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N3-(3-methylbutyl)-1-(2-methylpropyl)-N5-[(6-methylpyridin-2-yl)methyl]-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
3-[5-(2,3-dihydro-1H-inden-2-yl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]-N-(2-hydroxyethyl)propanamide
5-methyl-1-[3-(morpholin-4-yl)propyl]-5-phenylpiperidin-2-one
1-(6,7-dimethoxy-1,2,3,4-tetrahydroisoquinolin-2-yl)-2-[5-(pyrrolidin-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]ethan-1-one
1-(4-{[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]amino}-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl)ethan-1-one
5-hydroxy-N-[(4-methoxypyridin-2-yl)methyl]pyrazine-2-carboxamide
1-cyclopropanecarbonyl-N-(2-hydroxyethyl)-N-[(1-methyl-1H-imidazol-2-yl)methyl]piperidine-4-carboxamide
1-[2-({5-phenyl-5H,6H,7H-pyrrolo[3,2-d]pyrimidin-2-yl}amino)ethyl]pyrrolidine-2,5-dione
2-(5-amino-1H-1,2,3,4-tetrazol-1-yl)-N-[3-(2-phenylacetamido)phenyl]acetamide
1-benzoyl-4-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)piperazine
N-{1-[4-(2-chlorophenoxy)piperidin-1-yl]-1-oxopentan-2-yl}acetamide
8-[3-methyl-5-({[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]sulfanyl}methyl)-1H-1,2,4-triazol-1-yl]quinoline
3-tert-butyl-5-(4-methanesulfonylphenyl)-1-methyl-1H,4H-pyrazolo[3,4-d]imidazole
2-{4-[(3,4-difluorophenyl)methyl]-1-[1-(propan-2-yl)piperidin-4-yl]piperazin-2-yl}ethan-1-ol
2-methyl-N-{1-[1-(3-methylbut-2-enoyl)piperidin-4-yl]-1H-pyrazol-5-yl}benzamide
[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl][(6-methoxypyridin-3-yl)methyl]methylamine
4-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-N,N,6-trimethylpyrimidin-2-amine
4-(2,2-dimethyloxane-4-carbonyl)-9-methoxy-7-(6-methoxypyridazin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-{7-[2-hydroxy-4-(1H-pyrazol-1-yl)butan-2-yl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl}-2-[3-(trifluoromethyl)phenyl]ethan-1-one
N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-3-(2-methyl-1H-1,3-benzodiazol-1-yl)propanamide
N-(cyclopropylmethyl)-5-methyl-4-[(prop-2-en-1-yl)amino]thieno[2,3-d]pyrimidine-6-carboxamide
1-[3-(furan-2-yl)propanoyl]-N-[4-(1H-pyrazol-1-yl)phenyl]pyrrolidine-2-carboxamide
8-[(1-cyclopentyl-1H-imidazol-5-yl)methyl]-2-(cyclopropylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
4-(1H-1,2,3,4-tetrazol-1-yl)-N-{[2-(1H-1,2,4-triazol-1-yl)phenyl]methyl}benzamide
5-methanesulfonyl-2-methyl-4-{4-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}pyrimidine
4-[(4-phenyl-4H-1,2,4-triazol-3-yl)methyl]-1-{[5-(1H-pyrazol-5-yl)furan-2-yl]methyl}piperidine
2-[(2,6-dichlorophenyl)methyl]-5-(2-phenylazetidine-1-carbonyl)pyrimidin-4-ol
(3S,4R)-4-(hydroxymethyl)-1-(3-methyl-1-propyl-1H-pyrazole-4-carbonyl)piperidin-3-ol
1-(2-{2-[2-(4-hydroxyphenyl)ethyl]piperidin-1-yl}-2-oxoethyl)-1,2,3,6-tetrahydropyridazine-3,6-dione
N-ethyl-3,5,7-trimethyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-1H-indole-2-carboxamide
(3S,4R)-1-(2,5-dimethylbenzoyl)-4-(3-methoxyphenyl)pyrrolidine-3-carboxylic acid
2-(2-aminoethyl)-N-[1-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)ethyl]quinazolin-4-amine
4-[(3-methylphenyl)sulfanyl]-1-{5H,6H,7H,8H,9H-[1,2,3,4]tetrazolo[1,5-a]azepine-9-carbonyl}piperidine
(4aS,8aS)-2-cyclobutanecarbonyl-7-(1,2,5-trimethyl-1H-pyrrole-3-carbonyl)-decahydro-2,7-naphthyridin-4a-ol
N-(1-{3-fluoro-6-methylimidazo[1,2-a]pyridine-2-carbonyl}piperidin-4-yl)methanesulfonamide
N-[(3R,4S)-1-(1-acetylpiperidin-4-yl)-4-(propan-2-yl)pyrrolidin-3-yl]propane-1-sulfonamide
methyl N-{2-oxo-2-[2-oxo-3-(2-phenylethyl)-1-oxa-3,8-diazaspiro[4.5]decan-8-yl]ethyl}carbamate
1-(pyridin-2-ylmethyl)-5-{4H,5H,6H,7H-thieno[3,2-c]pyridine-5-carbonyl}piperidin-2-one
N-[2-hydroxy-2-(pyridin-3-yl)ethyl]-2-(2,4,7-trimethyl-1H-indol-3-yl)acetamide
1-(2H-1,3-benzodioxol-5-yl)-N-(2-ethylphenyl)-3-methyl-1H-1,2,4-triazole-5-carboxamide
3-[2-(2-fluorophenyl)ethyl]-1-[5-(1H-imidazol-1-ylmethyl)furan-2-carbonyl]piperidine
N-(2,1,3-benzoxadiazol-5-ylmethyl)-2-(2,5-dioxoimidazolidin-1-yl)acetamide
7-fluoro-3-methyl-N-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}-1-benzofuran-2-carboxamide
N-cyclobutyl-3-[(1H-pyrazol-3-ylmethyl)sulfamoyl]benzamide
N-methyl-2-(methylamino)-N-[1-(pyridin-3-yl)propyl]pyridine-3-carboxamide
2-[2-(2-fluorophenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-1-[2-(pyridin-2-yl)piperidin-1-yl]ethan-1-one
2-(2-methylpyrrolidine-1-carbonyl)-N-(prop-2-en-1-yl)aniline
3-{[7-(1-benzofuran-2-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]methyl}pyridine
2-(3-hydroxypropyl)-9-{[2-(methoxymethyl)pyrimidin-5-yl]methyl}-2,9-diazaspiro[5.5]undecan-3-one
1-[5-(methoxymethyl)furan-2-carbonyl]-4-[4-methyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine