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N-[2-(dimethylamino)-2-(furan-2-yl)ethyl]-1-methyl-2-oxo-1,2-dihydroquinoline-3-carboxamide
N-{[4-(1H-1,3-benzodiazol-2-yl)cyclohexyl]methyl}-3-propyl-1H-pyrazole-5-carboxamide
3-[3-(1-methyl-1H-imidazole-2-carbonyl)phenyl]pyridine
2-(2-methoxyethyl)-8-{5-[(methylsulfanyl)methyl]furan-2-carbonyl}-2,8-diazaspiro[5.5]undecan-3-one
6-[(2S,4R)-4-amino-2-(diethylcarbamoyl)pyrrolidin-1-yl]-N,N-dimethylpyridine-3-carboxamide
N-(1-{7-[(4-methoxy-2,5-dimethylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-1-methylpiperidine-4-carboxamide
3-(2-{4-methyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}ethyl)-1H-indole
1-(cyclopropylmethyl)-4-(2,3-difluoro-4-methoxybenzoyl)-2-(propan-2-yl)-1,4-diazepane
1-{2-[3-(hydroxymethyl)-3-propylpiperidin-1-yl]pyrimidin-4-yl}piperidin-4-ol
[(3aS,6aS)-2-{1-[5-(trifluoromethyl)pyridin-2-yl]piperidin-4-yl}-octahydrocyclopenta[c]pyrrol-3a-yl]methanol
2-{3-oxo-1-[(2E)-3-phenylprop-2-en-1-yl]piperazin-2-yl}-N-[3-(pyridin-3-yl)propyl]acetamide
4-(propan-2-yl)-5-[(2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazol-1-yl)methyl]-1,2,3-thiadiazole
2-(4-{1-[2-(pyridin-2-yl)ethyl]-1,2,3,6-tetrahydropyridin-4-yl}-1H-pyrazol-1-yl)pyridine
N-[(4-ethyl-1,3-thiazol-2-yl)methyl]-6-(3-ethyl-4-methylpiperazin-1-yl)pyridine-3-carboxamide
N-[(3-methyl-1-benzofuran-2-yl)methyl]-1,9-dioxaspiro[5.5]undecan-4-amine
6-[3-(1,2-dihydroacenaphthylene-5-carbonyl)piperidine-1-carbonyl]-1,3-dimethyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
(4aR,7aS)-1-(2-hydroxyethyl)-4-(3-phenoxypropanoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-(furan-2-yl)-5-({4-[(3-methylphenyl)methyl]piperazin-1-yl}methyl)pyrimidine
N-{[5-(2H-1,3-benzodioxol-5-ylmethyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}cyclobutanecarboxamide
8-[(6-ethoxypyridin-3-yl)methyl]-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
methyl[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]{[5-methyl-2-(thiophen-3-yl)-1,3-oxazol-4-yl]methyl}amine
9-hydroxy-4-oxo-N-[(1R,2S)-2-phenylcyclohexyl]-4H-pyrido[1,2-a]pyrimidine-3-carboxamide
2-[4-(2-phenylethyl)-4H-1,2,4-triazol-3-yl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
1-cyclobutanecarbonyl-N-{1-[4-(dimethylamino)phenyl]propan-2-yl}piperidine-4-carboxamide
N2-benzyl-N2,7,7-trimethyl-N5-(oxan-4-yl)-5,6,7,8-tetrahydroquinazoline-2,5-diamine
2-{1-[(3,5-dimethoxyphenyl)methyl]-4-(1,2-oxazol-3-ylmethyl)piperazin-2-yl}ethan-1-ol
(4aR,7aS)-1-benzyl-4-[2-(dimethylamino)acetyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2,2-dimethyl-N-{1-[1-(4,5,6,7-tetrahydro-1,2-benzoxazole-3-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}propanamide
(butan-2-yl)(pyridin-4-ylmethyl){[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}amine
(3S,5R)-1-[(2-ethylphenyl)methyl]-5-[(6-methylpyridin-3-yl)carbamoyl]piperidine-3-carboxylic acid
N-{[2-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}-2-(3-oxo-3,4-dihydro-2H-1,4-benzoxazin-6-yl)acetamide
2-{[4-(2-methoxy-5-methylphenyl)-5-(1H-pyrazol-4-yl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
N-[4-(3-methanesulfonamidopropanamido)-2-methylphenyl]pentanamide
2-methyl-3-oxo-4-phenyl-N-propyl-2,9-diazaspiro[5.5]undecane-9-carboxamide
ethyl 2-{[1,3-dimethyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]amino}acetate
2-[(2-ethylphenyl)methyl]-8-methyl-octahydro-1H-pyrazino[1,2-a]piperazine
3-(3-propylmorpholine-4-carbonyl)benzonitrile
4-[(2H-1,3-benzodioxol-5-ylmethyl)amino]-5-methyl-N-(3-methylbutyl)thieno[2,3-d]pyrimidine-6-carboxamide
3-[3-(2-ethyl-1H-imidazol-1-yl)propyl]-1-[3-(5-methyl-4H-1,2,4-triazol-3-yl)phenyl]urea
7-methoxy-4-(morpholine-4-carbonyl)-2-(1-propyl-1H-pyrazol-4-yl)quinoline
N-methyl-N-{[2-(methylamino)pyrimidin-5-yl]methyl}-3-(trimethyl-1H-pyrazol-4-yl)propanamide
3-(3-hydroxy-3-methylbutyl)-N-methyl-N-[(5-methyl-1H-1,3-benzodiazol-2-yl)methyl]benzamide
1-(2,2-dimethoxyethyl)-4-[(4-fluoro-2-methylphenyl)methyl]piperazine
(3S,4R)-1-(1-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carbonyl)-4-(2-methylphenyl)pyrrolidine-3-carboxylic acid
1-methyl-N-{2-[(pyridin-3-yl)amino]ethyl}-1H-indole-4-carboxamide
1-{4-[3-(1H-indol-3-ylmethyl)-4H-1,2,4-triazol-4-yl]phenyl}ethan-1-one
ethyl(methyl)[({1-[(2E)-2-methylpent-2-en-1-yl]piperidin-4-yl}methyl)sulfamoyl]amine
(2S,4R)-N,1-bis(propan-2-yl)-4-({[2-(trifluoromethyl)phenyl]methyl}amino)pyrrolidine-2-carboxamide
(1R,2R,6S,7S)-4-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-4-azatricyclo[5.2.1.02,6]decane
1-(1-{[2-(2-ethylphenyl)-1H-imidazol-1-yl]methyl}cyclopentyl)-4-methylpiperazine