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1-[(5-{1-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-1H-1,2,3-triazol-4-yl}thiophen-3-yl)methyl]piperidine
4-hydroxy-2-{[7-(hydroxymethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]methyl}quinoline-6-carboxamide
N-{[4-(1H-1,2,4-triazol-1-yl)phenyl]methyl}-1,2-oxazole-5-carboxamide
2-[(3-chlorophenyl)methyl]-N-methyl-N-[3-(morpholin-4-yl)propyl]-1,3-benzoxazole-6-carboxamide
3-(1,3-dimethyl-1H-pyrazol-5-yl)-4-(5-fluoro-2-methylphenyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
1-benzyl-N,5-dimethyl-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-1H-1,2,3-triazole-4-carboxamide
1-(4-{5-fluoro-2-[(2-methoxyphenyl)methyl]-1H-1,3-benzodiazol-1-yl}piperidin-1-yl)-2-(3-methoxyphenyl)ethan-1-one
2-(morpholin-4-yl)-1-[4-(thiophen-3-yl)phenyl]ethan-1-ol
2-(adamantan-1-yl)-N-{[5-(furan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}acetamide
N4-[3-(dimethyl-1H-1,2,4-triazol-1-yl)propyl]-5-ethylpyrimidine-2,4-diamine
2-[3-(2-methoxyethyl)-5-[(2-methylphenyl)methyl]-1H-1,2,4-triazol-1-yl]acetic acid
2-{[(2,1,3-benzoxadiazol-5-ylmethyl)amino]methyl}-5,8-dimethylquinolin-4-ol
N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-2-(ethylamino)-N-methylpyrimidine-5-carboxamide
methyl 1-[(3R,5S)-5-[4-(4-fluorophenyl)piperazine-1-carbonyl]-1-{[(4S)-4-(prop-1-en-2-yl)cyclohex-1-en-1-yl]methyl}pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
N-methyl-N-{[3-(pyridin-2-yl)-1,2-oxazol-5-yl]methyl}-4-(3,3,3-trifluoropropyl)pyrimidin-2-amine
2-(dimethylamino)-2-(2-fluorophenyl)-N-[1-(pyridin-4-ylmethyl)piperidin-4-yl]acetamide
methyl 3-[(2S)-1-acetylpyrrolidine-2-carbonyl]-7-oxo-9-[2-(thiophen-2-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
1-(cyclobutylmethyl)-3-({[(3,5-difluorophenyl)methyl]amino}methyl)-3-hydroxypiperidin-2-one
3-(naphthalen-1-ylmethyl)-N-(oxan-4-ylmethyl)-4,5-dihydro-1,2-oxazole-5-carboxamide
2-[cyclopentyl(methyl)amino]-1-[4-(4-methoxyphenoxy)piperidin-1-yl]ethan-1-one
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-2-[4-(1H-1,2,3,4-tetrazol-1-yl)phenyl]acetamide
N-ethyl-3-methyl-N-[2-(2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazol-1-yl)ethyl]aniline
2-(cyclohex-1-en-1-yl)-1-[(1S,6R)-3,9-diazabicyclo[4.2.1]nonan-9-yl]ethan-1-one
1-[(3R,4R)-4-amino-3-hydroxypiperidin-1-yl]-2-{[(3,5-dimethylphenyl)methyl]sulfanyl}ethan-1-one
N-[(1S,3aS,6aS)-octahydropentalen-1-yl]-2-propyl-1,3-thiazole-4-carboxamide
1-[4-(6-aminopyrimidin-4-yl)-6-hydroxy-1,4-diazepan-1-yl]ethan-1-one
10-methoxy-5-(3-phenyl-1,2-oxazole-5-carbonyl)-3,4,5,6-tetrahydro-2H-1,5-benzoxazocine
N-[2-(5-cyclopentyl-1,2,4-oxadiazol-3-yl)ethyl]-3-(1H-pyrazol-1-yl)benzamide
2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]-N-[2-(3,5-dimethoxyphenyl)ethyl]acetamide
3-[4-(1-{[4-(hydroxymethyl)phenyl]methyl}-4-phenyl-1H-imidazol-5-yl)phenyl]prop-2-yn-1-ol
4-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-4H-1,2,4-triazole
2-(dimethyl-1,2-oxazol-4-yl)-1-{3-[4-(2-methylphenyl)piperazin-1-yl]piperidin-1-yl}ethan-1-one
2-[4-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]-4-methoxypyrimidine
1-(3-{[5-(4-chlorophenyl)-4-phenyl-1H-imidazol-1-yl]methyl}piperidin-1-yl)ethan-1-one
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-(1-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}piperidin-3-yl)piperazine
3-[(2-ethylbutyl)amino]-N-[3-(1H-imidazol-1-yl)propyl]-5-(phenylsulfamoyl)benzamide
2-(dimethylamino)-2-(3-methylphenyl)-N-{[2-(pyrimidin-2-yl)-1,3-thiazol-4-yl]methyl}acetamide
(1S,6R)-9-{[5-(3-hydroxy-3-methylbut-1-yn-1-yl)thiophen-2-yl]methyl}-3-methyl-3,9-diazabicyclo[4.2.1]nonan-4-one
3-(4-methyl-1H-pyrazol-1-yl)-5-(pyrrolidine-1-sulfonyl)benzoic acid
6-methoxy-3-methyl-N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}-1-benzofuran-2-carboxamide
{[2-(1H-1,3-benzodiazol-1-yl)pyridin-3-yl]methyl}(2,3-dihydro-1-benzofuran-5-ylmethyl)amine
1-(4-{[4-(1-butyl-1H-imidazol-2-yl)piperidin-1-yl]methyl}thiophen-2-yl)ethan-1-one
3-{[2-(4-chloro-1-methyl-1H-indazol-3-yl)-1H-imidazol-1-yl]methyl}-1λ6-thiolane-1,1-dione
1-[2-methoxy-5-({[(5-methylthiophen-2-yl)methyl]amino}methyl)phenoxy]-3-[methyl(propan-2-yl)amino]propan-2-ol
4-[5-(hydroxymethyl)furan-2-carbonyl]-3-methyl-1-(2-methylpropyl)piperazin-2-one
(1S,5R)-3-[(1-methyl-1H-imidazol-4-yl)sulfonyl]-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
2-cyclopropyl-N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-4-methylpyrimidine-5-carboxamide
2,6-dimethyl-4-[2-(4-methyl-1,2,5-oxadiazol-3-yl)pyrrolidine-1-carbonyl]quinoline
2-methoxy-N-{1-[4-(1H-1,2,4-triazol-1-yl)phenyl]ethyl}-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
1-{4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-1-yl}-3-(3-hydroxy-1,2-oxazol-5-yl)propan-1-one