexyl)methyl]-2-{3-oxo-1-[(2E)-3-phenylprop-2-en-1-yl]piperazin-2-yl}acetamide
3-[1-(6-methylpyridine-2-carbonyl)piperidin-3-yl]-N-[4-(trifluoromethyl)phenyl]propanamide
8-(oxan-4-yl)-1-(2-phenylethyl)-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-(2H-1,2,3-benzotriazol-2-yl)-1-[(3R,4R)-3-(hydroxymethyl)-4-[(4-hydroxypiperidin-1-yl)methyl]pyrrolidin-1-yl]ethan-1-one
N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]quinoline-5-carboxamide
4-(5-methylfuran-2-yl)-N-[3-(1H-1,2,3,4-tetrazol-5-yl)propyl]benzamide
[(3R,4R)-1-[4-(dimethylamino)benzoyl]-4-(piperidin-1-ylmethyl)pyrrolidin-3-yl]methanol
5-phenyl-N-[1-(pyrazin-2-yl)piperidin-4-yl]-1,2-oxazole-3-carboxamide
3-(1-{[3-(2-fluoro-4-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}pyrrolidin-2-yl)-4-methyl-1,2,5-oxadiazole
N-[(3R,4S)-4-cyclopropyl-1-[(3-methylpyrazin-2-yl)methyl]pyrrolidin-3-yl]propane-1-sulfonamide
N-{5,6-dimethylthieno[2,3-d]pyrimidin-4-yl}-1-oxa-8-azaspiro[4.5]decan-3-amine
2,6,8-trimethyl-4-[4-(4H-1,2,4-triazol-3-yl)piperidine-1-carbonyl]quinoline
8-methyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-2-propyl-2,8-diazaspiro[4.5]decane-3-carboxamide
3-{[4-(pyridin-2-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}pyridin-2-amine
2-[2-(dimethylamino)-1,3-thiazol-5-yl]-N,1-bis(propan-2-yl)-1H-1,3-benzodiazole-5-sulfonamide
2-({4-[4-methyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)-1H-1,3-benzodiazole
4-(2-amino-4-ethyl-1,3-thiazole-5-carbonyl)-1-cyclopentylpiperazin-2-one
1-(methoxymethyl)-N-[2-(2-phenoxyphenyl)ethyl]cyclobutane-1-carboxamide
N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}-N-[3-(dimethylamino)propyl]acetamide
1-{5-[3-(2,3-dimethoxyphenyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}-1,4-diazepane
3-[4-(3-hydroxyphenyl)piperidine-1-carbonyl]-N,N-dimethylpiperidine-1-carboxamide
3-(3-hydroxy-1,2-oxazol-5-yl)-1-[(3R,4R)-3-(hydroxymethyl)-4-(morpholin-4-ylmethyl)pyrrolidin-1-yl]propan-1-one
2-methoxy-5-[3-(4-phenyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]pyrimidine
1-[1-(1,4-dimethyl-1H-indole-2-carbonyl)piperidin-4-yl]-3-methylbutan-1-ol
1-[(5-chlorothiophen-2-yl)methyl]-4-[4-(methoxymethyl)-1H-1,2,3-triazol-1-yl]piperidine
ethyl 3-benzyl-1-{[2-(methoxycarbonyl)phenyl]carbamoyl}piperidine-3-carboxylate
2-methoxyethyl 2-(pyrrolidine-1-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carboxylate
(3R,4R)-1-[(2-chlorophenyl)methyl]-4-[4-(pyridin-2-yl)piperazin-1-yl]piperidin-3-ol