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N-{1-[3-(5-methylfuran-2-yl)-1H-pyrazole-5-carbonyl]piperidin-4-yl}pyrimidin-2-amine
methyl(pyridin-3-ylmethyl){[5-(pyrrolidine-1-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}amine
({3-[(3-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)[1-(3-methoxyphenyl)ethyl]methylamine
2-[1-(2,2-dimethylpropyl)-3-oxopiperazin-2-yl]-N-[(3-methylpyridin-4-yl)methyl]acetamide
(1S,5R)-6-benzyl-3-[3-(2-methyl-1H-imidazol-1-yl)propyl]-3,6-diazabicyclo[3.2.2]nonane
1-[(3,4-dichlorophenyl)methyl]-4-(pyridin-4-ylmethyl)-1,4-diazepane
3-{5-benzyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-N-cyclopentylpropanamide
N-[2-(ethanesulfonyl)ethyl]-2-(1H-imidazol-2-yl)benzamide
[3-ethyl-1-(4-methoxybenzenesulfonyl)piperidin-3-yl]methanol
N-methyl-N-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}imidazo[1,2-a]pyrimidine-2-carboxamide
3-(2-methoxyphenoxy)-1-{5-[(methylsulfanyl)methyl]furan-2-carbonyl}azetidine
5-{[1-benzyl-3-(oxolan-3-yl)-1H-1,2,4-triazol-5-yl]methyl}-2,6-dimethyl-3,4-dihydropyrimidin-4-one
(1S,4S)-2-[5-(3-benzyl-1,2,4-oxadiazol-5-yl)pyridin-2-yl]-2-azabicyclo[2.2.1]heptane
1-[(1-benzyl-3-cyclopentyl-1H-1,2,4-triazol-5-yl)methyl]-4,6-dimethyl-1,2-dihydropyrimidin-2-one
N4-[(4-phenyloxan-4-yl)methyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
3-(1H-1,2,3-benzotriazol-1-yl)-1-[3-(2-fluorophenyl)pyrrolidin-1-yl]propan-1-one
(2R,6S)-4-{5-[(2H-1,3-benzodioxol-5-yloxy)methyl]-1H-pyrazole-3-carbonyl}-2,6-dimethylmorpholine
4-(4-{imidazo[1,2-b]pyridazine-3-carbonyl}piperazin-1-yl)quinazoline
(2S)-2-{4-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyrrolidine-1-carboxamide
2-amino-N-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-4-ethyl-N-methyl-1,3-thiazole-5-carboxamide
3-chloro-N-{1-[5-(ethylsulfanyl)-4-methyl-4H-1,2,4-triazol-3-yl]ethyl}benzamide
(1s,4s)-4-[4-(2-chlorophenoxy)piperidine-1-carbonyl]cyclohexan-1-ol
5-(4-benzylpiperidine-1-carbonyl)-N-methyl-N-(2-methylpropyl)-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3-carboxamide
2-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-7-propyl-2,7-diazaspiro[4.5]decan-6-one
1-(oxan-2-ylmethyl)-2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazole
N-(prop-2-en-1-yl)-2-[(quinolin-8-yloxy)methyl]-1,3-oxazole-4-carboxamide
5-(2-chlorophenyl)-N-{[4-(dimethylamino)oxan-4-yl]methyl}furan-2-carboxamide
4-[3-(propan-2-yl)-1H-pyrazol-1-yl]-1-(quinoxalin-2-yl)piperidine-4-carboxylic acid
8-(5,6-dimethylpyrimidin-4-yl)-2-(3-methylbutyl)-2,8-diazaspiro[5.5]undecan-3-one
3-[(1S,5R)-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-4,5,6,7-tetrahydro-1,2-benzoxazole
2-(1H-imidazol-1-yl)-N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]acetamide
1-[(3-hydroxypiperidin-3-yl)methyl]-3-[3-(4-methylpiperazine-1-carbonyl)phenyl]urea
9-ethyl-4-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
1-butyl-4-[5-oxo-1-(pyridin-2-ylmethyl)pyrrolidine-3-carbonyl]piperazin-2-one
2,5,7-trimethyl-N-[(1r,4r)-4-(4H-1,2,4-triazol-4-yl)cyclohexyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
1-[(4-chlorophenyl)methyl]-5-(1-propoxyethyl)-1H-1,2,4-triazole
(4aR,8aR)-2-cyclobutanecarbonyl-7-[(2,4-dimethylphenyl)methyl]-decahydro-2,7-naphthyridin-4a-ol
4-[3-(2-amino-1,3-thiazol-4-yl)propanoyl]-1-(3,5-dimethylphenyl)piperazin-2-one
4-(2-hydroxyethyl)-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
5-(azocane-1-carbonyl)-1-methyl-1H-1,3-benzodiazole
(1S,2S,4R)-4-(3-benzyl-1H-1,2,4-triazol-5-yl)-1,7,7-trimethylbicyclo[2.2.1]heptan-2-ol
9-[(2S)-2,4-diaminobutanoyl]-2-[2-(pyridin-3-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
1-(1,4-dithiepan-6-yl)-N-[4-(3-methylphenyl)phenyl]piperidine-4-carboxamide
4-{4-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]phenyl}piperidin-4-ol
3-[4-(dimethylamino)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]-6-methoxy-1,4-dihydroquinolin-4-one
1-{2-[3-(4,5-dimethyl-1H-pyrazol-3-yl)propanamido]ethyl}piperidine-3-carboxamide
5-{4-[1-(morpholin-4-yl)ethyl]piperidine-1-carbonyl}-1H-1,2,3-benzotriazole
4-[(4-fluorophenyl)methyl]-1-(2-hydroxyethyl)-3-(propan-2-yl)-1,4-diazepan-5-one
N-(1-{7-[(4-methoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-3-methylbutyl)pyridine-3-carboxamide
2-(2,4-dimethoxyphenyl)-1-[3-ethyl-3-(hydroxymethyl)piperidin-1-yl]ethan-1-one