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5-(1H-imidazol-1-ylmethyl)-N-methyl-N-[(1-phenyl-1H-pyrazol-4-yl)methyl]furan-2-carboxamide
[(5-{1-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]piperidin-3-yl}-4-methyl-4H-1,2,4-triazol-3-yl)methyl]dimethylamine
4-({4-[4-(methoxymethyl)-6-oxo-1,6-dihydropyrimidin-2-yl]phenyl}methyl)-N,N-dimethylpiperazine-1-carboxamide
N-methyl-N-[1-(pyridin-3-yl)pentyl]-6-(4H-1,2,4-triazol-4-yl)pyridine-3-carboxamide
5-(4-fluoro-2-methoxyphenyl)-1-(2-methanesulfonylethyl)-4-phenyl-1H-imidazole
2-butyl-N-(4-ethoxy-2-fluorophenyl)-4-methyl-3-oxopiperazine-1-carboxamide
(2S)-N1-[2-(propan-2-ylsulfanyl)phenyl]pyrrolidine-1,2-dicarboxamide
3-[2-(dimethylamino)ethyl]-3-ethyl-1-(2-methoxy-5-phenylphenyl)urea
N-[2-(5-methylfuran-2-yl)-2-(morpholin-4-yl)ethyl]-5,6,7,8-tetrahydroquinoline-3-carboxamide
N-{2-[2-(6-methoxynaphthalen-2-yl)morpholin-4-yl]-2-oxoethyl}acetamide
N,3,5-trimethyl-N-[1-(1,3-thiazol-2-yl)ethyl]-1H-indole-2-carboxamide
(1-{2-[(thian-4-yl)amino]ethyl}piperidin-2-yl)methanol
{[3-(1-benzofuran-2-yl)-1-benzyl-1H-pyrazol-4-yl]methyl}(methyl)[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]amine
3-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-[5-({[(4-ethylphenyl)methyl](methyl)amino}methyl)-2-methoxyphenoxy]-3-(4-methylpiperazin-1-yl)propan-2-ol
3-[4-(dimethylamino)-2-methyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]-1,2-dimethyl-1H-indol-5-ol
2-{3-methyl-5-[(4-methyl-1,4-diazepan-1-yl)methyl]-1H-1,2,4-triazol-1-yl}-1-propyl-1H-1,3-benzodiazole
4-{5-benzyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carbonyl}-1-methylpiperazin-2-one
4-[(3aS,6aS)-3a-(hydroxymethyl)-octahydrocyclopenta[c]pyrrole-2-carbonyl]-1,2-dihydroquinolin-2-one
4-[({[(2-fluoro-5-methylphenyl)carbamoyl]methyl}amino)methyl]-N-methylbenzamide
2,6-dimethyl-N-[2-(N-methylmethanesulfonamido)ethyl]quinoline-3-carboxamide
2-cyclopropyl-N-(2-methoxy-5-methylphenyl)-3-oxo-2,9-diazaspiro[5.5]undecane-9-carboxamide
4-{[2-(3,4-dimethoxyphenyl)ethyl]amino}-N-(furan-2-ylmethyl)-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
2-[(2-chloro-5-acetamidophenyl)formamido]-N-(4-fluoro-2-methylphenyl)propanamide
N-[3-(1-methyl-1H-1,3-benzodiazol-2-yl)propyl]-4-(trifluoromethyl)pyrimidin-2-amine
(3aS,6aS)-2-[(5-chlorofuran-2-yl)methyl]-5-cyclobutanecarbonyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N,1,4,6-tetramethyl-N-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]-2-oxo-1,2-dihydropyridine-3-carboxamide
2-chloro-N-{1-[1-(3-fluoropropyl)piperidin-4-yl]-1H-pyrazol-5-yl}benzamide
cyclopentyl 4-({[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]carbamoyl}amino)benzoate
1-{4-[(6-chloropyridin-3-yl)methyl]piperazin-1-yl}-2-(2-methyl-1,3-thiazol-4-yl)ethan-1-one
2-[1-(2,3-dihydro-1H-inden-2-yl)-5-(2-methyl-1,3-benzoxazol-6-yl)-1H-1,2,4-triazol-3-yl]acetamide
N-(1,1-dioxo-1λ6-thiolan-3-yl)-N-ethyl-5-[(4-methylpiperidin-1-yl)methyl]furan-2-carboxamide
2-(1H-pyrazol-1-yl)-N-{pyrazolo[1,5-a]pyridin-3-ylmethyl}butanamide
N-{[1-(4-methylphenyl)pyrrolidin-3-yl]methyl}pyrimidin-2-amine
7-{2-[4-(1H-1,2,3,4-tetrazol-1-yl)phenoxy]acetyl}-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3-carboxamide
2-{2-[4-methyl-3-oxo-2-(propan-2-yl)piperazin-1-yl]-2-oxoethyl}-5-(piperidin-1-yl)-2,3-dihydropyridazin-3-one
1-[2-(4-methoxyphenyl)ethyl]-8-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-3-(propan-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-methyl-5-[6-(4H-1,2,4-triazol-4-yl)pyridine-2-carbonyl]-4H,5H,6H,7H-thieno[3,2-c]pyridine-2-carboxamide
2-[(4-phenyl-1,3-thiazol-2-yl)methyl]-4-[4-(quinolin-4-ylmethyl)piperazin-1-yl]-2,3-dihydro-1H-isoindole-1,3-dione
5-{[3-(3-methoxyphenoxy)azetidin-1-yl]methyl}-2-(thiophen-2-yl)pyrimidine
(2R,3R,6R)-5-(3-methoxybenzoyl)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
2-(1-{2-[methyl(pyridin-4-ylmethyl)amino]acetyl}pyrrolidin-3-yl)benzoic acid
1-[(4-{[3-(2-methoxyphenoxy)azetidin-1-yl]methyl}phenyl)methyl]-1H-pyrazole
ethyl 2,4-dimethyl-5-{1-methyl-5-oxo-1,4,9-triazaspiro[5.5]undecane-9-carbonyl}-1H-pyrrole-3-carboxylate
4-hydroxy-3-{pyrazolo[1,5-a]pyridin-7-yl}benzonitrile
4-chloro-2-[1-(piperidin-4-yl)-1H-1,2,3-triazol-4-yl]-6-(trifluoromethyl)-1H-1,3-benzodiazole
7-[3-(pyridin-4-yl)propyl]-2-oxa-7-azaspiro[4.5]decan-8-one
N-[(4-methyl-2-propyl-1,3-thiazol-5-yl)methyl]-3-(1-methylpiperidin-2-yl)propanamide
[2-(6-{[(5-methyl-1,2-oxazol-3-yl)methyl]sulfamoyl}-1,2,3,4-tetrahydroisoquinolin-2-yl)-2-oxoethyl]urea
5-[4-(4-methoxyphenyl)butanoyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid