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2-cyclopropyl-5-[4-(2-methylphenyl)-1,4-diazepane-1-carbonyl]-3,4-dihydropyrimidin-4-one
6-(5-propyl-1,3,4-oxadiazole-2-carbonyl)-1H,2H,3H,4H,5H,6H,7H,8H-pyrazolo[3,4-d]azepin-3-one
3-(methoxymethyl)-1-{[3-(3-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}piperidine
(3S,5R)-5-[(pyridin-2-ylmethyl)carbamoyl]-1-(3,3,3-trifluoropropyl)piperidine-3-carboxylic acid
N-[(3R,4S)-1-(carbamoylmethyl)-4-(propan-2-yl)pyrrolidin-3-yl]-2-(1,1-dioxo-1λ6-thian-4-yl)acetamide
4,4,4-trifluoro-N-[1-(pyridin-3-yl)propan-2-yl]butanamide
4-[3-(2,5-dimethylphenyl)-1H-pyrazol-4-yl]-6-oxo-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridine-3-carboxylic acid
N-[2-(dimethylamino)ethyl]-N-ethyl-4-(morpholin-4-yl)pyridine-2-carboxamide
3-[(2R,3S,6R)-3-(3,5-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]propanamide
3-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]-1-{3-fluoroimidazo[1,2-a]pyridine-2-carbonyl}piperidine
N-methyl-1-(2-phenylethyl)-5-[(pyridin-4-ylmethyl)amino]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
[(1-tert-butyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl](methyl)[1-(4-methylpyridin-2-yl)propan-2-yl]amine
4-(1-butyl-1H-imidazol-2-yl)-1-{[4-(1H-pyrazol-1-yl)phenyl]methyl}piperidine
1-cyclohexyl-N-[(2,2-dimethyl-2,3-dihydro-1-benzofuran-5-yl)methyl]-1H-1,2,3-triazole-4-carboxamide
2-(2-ethoxyphenyl)-2-[4-(thiomorpholin-4-yl)piperidin-1-yl]acetic acid
1-[3-({4-[(2-fluoro-4-methoxyphenyl)methyl]-3-(2-hydroxyethyl)piperazin-1-yl}methyl)phenyl]ethan-1-one
(2S,4R)-1-benzyl-N-ethyl-4-[2-(morpholin-4-yl)acetamido]pyrrolidine-2-carboxamide
(4-{[4-(benzyloxy)-3-methoxyphenyl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl)(pyridin-4-yl)methanol
8-(1,3-thiazol-2-ylmethyl)-8-azaspiro[4.5]decane-7,9-dione
N-{8-oxatricyclo[7.4.0.02,7]trideca-1(9),2,4,6-tetraen-6-yl}-2-oxo-1,3-dioxa-8-azaspiro[4.5]decane-8-carboxamide
(3S,5S,9S)-5-{[(2,5-dimethylphenyl)methyl]amino}-1,7-diazatricyclo[7.3.0.03,7]dodecane-2,8-dione
4-({2-[(benzenesulfonyl)methyl]phenyl}methyl)-2-(trifluoromethyl)morpholine
1-[4-(3-fluorophenyl)phenyl]-N-(piperidin-4-yl)piperidin-4-amine
4-[1-(cyclopent-3-en-1-yl)-4-phenyl-1H-imidazol-5-yl]-2,6-dimethoxyphenol
N-[(3-ethyl-1,2-oxazol-5-yl)methyl]-N-methyl-2-[2-(propan-2-yl)-1H-imidazol-1-yl]propanamide
5-ethyl-2-({4-[3-(propan-2-yl)-1H-pyrazol-5-yl]piperidin-1-yl}methyl)pyridine
N-({5-methanesulfonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-1,3-thiazole-4-carboxamide
N-methyl-N-{[3-(3-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl}-2-(pyridin-4-yl)pyrimidine-5-carboxamide
N-{[5,8-dimethoxy-2-(4-methylphenyl)quinolin-3-yl]methyl}-N-[2-(dimethylamino)ethyl]furan-3-carboxamide
N-{[2-(1H-1,3-benzodiazol-1-yl)pyridin-3-yl]methyl}-6-(methoxymethyl)pyrimidin-4-amine
1-[(2S)-2-{4-[(4-cyclopropyl-1H-1,2,3-triazol-1-yl)methyl]piperidine-1-carbonyl}pyrrolidin-1-yl]ethan-1-one
3-[(5-{3-[(4-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}pyridin-2-yl)amino]propan-1-ol
N-[1-(5-amino-1,3,4-thiadiazol-2-yl)ethyl]-3-phenyl-1H-pyrazole-4-carboxamide
3-{2-[3-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]ethyl}quinoxalin-2-ol
N-[(3S,4R)-1-[1-(3-methoxyphenyl)piperidin-4-yl]-4-(propan-2-yl)pyrrolidin-3-yl]acetamide
4-(3-methyl-1H-pyrazole-4-carbonyl)-2-(2-phenylethyl)morpholine
1-(4-{[4-(1H-pyrazol-1-yl)butan-2-yl]amino}-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl)ethan-1-one
4-cyclopropyl-1-[3-(2-methoxyphenoxy)propyl]-4-methylpyrrolidin-2-one
N-(1-{1-[(2-methyl-1,3-thiazol-5-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-2H-1,3-benzodioxole-5-carboxamide
N,N-bis(1,3-oxazol-4-ylmethyl)-2-(3-oxo-3,4-dihydro-2H-1,4-benzoxazin-4-yl)acetamide
7-[(3-methylphenyl)methyl]-2-(pyridin-3-ylmethyl)-2,7-diazaspiro[4.5]decan-6-one
N-(1-phenylethyl)-2-propanoyl-1,2,3,4-tetrahydroisoquinoline-6-sulfonamide
ethyl 4-({methyl[1-(2-phenylethyl)piperidin-3-yl]amino}methyl)-1H-pyrazole-3-carboxylate
3-methyl-5-(2-oxo-2-{6-oxo-7-propyl-2,7-diazaspiro[4.5]decan-2-yl}ethyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-methyl-4-(4-{1-[(5-methylpyrazin-2-yl)methyl]-1H-imidazol-2-yl}phenyl)but-3-yn-2-ol
4-methyl-N-{[4-(4-methylphenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}pyrimidine-5-carboxamide
4-(1H-1,3-benzodiazol-1-yl)-1-(4-methyl-1H-imidazole-5-carbonyl)piperidine-4-carboxylic acid
6,8-dimethyl-4-{[(oxolan-2-ylmethyl)(pyridin-2-ylmethyl)amino]methyl}-2H-chromen-2-one
1-[(2-fluoro-4,5-dimethoxyphenyl)methyl]-3-(piperidin-1-ylmethyl)pyrrolidin-3-ol
2-[3-(2-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-N-(pyridin-2-yl)propanamide