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1-({4-oxo-4H-pyrido[1,2-a]pyrimidin-2-yl}methyl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
5-(4-{5-[(dimethylamino)methyl]-4-ethyl-4H-1,2,4-triazol-3-yl}piperidine-1-carbonyl)pyridine-2-carbonitrile
[1-(2-aminopyrimidin-4-yl)-3-[(2,4-difluorophenyl)methyl]piperidin-3-yl]methanol
1-[3-(2,5-dimethoxyphenyl)pyrrolidin-1-yl]-2-(1H-1,2,4-triazol-1-yl)ethan-1-one
3-{[7-acetyl-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl]amino}-N,N-dimethylpropanamide
methyl 6-{3-[3-(propan-2-yloxy)benzoyl]piperidin-1-yl}pyrazine-2-carboxylate
N-[2-(benzyloxy)ethyl]-1-methylpiperidine-2-carboxamide
3-(1-{[1-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}piperidin-4-yl)-N-(oxolan-2-ylmethyl)propanamide
2-(methoxymethyl)-6-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]pyridine
1-(pyridin-2-ylmethyl)-4-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)pyrrolidin-2-one
N-(oxolan-2-ylmethyl)-3-[1-(quinoxalin-2-yl)piperidin-4-yl]propanamide
1-(1'-{6-[ethyl(methyl)amino]pyrimidin-4-yl}-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl)propan-1-one
{[2-(morpholine-4-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}({[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl})amine
4-(azepan-1-yl)-N-methyl-4-oxo-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}butanamide
5-[3-(2-methoxyphenoxy)azetidine-1-carbonyl]-1-methyl-3-(trifluoromethyl)-1H-pyrazole
N-[1-(4-methoxyphenyl)-4-(propan-2-yloxy)-1H-indazol-3-yl]-1-methyl-1H-pyrazole-3-carboxamide
3-(methanesulfonylmethyl)-1-{[3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}piperidine
1,3,5-trimethyl-4-(1-methyl-5-{4H,5H,6H,7H-thieno[3,2-c]pyridine-5-carbonyl}-1H-pyrazol-3-yl)-1H-pyrazole
(1-{1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]piperidin-3-yl}piperidin-4-yl)methanol
N-cyclopropyl-1-{1-[(3-fluoro-2-methylphenyl)methyl]piperidin-4-yl}piperidine-3-carboxamide
1-{[5-(2-chlorophenyl)furan-2-yl]methyl}-4-(prop-2-en-1-yl)-1,4-diazepan-5-one
(2S,4R)-N-{[2-(azocan-1-yl)pyridin-3-yl]methyl}-4-hydroxypyrrolidine-2-carboxamide
1-(2,5-dimethylpyrimidin-4-yl)-3-(3-methoxypropyl)piperidine-3-carboxylic acid
2-amino-3-ethyl-N-{[4-(1H-1,2,4-triazol-1-yl)phenyl]methyl}-3H-imidazo[4,5-b]pyridine-6-carboxamide
3-({[3-(2,3-dihydro-1H-indol-1-yl)propyl]amino}methyl)pyrrolidin-3-ol
4-({1-[3-(methylsulfanyl)propanoyl]pyrrolidin-3-yl}methyl)benzoic acid
(3aR,6aR)-2-(cyclobutylmethyl)-5-(4-oxo-4-phenylbutanoyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
(2S,4R)-N-ethyl-1-(3-methylbut-2-en-1-yl)-4-(5-methylthiophene-3-amido)pyrrolidine-2-carboxamide
5-(4-ethylpiperazin-1-yl)-3-(piperidine-1-carbonyl)-1-propyl-4,5,6,7-tetrahydro-1H-indazole
2-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)-1-(4-hydroxy-1,2-oxazolidin-2-yl)ethan-1-one
(3S,4S)-1-{[2-(2,3-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidine-3,4-diol
ethyl 4-[(4-chlorophenyl)methyl]-1-[(2,4-dimethylphenyl)carbamoyl]piperidine-4-carboxylate
3-(1H-pyrazol-4-yl)-N-[1-(thian-4-yl)piperidin-4-yl]benzamide
2-methoxy-5-({3-[4-(4-methoxyphenyl)piperazin-1-yl]piperidin-1-yl}methyl)phenol
N-(2-methoxyethyl)-N-methyl-1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
N-[(3S,4R)-1-[2-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)acetyl]-4-propylpyrrolidin-3-yl]acetamide
3-ethyl-4-methyl-N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-N-(oxolan-2-ylmethyl)-1H-pyrazole-5-carboxamide
{[2-(difluoromethoxy)phenyl]methyl}(methyl)[1-(pyridin-3-yl)ethyl]amine
2-[6-(cyclopentylamino)-1H-pyrrolo[2,3-b]pyridin-4-yl]-N-(propan-2-yl)pyridine-4-carboxamide
N-(furan-2-ylmethyl)-6-({6-methylimidazo[2,1-b][1,3]thiazol-5-yl}methyl)-6-azaspiro[2.5]octane-1-carboxamide
3,5-dimethyl-1-{[5-methyl-2-(3-methylthiophen-2-yl)-1,3-oxazol-4-yl]methyl}-1H-1,2,4-triazole
3-{[(1-{pyrazolo[1,5-a]pyridine-3-carbonyl}piperidin-4-yl)oxy]methyl}pyridine
2-(1-{[3-(2-fluorophenyl)-1-methyl-1H-pyrazol-4-yl]methyl}piperidin-3-yl)-1H-1,3-benzodiazole
2-{5-[2-(3-chlorophenyl)-1H-imidazol-1-yl]-1H-1,3-benzodiazol-1-yl}ethan-1-ol
3-propoxy-N-[4-(1H-1,2,4-triazol-1-yl)phenyl]piperidine-1-carboxamide
N-(2-methoxyethyl)-1-(3-methylbutyl)-5-(pyridine-3-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-benzyl-8-(1-methoxypropan-2-yl)-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-[(2-methyl-1,3-oxazol-4-yl)methyl]-4-[1-(pyrrolidin-1-yl)ethyl]piperidine
2-(2-methoxy-4-methylphenoxymethyl)-N-methyl-N-(pyridin-3-ylmethyl)-1,3-oxazole-4-carboxamide
2-(2-amino-4,6-dimethylpyrimidin-5-yl)-1-{3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one