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N-[2-(4-fluorobenzenesulfonyl)ethyl]-1,3-dimethyl-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
4-methyl-2-(4-methylpiperazin-1-yl)-5-[1-phenyl-3-(propan-2-yl)-1H-1,2,4-triazol-5-yl]pyrimidine
N-{[1-(pyrrolidin-1-yl)cyclopentyl]methyl}-1H-pyrazole-4-carboxamide
(4aR,7aS)-1-(2-hydroxyethyl)-4-(naphthalen-1-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
6-(2,5-dimethylfuran-3-yl)-N-ethyl-N,7-dimethyl-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
2-{4-cyclopentyl-1-[(2-fluorophenyl)methyl]piperazin-2-yl}ethan-1-ol
N-{[2-(cyclopentanesulfonyl)-1-(3-methoxypropyl)-1H-imidazol-5-yl]methyl}-N-methylcyclohexanamine
2-(2-methoxyethyl)-8-(1-methyl-1H-indole-3-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
1-methyl-5-{8-oxatricyclo[7.4.0.02,7]trideca-1(9),2(7),3,5,10,12-hexaen-6-yl}-1H,4H-pyrazolo[3,4-d]imidazole
methyl 4-[({1-[4-(morpholine-4-carbonyl)phenyl]piperidin-4-yl}amino)methyl]benzoate
1-({1-[(4-acetamidophenyl)methyl]piperidin-3-yl}methyl)-N,N-diethyl-1H-1,2,3-triazole-4-carboxamide
4-(4-chlorophenyl)-N-methyl-N-[1-(1,2-oxazol-3-yl)ethyl]butanamide
5-(1,4-oxazepan-4-ylmethyl)isoquinoline
2-(2,5-dioxoimidazolidin-4-yl)-N-{2-[2-(propan-2-yl)-1,3-thiazol-4-yl]ethyl}acetamide
{4-[(4-methoxyphenyl)methyl]-1-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}piperidin-4-yl}methanol
1-(2-methoxyethyl)-N-[(3-phenylphenyl)methyl]piperidine-3-carboxamide
(1R,6S)-3-[5-(methoxymethyl)furan-2-carbonyl]-9-methyl-3,9-diazabicyclo[4.2.1]nonane
2-[5-(oxolan-2-yl)thiophene-2-carbonyl]-2,3-dihydro-1H-isoindole
4-(4-ethyl-5-methylthiophene-3-carbonyl)-1-(3-methoxyphenyl)piperazin-2-one
1-[(2,2-dimethyloxan-4-yl)methyl]-4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazine
(4aS,7aR)-1-(2-aminopyridine-4-carbonyl)-4-(3-methylbut-2-en-1-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-{1-[1-(2,3-dihydro-1H-inden-2-yl)-1H-1,2,4-triazol-5-yl]ethyl}methanesulfonamide
N-{1-[(4-chlorophenyl)methyl]piperidin-3-yl}-2-(2-oxo-1,3-oxazolidin-3-yl)acetamide
N-[2-(3-methyl-1H-pyrazol-1-yl)ethyl]-4-(trimethyl-1H-pyrazol-4-yl)pyrimidin-2-amine
1-(3-chloro-4-methoxyphenyl)-4-[3-(pyridazin-3-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-2-one
1-(diethylamino)-3-{2-methoxy-4-[(4-methyl-1,2,3,6-tetrahydropyridin-1-yl)methyl]phenoxy}propan-2-ol
N-[(2,3-difluoro-4-methoxyphenyl)methyl]-5-(morpholin-4-ylmethyl)furan-3-carboxamide
N-(6,6-dimethyl-1-phenyl-4,5,6,7-tetrahydro-1H-indazol-4-yl)-4-(2-oxopyrrolidin-1-yl)butanamide
N-({5-cyclohexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-1-ethyl-5-methyl-1H-pyrazole-4-carboxamide
2-[5-(2-phenylethyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl]pyridine
N-[6,6-dimethyl-1-(2-methylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-4-methyl-1,2,5-oxadiazole-3-carboxamide
2-[9-(3-hydroxy-4-methoxybenzoyl)-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl]acetamide
N-({2-[2-(2-cyclopentylacetamido)phenyl]-5-methyl-1,3-oxazol-4-yl}methyl)-1-methyl-3-propyl-1H-pyrazole-5-carboxamide
3-[2-(10-methoxy-3,4,5,6-tetrahydro-2H-1,5-benzoxazocin-5-yl)-2-oxoethyl]imidazolidine-2,4-dione
2-[(3S,4R)-3-(dimethylamino)-4-(4-methoxyphenyl)pyrrolidin-1-yl]pyridine-4-carboxylic acid
1-cyclopentanecarbonyl-N-{2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-yl}piperidin-4-amine
3-{2-oxo-2-[4-(thiomorpholin-4-yl)piperidin-1-yl]ethyl}-4-(pyridin-3-ylmethyl)piperazin-2-one
N-{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-N-methylpyrazolo[1,5-a]pyrimidine-3-carboxamide
5-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}-4H,5H,6H,7H-[1,3]thiazolo[5,4-c]pyridin-2-amine
2-methyl-4-propyl-6-{4-[4-(1H-pyrazol-1-ylmethyl)piperidin-1-yl]piperidin-1-yl}pyrimidine
N-ethyl-N-methyl-6-(3-{1-[(1-methylpyrrolidin-3-yl)methyl]-1H-pyrazol-3-yl}phenyl)pyrimidin-4-amine
5-(2-phenylmethanesulfonylbenzoyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
(4aS,8aR)-6-[2-(1H-imidazol-1-yl)acetyl]-1-[2-(methylamino)ethyl]-decahydro-1,6-naphthyridin-2-one
4-[2-(2-chlorophenyl)ethyl]-11-(4-ethylpiperazin-1-yl)-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
N-[(3S)-1-benzylpyrrolidin-3-yl]-3-(2-methylpropyl)-1,2-oxazole-5-carboxamide
4-hydroxy-1-(3-phenoxybenzenesulfonyl)piperidine-4-carboxylic acid
2-(methylamino)-2-phenyl-N-({5-propyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)acetamide
(4aR,8aS)-6-{[4-(dimethylamino)phenyl]methyl}-1-[3-(2-oxopyrrolidin-1-yl)propyl]-decahydro-1,6-naphthyridin-2-one
N5,N5-dimethyl-N6-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
2-(4-{2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}piperazin-1-yl)pyridine-3-carbonitrile