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6-cyclopentyl-2-{3-[(3,3-difluoropiperidin-1-yl)methyl]phenyl}-3,4-dihydropyrimidin-4-one
2-methyl-N-({1-[(2-methyl-1H-imidazol-1-yl)methyl]cyclopropyl}methyl)thieno[2,3-d]pyrimidin-4-amine
1-[2-(2-oxo-2,3-dihydro-1,3-benzoxazol-3-yl)ethyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
5-methanesulfonyl-1'-(pyrimidin-2-yl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
1,3-dimethyl-N-{[2-(pyrimidin-2-yl)-1,3-thiazol-4-yl]methyl}-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
6-methyl-N-[(3-methylpyridin-4-yl)methyl]-2-(piperidin-1-yl)pyrimidin-4-amine
5-(azepane-1-carbonyl)-N-(1-benzothiophen-2-ylmethyl)-1-(butan-2-yl)-4-oxo-1,4-dihydropyridine-3-carboxamide
N-methyl-N-(oxolan-3-yl)-4-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzamide
N-(oxolan-2-ylmethyl)-N-(thiophen-3-ylmethyl)-2-(thiophene-2-sulfonamido)acetamide
1-[(3,5-dimethyl-1H-pyrazol-4-yl)sulfonyl]-N-methyl-N-(2-phenylethyl)piperidin-3-amine
N-(1,4-dioxan-2-ylmethyl)-6-ethyl-N,2-dimethylquinoline-4-carboxamide
[1-(2,6-difluorobenzenesulfonyl)-4-(3-phenylpropyl)piperidin-4-yl]methanol
2-(4-cyclohexyl-6-hydroxy-1,4-diazepane-1-carbonyl)benzonitrile
N-[(2-fluorophenyl)methyl]-1-{2-[(2,3,4-trimethoxyphenyl)formamido]ethyl}-1H-1,2,3-triazole-4-carboxamide
2-(3-fluorophenyl)-N-[4-(4-{[1-(2-methyl-1,3-thiazol-4-yl)ethyl]amino}piperidin-1-yl)phenyl]acetamide
N-[(1-hydroxycyclohexyl)methyl]-1-[(2-methoxyphenyl)methyl]-6-oxopiperidine-3-carboxamide
5-[3-(2-methoxyphenoxy)azetidine-1-carbonyl]-N,N,4-trimethylpyrimidin-2-amine
(1R,5R)-3-methanesulfonyl-6-(thiophen-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
3-(4-acetyl-3,5-dimethyl-1H-pyrazol-1-yl)-N-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)propanamide
(2S,4S)-4-amino-N,N-diethyl-1-(2-methoxypyrimidine-5-carbonyl)pyrrolidine-2-carboxamide
2-amino-6-cyclohexyl-4-{5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl}pyridine-3-carbonitrile
3-(5-methyl-1,3,4-thiadiazol-2-yl)-N-[(5-methyl-1H-pyrazol-3-yl)methyl]aniline
(3S,4R)-1-(5-ethyl-2,6-dimethylpyrimidin-4-yl)-4-(4-methoxyphenyl)-N,N-dimethylpyrrolidin-3-amine
N6-benzyl-N5-methyl-N5-[2-(morpholin-4-yl)ethyl]-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
1-[4-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]-2-(2-methylphenoxy)ethan-1-one
4-{4-[(2,1,3-benzothiadiazol-5-ylmethyl)amino]piperidin-1-yl}-N-[(3S)-2-oxoazepan-3-yl]benzamide
N-benzyl-3-[(3R)-3-hydroxy-3,4,4-trimethylpyrrolidin-1-yl]-N-methylpropanamide
N-({5-methyl-2-[2-(2-phenylacetamido)phenyl]-1,3-oxazol-4-yl}methyl)-3-(pyridin-4-yl)propanamide
4-(4-methylpiperazin-1-yl)-6-(1H-pyrazol-4-yl)quinazoline
6,6-dimethyl-1-phenyl-4,5,6,7-tetrahydro-1H-indazol-4-amine
N-{[5-fluoro-2-(trifluoromethyl)phenyl]methyl}-5-oxo-1-(propan-2-yl)pyrrolidine-3-carboxamide
3-cyclopentyl-5-(1H-imidazol-1-ylmethyl)-1-(2-phenylethyl)-1H-1,2,4-triazole
(2,1,3-benzothiadiazol-5-ylmethyl)({[1-(2-methoxyethyl)piperidin-4-yl]methyl})(pyridin-4-ylmethyl)amine
1-(1,3-dimethyl-1H-pyrazole-4-carbonyl)-3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine
(2R)-2-{[1,3-dimethyl-6-(pyridin-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]amino}-3-phenylpropan-1-ol
1-(2,3-dihydro-1-benzofuran-5-ylmethyl)-N-[2-(3,4-dimethoxyphenyl)ethyl]-N-methylpiperidin-3-amine
N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-2-{2-[(dimethylamino)methyl]-4-phenylphenoxy}acetamide
1-[(3,4-dimethoxyphenyl)methyl]-3-[5-methyl-1-(propan-2-yl)-1H-1,2,4-triazol-3-yl]urea
2-(3-hydroxypropyl)-9-(4-methoxy-3-methylbenzoyl)-2,9-diazaspiro[5.5]undecan-3-one
1-[(1-cyclopropyl-1H-imidazol-5-yl)methyl]-5-methyl-5-(4-methylpent-3-en-1-yl)piperidin-2-one
2-{2-chloro-4-[(3-hydroxyazetidin-1-yl)methyl]phenoxy}propanoic acid
1-cyclopentyl-N5-[furan-2-yl(phenyl)methyl]-N3-methyl-N3-(2-methylpropyl)-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
5-{1-[3-(3-methoxyphenyl)-1H-pyrazole-4-carbonyl]pyrrolidin-2-yl}-3-methyl-1,2-oxazole
1-benzyl-4-[2-(1-methyl-1H-1,3-benzodiazol-2-yl)-1H-imidazol-1-yl]pyrrolidin-2-one
8-[3-(2-methyl-1H-imidazol-1-yl)propyl]-2-(3-methylbutyl)-2,8-diazaspiro[5.5]undecan-3-one
5-{2-phenyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl}-4H,5H,6H,7H-[1,3]thiazolo[5,4-c]pyridin-2-amine
1,3,6-trimethyl-5-{6-[(pyridin-3-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
9-[6-methyl-2-(methylamino)pyrimidin-4-yl]-2-(1-methylpyrrolidin-3-yl)-2,9-diazaspiro[5.5]undecan-3-one
(4aS,8aR)-6-{2-[cyclopentyl(methyl)amino]acetyl}-1-[2-(methylamino)ethyl]-decahydro-1,6-naphthyridin-2-one
3-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}-N-(2-methoxyphenyl)piperidine-1-carboxamide