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N-[(4-methanesulfonylmorpholin-2-yl)methyl]-2-(propan-2-yl)pyrimidine-5-carboxamide
3-[(3S,4R)-3-benzyl-4-hydroxy-4-methylpiperidine-1-carbonyl]-1,4,6-trimethyl-1,2-dihydropyridin-2-one
1-methyl-4-(2-methyl-1,2,3,4-tetrahydroisoquinoline-3-carbonyl)-1,4,9-triazaspiro[5.5]undecane
4-[4-(2,6-dimethylpyridin-4-yl)piperazine-1-carbonyl]-1-ethylpyrrolidin-2-one
N-ethyl-N-[1-(5-ethyl-2-methylpyrimidin-4-yl)pyrrolidin-3-yl]acetamide
N-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-1-[3-(pyridin-4-yl)propanoyl]piperidine-4-carboxamide
N,7-dimethyl-N-(1,2-oxazol-3-ylmethyl)-2-[1-(propan-2-yl)-1H-pyrazol-4-yl]quinoline-4-carboxamide
6-cyano-N-methyl-N-(quinolin-5-ylmethyl)pyridine-3-carboxamide
2-{6-[(pyridin-2-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}-1,3-thiazole-4-carboxamide
2-(4-{4-methyl-5-[(4-methylpiperazin-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)pyridine-3-carbonitrile
2-chloro-6-methoxy-4-(1-{[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}-1H-imidazol-2-yl)phenol
(3R,9aR)-8-(naphthalene-1-sulfonyl)-3-(propan-2-yl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
2-methyl-2-{2-[methyl(oxan-2-ylmethyl)amino]-4-(morpholin-4-yl)pyrimidin-5-yl}propanoic acid
3-amino-N-[2-(morpholin-4-yl)butyl]-1H-1,2,4-triazole-5-carboxamide
N-[(1S,3aS,6aS)-octahydropentalen-1-yl]-1-(pyrrolidin-1-yl)cyclopentane-1-carboxamide
3-(methoxymethyl)-5-{2-[2-(3-methylthiophen-2-yl)-1H-imidazol-1-yl]ethyl}-1,2,4-oxadiazole
1-cyclohexyl-N-{2-[(4-methylpyridin-2-yl)amino]ethyl}piperidine-4-carboxamide
4-{[1-(2,3-dihydro-1H-inden-2-yl)-5-oxopyrrolidin-3-yl]amino}-2-methoxypyridine-3-carbonitrile
methyl 3-[(furan-3-ylformamido)methyl]-5-[3-(trifluoromethyl)benzenesulfonamido]benzoate
1-(1-{[4-(prop-2-en-1-yloxy)phenyl]methyl}piperidin-4-yl)pyrrolidin-2-one
2-{4-[6,8-dimethyl-4-(2-methylpiperidine-1-carbonyl)quinolin-2-yl]-1H-pyrazol-1-yl}ethan-1-ol
methyl (2S,4S,5R)-1,2-dimethyl-5-(2-methylphenyl)-4-{[(6-methylpyridin-2-yl)methyl]carbamoyl}pyrrolidine-2-carboxylate
5-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}-3-methyl-1,2-benzoxazole
N-[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl]-2-phenylimidazo[1,2-a]pyridine-6-carboxamide
3-[1-(1-benzoylpiperidin-4-yl)-1H-pyrazol-5-yl]-1-(2-methoxyphenyl)urea
N-[(3-methylpyridin-2-yl)methyl]-2-(phenylamino)-N-(propan-2-yl)pyrimidine-5-carboxamide
(3S)-1-{1-methyl-5-[(2R)-2-methylpiperazine-1-carbonyl]-1H-1,3-benzodiazol-2-yl}pyrrolidin-3-ol
1-[1-(methoxymethyl)cyclobutanecarbonyl]-3-[4-(4-methylphenyl)-1H-pyrazol-5-yl]piperidine
N-[2-(dimethylamino)ethyl]-2-[methyl(2-phenylethyl)amino]-2,3-dihydro-1H-indene-2-carboxamide
5-methyl-N-(quinolin-2-ylmethyl)pyrazolo[1,5-a]pyrimidin-7-amine
2-[3-cyclopropyl-5-(2-methoxypyridin-4-yl)-1H-1,2,4-triazol-1-yl]ethan-1-ol
N-[1-(4-chlorophenyl)-3-hydroxypropan-2-yl]-4,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
4-[1-(3-methylbut-2-en-1-yl)piperidin-4-yl]pyridine
[(3R,4S)-1-[(2,3-dichlorophenyl)methyl]-4-[(4-ethylpiperazin-1-yl)methyl]pyrrolidin-3-yl]methanol
N-[(1S)-3-(methylsulfanyl)-1-[3-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]propyl]acetamide
N-[2-(2-methyl-1-phenyl-1H-indol-3-yl)ethyl]-2-(1-methyl-3-oxopiperazin-2-yl)acetamide
methyl 5-oxo-5-[3-(2-phenylethyl)piperidin-1-yl]pentanoate
1-(1-{[2-(prop-2-en-1-yloxy)phenyl]methyl}piperidin-3-yl)-N-(propan-2-yl)-1H-1,2,3-triazole-4-carboxamide
3-{[1-(hydroxymethyl)cyclopropyl]methyl}-3-methyl-1-[2-(2-methylphenyl)-1,3-benzoxazol-6-yl]urea
2-methyl-N-[3-(2-methyl-1H-imidazol-1-yl)-1-phenylpropyl]-6-oxo-1,6-dihydropyrimidine-5-carboxamide
6-ethyl-1-methyl-N-[4-(pyridin-2-yl)butyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-[(2-ethyl-4-methyl-1,3-thiazol-5-yl)methyl]-2-methyl-1-benzofuran-5-carboxamide
5-[3-(4-methoxyphenyl)-1H-pyrazol-5-yl]-3-[(methylsulfanyl)methyl]-1,2,4-oxadiazole
2-{2-[2-(5-methylfuran-2-yl)-1H-imidazol-1-yl]ethyl}-1H-1,3-benzodiazole
3-{[1-(1H-imidazole-5-carbonyl)piperidin-4-yl]methyl}-1-methyl-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
1-[1-(2-methoxy-3-methylbenzoyl)piperidin-4-yl]pyrrolidin-2-one
3-(2-methylphenyl)-5-[3-(propan-2-yl)-4,5-dihydro-1,2-oxazol-5-yl]-1,2,4-oxadiazole
1-(3-{[4-(hydroxymethyl)phenyl]methyl}pyrrolidin-1-yl)-2-(2-methylphenyl)ethan-1-one
N-(4-methoxy-3-propanamidophenyl)-4-(pyridin-4-yl)piperazine-1-carboxamide
3-chloro-5-[(4S)-4-hydroxy-4-(methoxymethyl)-3,3-dimethylpiperidine-1-carbonyl]-1,2-dihydropyridin-2-one