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1-(2-methoxyethyl)-4-{[2-(2-methoxyphenyl)-1,3-thiazol-5-yl]methyl}piperazine
(4aS,8aR)-1-butyl-6-[(1-methyl-1H-pyrazol-4-yl)methyl]-decahydro-1,6-naphthyridin-2-one
1-(3-methoxypropyl)-3-(naphthalen-2-ylmethyl)-8-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
7-(5-chloropyridin-2-yl)-4-(pyrazine-2-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2-{4-[1-(thiophen-3-ylmethyl)piperidin-4-yl]piperazin-1-yl}ethan-1-ol
N-[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl]-3-[(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)amino]-5-(dimethylsulfamoyl)benzamide
6-(2-aminoethyl)-N-ethyl-N-[(5-methylfuran-2-yl)methyl]pyrimidin-4-amine
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-5-(1H-pyrazol-1-ylmethyl)furan-2-carboxamide
5-{[1-(2-fluoro-4-methoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}-2-methyl-1,3-thiazole
9-methyl-3-[(5-propylfuran-2-yl)methyl]-3,9-diazaspiro[5.6]dodecan-10-one
1-benzyl-3-[3-(pyridin-3-yl)propyl]-8-(1,3-thiazol-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-({2-amino-6-[3-(dimethylamino)phenyl]pyrimidin-4-yl}amino)ethan-1-ol
1-[3-oxo-3-(3-oxo-4-phenylpiperazin-1-yl)propyl]azepan-2-one
1-{1-[(3-ethyl-1H-pyrazol-5-yl)methyl]piperidin-4-yl}pyrrolidin-2-one
N-({1-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]cyclopropyl}methyl)-5-oxo-1-(pyridin-3-ylmethyl)pyrrolidine-3-carboxamide
5-(2-chloro-4-fluorophenoxymethyl)-N-methyl-N-[(5-methylfuran-2-yl)methyl]-1,2-oxazole-3-carboxamide
4-methyl-2-(2-{[3-(1H-pyrazol-1-yl)phenyl]formamido}ethyl)-1,3-thiazole-5-carboxylic acid
3-(pyridin-4-yl)-1-[4-(pyrimidin-2-yloxy)piperidin-1-yl]propan-1-one
2-[3-({methyl[(1-methyl-1H-indol-3-yl)methyl]amino}methyl)piperidin-1-yl]ethan-1-ol
5-acetyl-N-{2-[methyl(phenyl)amino]propyl}thiophene-3-carboxamide
(1R,5R)-3-benzoyl-6-({6-methylimidazo[1,2-a]pyridin-2-yl}methyl)-3,6-diazabicyclo[3.2.2]nonane
N-ethyl-N-{[2-(prop-2-en-1-yloxy)phenyl]methyl}azepane-4-carboxamide
N-[(3R,5S)-5-(diethylcarbamoyl)-1-propanoylpyrrolidin-3-yl]-2-hydroxypyridine-3-carboxamide
1-(1-carbamoylcyclopropanecarbonyl)-N-[3-(3-methylphenyl)phenyl]pyrrolidine-2-carboxamide
7-(1,3-benzothiazol-2-yl)-4-(pyrrolidine-1-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-(3-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}-3-oxopropyl)-3-methoxybenzamide
(2S,4S)-4-amino-N-ethyl-1-[1-(furan-2-ylmethyl)piperidine-4-carbonyl]pyrrolidine-2-carboxamide
N-(6-chloropyridin-3-yl)-4-ethylpiperazine-1-carboxamide
2-{[3-(trifluoromethyl)phenyl]methyl}-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
(3S,4R)-1-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-4-(3-methoxyphenyl)pyrrolidine-3-carboxylic acid
7-amino-4-(3-hydroxyphenyl)-1,2,3,4-tetrahydro-1,8-naphthyridin-2-one
1-[(4-chlorophenyl)methyl]-5-(3-ethyl-1,2,4-oxadiazol-5-yl)piperidin-2-one
N-(propan-2-yl)-2-{[3-(trifluoromethyl)-1H-pyrazol-5-yl]formamido}acetamide
N,2-diethyl-N-methyl-4-phenyl-2,9-diazaspiro[5.5]undecane-9-sulfonamide
N-{2-[(1S,9aR)-octahydro-1H-quinolizin-1-yl]ethyl}pyrimidin-4-amine
3-[(2-fluorophenyl)methyl]-4-(2-methylphenyl)-4H-1,2,4-triazole
N-[2-(dimethylamino)-3-methylbutyl]-[1,2,3,4]tetrazolo[1,5-a]pyridine-6-carboxamide
2-[5-(2,6-dimethylpyrimidin-4-yl)-3-(thiophen-2-ylmethyl)-1H-1,2,4-triazol-1-yl]acetic acid
N-[(4-ethyl-1,3-thiazol-2-yl)methyl]-6-{methyl[(1-methylpyrrolidin-2-yl)methyl]amino}pyridine-3-carboxamide
3-ethoxy-1-{3-[2-methyl-6-(morpholin-4-yl)pyrimidin-4-yl]piperidin-1-yl}propan-1-one
N3-ethyl-1-(2-methylpropyl)-4-oxo-N5-[(5-phenyl-1,2-oxazol-3-yl)methyl]-1,4-dihydropyridine-3,5-dicarboxamide
N-[(4-methyl-1,3-thiazol-2-yl)methyl]-2-[(quinolin-8-yloxy)methyl]-1,3-oxazole-4-carboxamide
N3-tert-butyl-N5-{[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
{[3-(2H-1,3-benzodioxol-5-yl)-1-benzyl-1H-pyrazol-4-yl]methyl}(methyl)[(5-propyl-1H-pyrazol-3-yl)methyl]amine
4-{4-[(3-ethoxy-4-methoxyphenyl)methyl]piperazin-1-yl}-2-(thiophen-3-ylmethyl)-2,3-dihydro-1H-isoindole-1,3-dione
4-{3-[(4S,4aS,8aR)-4-hydroxy-4-phenyl-decahydroquinoline-1-carbonyl]piperidin-1-yl}-2-[2-(1H-pyrazol-1-yl)ethyl]-2,3-dihydro-1H-isoindole-1,3-dione
1-{[3-(4-fluorophenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}-4-(furan-2-carbonyl)piperazine
1-{[2-(trifluoromethyl)phenyl]methyl}-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
1-(2-chlorophenyl)-3-{1-[1-(4-fluorobenzoyl)piperidin-4-yl]-1H-pyrazol-5-yl}urea
({5-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]-4-ethyl-4H-1,2,4-triazol-3-yl}methyl)dimethylamine