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2-[5-fluoro-4-(morpholin-4-yl)pyrimidin-2-yl]-1-methyl-1H-indole
3,3-dimethyl-1-({5-[(2,4,6-trifluorophenyl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)urea
3-(azepane-1-carbonyl)-N,N-dimethyl-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
2-(4-{[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]amino}piperidin-1-yl)pyridine-3-carbonitrile
({5-[(1S,5R)-3-benzyl-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]furan-2-yl}methyl)dimethylamine
3-[(8-methyl-2-oxo-1,2-dihydroquinolin-3-yl)methyl]-3,9-diazaspiro[5.6]dodecan-10-one
[3-ethyl-1-(3-methoxy-5-methylthiophene-2-carbonyl)piperidin-3-yl]methanol
1-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]-3-(3-methylthiophene-2-carbonyl)piperidine
N-(3-{4-[(5-hydroxyadamantan-2-yl)amino]piperidin-1-yl}phenyl)cyclopropanecarboxamide
N-[1-(2,3-dihydro-1,4-benzodioxin-6-yl)ethyl]-N-methyl-1-(4-methylquinazolin-2-yl)piperidine-4-carboxamide
(3R,4S)-1-{[2-(cyclopentylmethyl)-1H-imidazol-4-yl]methyl}-3,4-dimethylpiperidin-4-ol
N-[3-(4-{[3-(dimethyl-1,2-oxazol-4-yl)propanamido]methyl}-5-methyl-1,3-oxazol-2-yl)phenyl]-2-methylfuran-3-carboxamide
(1S,4S)-2-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-5-methyl-2,5-diazabicyclo[2.2.1]heptane
N-butyl-2-[1-(2,3-dihydro-1H-inden-2-yl)-3-oxopiperazin-2-yl]-N-(propan-2-yl)acetamide
1-[(2-fluorophenyl)methyl]-4-[3-(piperidin-3-yl)benzoyl]piperazine
1-[1-(1,7-dimethyl-1H-indole-2-carbonyl)piperidin-4-yl]-3-methylbutan-1-ol
1-(1-cyclohexylpiperidin-3-yl)-4-(2-methoxyphenyl)piperazine
N-(1,3-benzothiazol-2-ylmethyl)-3-{5-[methoxy(phenyl)methyl]-1,3,4-oxadiazol-2-yl}propanamide
5-ethyl-N-[2-(1-methyl-1H-pyrrol-2-yl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine
3-[4-(benzyloxy)piperidine-1-carbonyl]-2-methoxypyridine
N-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-6-methoxy-N,3-dimethyl-1-benzofuran-2-carboxamide
1-{6-[4-(trifluoromethyl)phenyl]imidazo[2,1-b][1,3]thiazole-3-carbonyl}piperidin-3-ol
N-[(2-chlorophenyl)methyl]-2-methyl-3-[(pyridin-3-ylmethyl)amino]benzamide
2-{1-[(2-fluoro-4-methoxyphenyl)methyl]-4-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]piperazin-2-yl}ethan-1-ol
1-{4-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}-4-(1H-1,2,4-triazol-1-yl)butan-1-one
5-[4-(1-butyl-1H-1,2,4-triazol-5-yl)phenyl]-2-methyl-2H-1,2,3,4-tetrazole
4-[4-(2-ethoxyphenyl)piperazine-1-carbonyl]-2,6-dimethylpyrimidine
N-[2-(methylamino)ethyl]-1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidine-3-carboxamide
1-methyl-4-(4-phenoxybutanoyl)-1,4,9-triazaspiro[5.6]dodecan-10-one
6-(2,5-dimethylfuran-3-yl)-N-(3-ethoxypropyl)-7-methyl-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
1-cyclohexyl-5-[3-(1H-imidazol-1-yl)propyl]-1H-1,2,4-triazole
N-[2-(dimethylamino)ethyl]-4-[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]-N-(oxolan-2-ylmethyl)butanamide
ethyl 4-({4-[(1-{imidazo[1,2-a]pyridine-2-carbonyl}piperidin-3-yl)methoxy]phenyl}methyl)piperazine-1-carboxylate
2,4-dimethyl-5-{2-[2-(pyrrolidin-1-yl)ethyl]piperidine-1-carbonyl}pyrimidine
N-(2,1,3-benzoxadiazol-5-ylmethyl)-2-methyl-3-[(pyridin-3-ylmethyl)amino]benzamide
(2E)-N-[(3,4-dimethoxyphenyl)methyl]-3-(4-methoxyphenyl)-N-(pyridin-4-ylmethyl)prop-2-enamide
{[3-(2H-1,3-benzodioxol-5-yl)-1-benzyl-1H-pyrazol-4-yl]methyl}(methyl)[2-(2-methyl-1H-imidazol-1-yl)ethyl]amine
N-[(2-ethoxypyridin-3-yl)methyl]-2,7-dioxo-1,3-diazepane-4-carboxamide
2-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}-6-(pyrrolidine-1-carbonyl)pyrazine
(2S)-2-(hydroxymethyl)-N-(1-methyl-1H-indazol-5-yl)pyrrolidine-1-carboxamide
N,N-diethyl-3-(3-hydroxy-3-methylbutyl)benzamide
4-(2H-1,3-benzodioxol-5-yl)-2-{4-[4-(4-fluorophenyl)piperazine-1-carbonyl]-5-methyl-1H-pyrazol-1-yl}pyrimidine
4-[(1R,6S)-9-methyl-3,9-diazabicyclo[4.2.1]nonan-3-yl]-6-(thiophen-2-ylsulfanyl)pyrimidin-2-amine
N-[1-(1-ethyl-1H-1,2,4-triazol-5-yl)ethyl]-2,5,6-trimethylpyrimidin-4-amine
4-(4-{3-[(4-fluorophenyl)methyl]piperidin-1-yl}-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-2-yl)pyridine
(3S,4S)-1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-4-(propan-2-yloxy)pyrrolidin-3-ol
4-(4-methyl-4H-1,2,4-triazol-3-yl)-1-[2-(thiophen-2-yl)-1,3-thiazole-4-carbonyl]piperidine
2-(2H-1,3-benzodioxol-5-yl)-1-[(3R,4R)-3-{[ethyl(2-hydroxyethyl)amino]methyl}-4-(hydroxymethyl)pyrrolidin-1-yl]ethan-1-one
3-methyl-5-{1-[2-(methylsulfanyl)-1,3-thiazole-4-carbonyl]pyrrolidin-2-yl}-1H-1,2,4-triazole
1-[4-(1-butyl-1H-imidazol-2-yl)piperidin-1-yl]-3-(trimethyl-1H-pyrazol-4-yl)propan-1-one