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3-[1-(2,5-dimethylfuran-3-carbonyl)piperidin-3-yl]-N-methyl-N-[2-(pyridin-2-yl)ethyl]propanamide
1-(cyclopropylmethyl)-4-[(5-methyl-2-phenyl-1H-imidazol-4-yl)methyl]piperazine
N-cyclopropyl-1,3-dimethyl-N-{[7-methyl-2-(3-methylphenyl)quinolin-3-yl]methyl}-1H-pyrazole-5-carboxamide
2-(4-{[3-(4-chlorophenyl)piperidin-1-yl]methyl}-3,5-dimethyl-1H-pyrazol-1-yl)ethan-1-ol
1-methyl-3-[2-(propylsulfanyl)phenyl]-1-[1-(pyrimidin-4-yl)ethyl]urea
{1-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]piperidin-4-yl}(thiophen-2-yl)methanol
4-[(4-chlorophenyl)methyl]-1-[6-(propan-2-yl)pyridazin-3-yl]piperidine-4-carboxylic acid
2-amino-4-ethyl-N-methyl-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-1,3-thiazole-5-carboxamide
(3R,4R)-3-methyl-4-(oxan-4-yl)-1-{[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}piperidin-4-ol
2-(1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}piperidin-2-yl)ethan-1-ol
N-[2-(1H-indol-1-yl)ethyl]-5-methanesulfonyl-N,2-dimethylpyrimidin-4-amine
4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-N-propyl-1,4-diazepane-1-carboxamide
(1S,5R)-6-(3-methylbut-2-en-1-yl)-3-{6-methylimidazo[1,2-a]pyridine-2-carbonyl}-3,6-diazabicyclo[3.2.2]nonan-7-one
N-(2,6-dimethylphenyl)-4-[(4-ethoxypiperidin-1-yl)methyl]benzamide
1-ethyl-3-(propan-2-yl)-N-{2-[4-(pyrimidin-2-yl)piperazin-1-yl]ethyl}-1H-pyrazole-5-carboxamide
butyl(furan-2-ylmethyl){[3-(pyrimidin-2-yloxy)phenyl]methyl}amine
2-{imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-4-{4-[2-(trifluoromethyl)benzoyl]piperazin-1-yl}-2,3-dihydro-1H-isoindole-1,3-dione
1-cyclopropyl-N-{[1-methyl-2-(methylsulfanyl)-1H-imidazol-5-yl]methyl}-5-oxopyrrolidine-3-carboxamide
N-(carbamoylmethyl)-N'-(3,5-dimethylphenyl)propanediamide
6-[(3S,4S)-3-hydroxy-4-(naphthalen-2-yl)piperidin-1-yl]-N,N-dimethylpyridine-3-carboxamide
N-cyclopentyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)-6-oxo-1,4,5,6-tetrahydropyridazine-3-carboxamide
(2E)-1-(4-{1-[methyl(pyridin-4-ylmethyl)amino]-2-phenylethyl}piperidin-1-yl)-3-phenylprop-2-en-1-one
7-chloro-3-({methyl[2-(1H-pyrazol-1-yl)ethyl]amino}methyl)-1-(pyridin-2-ylmethyl)-1,2-dihydroquinolin-2-one
4-[4-(1-ethyl-1H-imidazol-2-yl)piperidine-1-carbonyl]pyridine
1-methyl-4-[2-(pyrrolidin-1-ylmethyl)-1,3-thiazole-5-carbonyl]-1,4-diazepane
N-[2-(1H-imidazol-1-yl)ethyl]-5-oxo-1-(pyridin-2-ylmethyl)pyrrolidine-3-carboxamide
1-{[6-(3-chlorophenyl)pyridin-3-yl]methyl}-4-methylpiperazine
1-cyclohexyl-3-cyclopropyl-5-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-1H-1,2,4-triazole
N-(2,4-dimethylphenyl)-3-[5-(oxolan-3-yl)-4-phenyl-1H-imidazol-1-yl]propanamide
5-[(1R,6S)-9-methyl-3,9-diazabicyclo[4.2.1]nonane-3-carbonyl]-2-(thiophen-2-yl)pyrimidin-4-ol
8-chloro-2-({[3-(4-methyl-1H-pyrazol-1-yl)propyl]amino}methyl)quinolin-4-ol
2-[3-(3,5-dimethyl-1H-pyrazol-1-yl)azetidine-1-carbonyl]-8-fluoroquinoline
N,N-dimethyl-1-(5-{3-[3-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl}pyridin-2-yl)pyrrolidin-3-amine
N-[2-(pyrrolidin-1-yl)ethyl]-4-(4H-1,2,4-triazol-4-yl)benzamide
1-[(3R,4R)-3-({[2-(dimethylamino)ethyl](methyl)amino}methyl)-4-(hydroxymethyl)pyrrolidin-1-yl]-2-(3-methylphenyl)ethan-1-one
(1R,3S)-7-[4-(1H-pyrazol-3-yl)benzoyl]-7-azaspiro[3.5]nonane-1,3-diol
4-methoxy-6-(3-{1-[(5-methyl-1,2-oxazol-3-yl)methyl]-1H-pyrazol-3-yl}phenyl)pyrimidine
1-methyl-4-{2-[3-(2-methylphenoxy)azetidine-1-carbonyl]pyrrolidin-1-yl}piperidine
3-[4-(2H-1,3-benzodioxol-5-ylmethyl)piperazin-1-yl]-N-benzylpiperidine-1-carboxamide
3-ethoxy-1-{4-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}propan-1-one
N3-(cyclopropylmethyl)-N5-[2-(3-fluorophenyl)ethyl]-4-oxo-1-(oxolan-2-ylmethyl)-N3-propyl-1,4-dihydropyridine-3,5-dicarboxamide
3-(2-fluorophenyl)-1-(6-methoxy-3-methyl-1-benzofuran-2-carbonyl)pyrrolidine
N-methyl-4-[4-(quinazolin-4-yl)piperazine-1-carbonyl]-1,3-thiazol-2-amine
1,3-dimethyl-5-{[(1S,5R)-3-methyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]sulfonyl}-2,3-dihydro-1H-1,3-benzodiazol-2-one
4-(1-{8-methylimidazo[1,2-a]pyridine-2-carbonyl}pyrrolidin-3-yl)-2-(pyridin-4-yl)pyridine
N-(oxolan-3-yl)-4-(3,3,3-trifluoropropyl)pyrimidin-2-amine
3-[2-(dimethylamino)ethyl]-8-[(2E)-3-phenylprop-2-en-1-yl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
(1H-imidazol-2-ylmethyl)(methyl)[1-(pyridin-3-yl)propyl]amine
3,4,4-trimethyl-1-{4-[(pyridin-2-ylsulfanyl)methyl]benzoyl}pyrrolidin-3-ol
8-[4-(methylamino)pyrimidin-2-yl]-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one