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N-{[2-(morpholin-4-yl)pyridin-3-yl]methyl}-2-(pyrimidin-2-ylsulfanyl)acetamide
ethyl 4-(oxan-2-ylmethyl)-1-[3-(prop-2-en-1-yloxy)benzoyl]piperidine-4-carboxylate
2-methyl-6-{1-[3-(5-methylfuran-2-yl)butyl]piperidin-4-yl}pyrimidin-4-ol
5-[(2S)-2-(methoxymethyl)pyrrolidine-1-carbonyl]-3-(3-methoxyphenyl)-1H-pyrazole
3-(5-methyl-1H-1,2,4-triazol-3-yl)-N-[(3R,4S)-1-(oxan-4-yl)-4-propylpyrrolidin-3-yl]propanamide
1-(cyclopropylmethyl)-4-[(2-ethylpyrimidin-5-yl)methyl]-2-(propan-2-yl)-1,4-diazepane
N-[1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]-3-(pyrrolidin-1-yl)propanamide
1-[2-(4-methanesulfonylphenyl)ethyl]-1H-imidazole
2-(2,4-difluorophenyl)-1-{2-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl}ethan-1-one
7-[(2-ethylphenyl)methyl]-2-(furan-2-carbonyl)-2,7-diazaspiro[4.5]decane
5-(5-methyl-3-phenyl-1,2-oxazol-4-yl)-3-(oxolan-3-yl)-1,2,4-oxadiazole
2-[(5-fluoro-1H-1,3-benzodiazol-2-yl)methoxy]-1-{2-oxa-7-azaspiro[4.5]decan-7-yl}ethan-1-one
3-methoxy-5-{thieno[3,2-d]pyrimidin-4-yl}pyridine
1-[(2R,3R,6R)-3-(3-hydroxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]cyclopropane-1-carboxamide
3-methyl-N-[2-(6-oxo-3-phenyl-1,6-dihydropyridazin-1-yl)ethyl]-1-propyl-1H-pyrazole-4-carboxamide
6-(2-chlorophenyl)-N-ethyl-N-methyl-8-oxo-7-(prop-2-en-1-yl)-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
(4aS,8aR)-1-(2-aminoethyl)-6-(1,8-naphthyridine-2-carbonyl)-decahydro-1,6-naphthyridin-2-one
3-[(3S,4S)-4-ethoxy-1-methylpyrrolidin-3-yl]-1-[2-(3-methoxyphenyl)phenyl]urea
methyl[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]{[3-(3-methylphenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}amine
N-methyl-2-{2-[(5-methylpyrazin-2-yl)methyl]-3-oxo-2,9-diazaspiro[5.5]undecan-9-yl}acetamide
1-(2-ethyl-6-methylphenyl)-N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-5-oxopyrrolidine-3-carboxamide
2-{3-[1-(pyrrolidin-1-yl)ethyl]phenyl}-4-(trifluoromethyl)pyrimidine
1-[(1-cyclohexyl-3-cyclopentyl-1H-1,2,4-triazol-5-yl)methyl]-5-methyl-1H-1,2,3,4-tetrazole
9-(2,8-dimethylquinoline-3-carbonyl)-1,4-dimethyl-1,4,9-triazaspiro[5.5]undecane
N-methyl-5-(propan-2-yl)-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}thiophene-3-carboxamide
(2S)-N2-ethyl-N1-[2-(3-methylphenoxy)phenyl]pyrrolidine-1,2-dicarboxamide
5-(2,6,8-trimethylquinoline-4-carbonyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-3-carboxamide
2-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}-N-methyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-amine
1-(3,5-dimethylphenyl)-4-{5-[(methylsulfanyl)methyl]furan-2-carbonyl}piperazin-2-one
N-[2-methoxy-1-(pyridin-2-yl)ethyl]-6-methyl-2-(piperidin-1-yl)pyrimidin-4-amine
N-[2-(5,7-difluoro-2-methyl-1H-indol-3-yl)ethyl]-6-methyl-4-oxo-4H-pyran-2-carboxamide
(2-{1H-pyrrolo[2,3-b]pyridin-4-yl}-1,3-thiazol-4-yl)methanol
2-methyl-4-(2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazol-1-yl)-2H-1,2,3-benzotriazole
1-(6-amino-2-{[(2-methylphenyl)methyl]sulfanyl}pyrimidin-4-yl)-3-(hydroxymethyl)piperidin-3-ol
N-[(1-hydroxycyclohexyl)methyl]-3-(2-methylpropyl)-1,2-oxazole-5-carboxamide
1-[(2-ethylpyrimidin-5-yl)methyl]-4-(2-methoxyphenoxy)piperidine-4-carboxylic acid
4-[({[2-(4-methoxyphenyl)-7-(methylsulfanyl)quinolin-3-yl]methyl}amino)methyl]benzene-1-sulfonamide
(1S,6R)-9-[1-(3-methoxyphenyl)piperidin-4-yl]-3,9-diazabicyclo[4.2.1]nonan-4-one
2-methyl-6-[3-(propan-2-yl)-1-(quinolin-8-yl)-1H-1,2,4-triazol-5-yl]-2,3,4,5-tetrahydropyridazin-3-one
N-(3-methoxypropyl)-5-methyl-6-(pyrrolidine-1-carbonyl)thieno[2,3-d]pyrimidin-4-amine
N,2,6-trimethyl-N-{[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]methyl}quinoline-3-carboxamide
N-cyclopropyl-N-ethyl-4-{[(3-methylthiophen-2-yl)methyl]amino}benzamide
N-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-2,6-dimethoxypyrimidine-4-carboxamide
5-(1-cyclopentyl-4-hydroxypiperidin-4-yl)-N-(oxolan-2-ylmethyl)-1-benzofuran-2-carboxamide
4-{3-[3-(methoxymethyl)pyrrolidine-1-carbonyl]phenoxy}-1-(1-methylpiperidin-4-yl)piperidine
N-[1-(2,2-dimethylpropyl)-5-oxopyrrolidin-3-yl]-3-ethyl-4-methyl-1H-pyrazole-5-carboxamide
2-[2-(3-benzyl-1,2,4-oxadiazol-5-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
3-{1-[(dimethyl-1,2-oxazol-4-yl)methyl]piperidin-3-yl}benzoic acid
N-(2-{imidazo[1,2-a]pyridin-2-yl}ethyl)-5-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]pyridin-2-amine
{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}({[3-(2-methylpropyl)-1,2-oxazol-5-yl]methyl})amine