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2-(1H-indol-1-yl)-N-methyl-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}acetamide
2-[2-(3-hydroxyphenyl)phenoxy]propanamide
2-(4-methoxyphenyl)-N-[(5-methylthiophen-2-yl)methyl]acetamide
3-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]-1-{[4-(methylsulfanyl)phenyl]methyl}piperidine
N-[1-(2-fluorophenyl)piperidin-4-yl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
N-{imidazo[1,2-a]pyrazin-3-ylmethyl}-1H-indazole-3-carboxamide
1-[3-(2-methoxyethoxy)phenyl]-3-{2-[(2R)-pyrrolidin-2-yl]ethyl}urea
2-amino-6-(3,5-dimethylphenyl)-4-(1H-imidazol-4-yl)-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
2-(3,5-dimethyl-1H-pyrazol-1-yl)-N-({7-[2-(trifluoromethyl)phenyl]-2,3-dihydro-1-benzofuran-2-yl}methyl)acetamide
1-[1-(1,3-dimethyl-1H-pyrazole-5-carbonyl)piperidin-3-yl]-4-(2-fluorophenyl)piperazine
3-({6-methyl-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-yl}amino)-1-(pyrrolidin-1-yl)propan-1-one
N-(4-{thieno[2,3-d]pyrimidin-4-yl}-1H-pyrrolo[2,3-b]pyridin-6-yl)piperidin-4-amine
5-[(4-methylpiperazin-1-yl)methyl]-N-(1-phenylbutyl)furan-2-carboxamide
2-{1-[(2-chloro-6-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-(2-methoxyethyl)-N-methylacetamide
2-[2-(propan-2-yl)pyrimidin-4-yl]pyridine-4-carboxylic acid
3-(3-phenyl-1,2,4-oxadiazol-5-yl)-1-[3-(pyridin-3-yl)azetidin-1-yl]propan-1-one
6-{[(3R)-3-hydroxypyrrolidin-1-yl]methyl}-2-oxo-N-(quinolin-3-ylmethyl)-1,2-dihydropyridine-3-carboxamide
1-{3-[6-(hydroxymethyl)-1,4-oxazepan-4-yl]-3-oxopropyl}-2,3-dihydro-1H-1,3-benzodiazol-2-one
4-{2-[2-(2-methoxyphenyl)pyrrolidin-1-yl]-2-oxoethyl}-2H,3H,4H-pyrido[3,2-b][1,4]oxazin-3-one
N-ethyl-N'-(5-methyl-1,2-oxazol-3-yl)-N-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}ethanediamide
5-[2-(2-hydroxyphenyl)-6-methylpyrimidin-4-yl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
5-[4-(pyrrolidine-1-sulfonyl)phenyl]pyrazin-2-amine
N-cyclopropyl-3-{1-[(4,5-dimethylfuran-2-yl)methyl]piperidin-3-yl}propanamide
4,6-dimethyl-1-(3-oxo-3-{4-[(pyrimidin-2-yl)amino]piperidin-1-yl}propyl)-1,2-dihydropyrimidin-2-one
8-{[2-(cyclopentyloxy)phenyl]methyl}-1,3-dioxa-8-azaspiro[4.5]decan-2-one
methyl 1-({4-[(2E)-2-methylbut-2-en-1-yl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}methyl)piperidine-2-carboxylate
6-[(4-hydroxy-1,2,3,4-tetrahydroisoquinolin-2-yl)methyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-[2-(dimethylamino)ethyl]-9-[(5-hydroxy-2-methoxyphenyl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
3-(2-{3-[2-(dimethylamino)ethyl]-2-oxo-1-oxa-3,8-diazaspiro[4.5]decan-8-yl}-2-oxoethyl)imidazolidine-2,4-dione
9-[2-(4-fluorophenyl)acetyl]-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
1'-(1H-1,2,3-benzotriazole-5-carbonyl)-5-methyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
4-{2-[(4-fluorophenyl)methyl]-3H-imidazo[4,5-b]pyridin-3-yl}-1-(5-phenoxyfuran-2-carbonyl)piperidine
1-[1'-(3-ethyl-1H-pyrazole-5-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]propan-1-one
2-[1-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-methyl-1H-1,2,4-triazol-5-yl]-3-methylpyridine
1-(4-benzylpiperazin-1-yl)-3-[1-(3-ethyl-1-methyl-1H-pyrazole-5-carbonyl)piperidin-3-yl]propan-1-one
3-({4-[(3S,4R)-4-hydroxyoxolan-3-yl]-1,4-diazepan-1-yl}methyl)benzonitrile
3,3,3-trifluoro-N-{1-[2-(4-methoxyphenyl)ethyl]-5-oxopyrrolidin-3-yl}propanamide
1-(4-chloro-2-hydroxybenzoyl)-3-ethylpiperidine-3-carboxylic acid
2-(methylamino)-1-[4-(2-methylpyridin-4-yl)-1,4-diazepan-1-yl]-2-phenylethan-1-one
3,6-dimethyl-N-[2-(piperidin-1-yl)-2-(pyridin-3-yl)ethyl]-[1,2]oxazolo[5,4-d]pyrimidin-4-amine
4-[(1S,2R)-2-({5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)-1-hydroxypropyl]phenol
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
N-({3-[1-(dimethylamino)ethyl]phenyl}methyl)-N-(pyridin-3-ylmethyl)cyclopropanamine
N-[1-benzyl-4-(propan-2-yloxy)-1H-indazol-3-yl]-1,2-oxazole-3-carboxamide
2-(methylsulfanyl)-1-{4-[(2-phenylethyl)amino]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl}ethan-1-one
2-[1-(2-chlorophenyl)-5-oxo-3-phenyl-4,5-dihydro-1H-1,2,4-triazol-4-yl]-N-(cyclopropylmethyl)acetamide
N-({5-acetyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)quinoxaline-5-carboxamide
N-(1-methyl-4-phenyl-1H-pyrazol-5-yl)-2-{1H-pyrazolo[3,4-b]pyridin-1-yl}acetamide
1-(4-fluorophenyl)-4-{1-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]piperidin-3-yl}piperazine
(1R,2R,6S,7S)-4-(5-methanesulfonyl-2-methylpyrimidin-4-yl)-10-oxa-4-azatricyclo[5.2.1.02,6]decane