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(2E)-N-{[5-chloro-7-(pyrimidin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-(2,3-difluorophenyl)prop-2-enamide
2-[(cyclopropylmethyl)sulfanyl]-1-{4-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
8-[4-(hydroxymethyl)benzoyl]-3-methyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-(2H-1,3-benzodioxol-5-yl)-1-{[4-methoxy-3-(methoxymethyl)phenyl]methyl}piperidin-3-amine
N-(2-hydroxyethyl)-1-[2-(4-methoxyphenyl)ethyl]-N-methyl-6-oxopiperidine-3-carboxamide
N-(2H-1,3-benzodioxol-5-yl)-2-(1,3-thiazol-2-yl)piperidine-1-carboxamide
N-(2-methoxyethyl)-N-(thiophen-2-ylmethyl)pyrrolidine-3-carboxamide
6-[(diethylamino)methyl]-N-(3-hydroxy-4-methoxyphenyl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
2-{1-[1-(furan-2-ylmethyl)piperidine-4-carbonyl]pyrrolidin-2-yl}pyridine
(1R,5R)-N,N-dimethyl-6-[3-(thiophen-2-yl)propanoyl]-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
{[1-(4-butylphenyl)-1H-pyrazol-4-yl]methyl}[2-methyl-1-(1-methyl-1H-imidazol-2-yl)propyl]amine
5-{2-[2-(dimethylamino)ethyl]piperidine-1-carbonyl}-N-(3-methylbutyl)-1-(2-methylpropyl)-4-oxo-1,4-dihydropyridine-3-carboxamide
2-{2-[2-(4-fluorophenyl)piperidin-1-yl]ethoxy}ethan-1-ol
N-[1-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-2-[4-(methylsulfanyl)phenyl]acetamide
4-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]-1-{2-methylimidazo[1,2-a]pyridine-3-carbonyl}piperidine
{[1-({1-[(2,6-dimethylphenyl)methyl]piperidin-3-yl}methyl)-1H-1,2,3-triazol-4-yl]methyl}urea
N-(3,5-dimethoxyphenyl)-3-{1-[2-(2-oxopyrrolidin-1-yl)acetyl]piperidin-3-yl}propanamide
N-(2-hydroxybutyl)-4-{[(2-methoxyphenyl)methyl]amino}-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-{1H-pyrrolo[2,3-b]pyridin-6-yl}piperidin-3-ol
ethyl 4-[4-(4-{[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]amino}piperidin-1-yl)benzoyl]piperazine-1-carboxylate
N-[(2,5-difluorophenyl)methyl]-2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-amine
9-(2,5-difluorobenzoyl)-2-(2-hydroxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-(dicyclopropylmethyl)-5-[(4-hydroxypiperidin-1-yl)methyl]-N-methyl-1,2-oxazole-3-carboxamide
3-{3-cyclobutyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}-2-methyl-1,2,3,4-tetrahydroisoquinoline
3-[(5-amino-1,3,4-thiadiazol-2-yl)methyl]-1-[2-chloro-5-(pyrrolidine-1-carbonyl)phenyl]urea
N-methyl-N-[1-(4-methylpyridin-2-yl)propan-2-yl]-2-(pyridin-3-yloxy)acetamide
8-[(1-methyl-1H-imidazol-2-yl)methyl]-3-(2-phenylpropyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-cyclopentyl-5-[(5-acetamidothiophen-2-yl)methyl]-1-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
5-{1-[1-(2-ethoxyethyl)-3-methyl-1H-pyrazole-5-carbonyl]pyrrolidin-2-yl}-3-(propan-2-yl)-1,2,4-oxadiazole
3-{1-cyclohexyl-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}benzonitrile
1-methyl-3-(3-{4-[3-(morpholin-4-yl)azetidin-1-yl]piperidin-1-yl}phenyl)imidazolidin-2-one
N-ethyl-2-{4-[(1-ethyl-1H-indol-4-yl)methyl]piperazin-1-yl}acetamide
[4-(2-phenoxyethyl)-1-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}piperidin-4-yl]methanol
1-methyl-N-[3-(3-methylbenzamido)phenyl]piperidine-2-carboxamide
6-[1-tert-butyl-3-(oxan-4-yl)-1H-1,2,4-triazol-5-yl]-2,3,4,5-tetrahydropyridazin-3-one
3-(1-methylpiperidin-3-yl)-1-[4-(3-methylpyridin-4-yl)piperazin-1-yl]propan-1-one
(4-{5-[1-(propan-2-yl)piperidin-4-yl]-1,2,4-oxadiazol-3-yl}phenyl)methanol
2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-methyl-N-[1-(1,3-thiazol-5-yl)ethyl]-1,3-oxazole-4-carboxamide
N-[(1-benzyl-1H-pyrazol-4-yl)methyl]-6-ethyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
4-(5-{[3-(4-tert-butylbenzoyl)piperidin-1-yl]methyl}-1,3-thiazol-2-yl)morpholine
(3S,4R)-3-methoxy-1-(4-methoxy-3,5-dimethylbenzoyl)piperidin-4-amine
(2S,4S)-4-(1H-1,3-benzodiazol-2-ylsulfanyl)-1-[(3-methylphenyl)methyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
4-[1-(cyclohex-3-ene-1-carbonyl)piperidin-4-yl]-5-(3-methylphenyl)-2-(pyridin-4-yl)pyrimidine
1-(1-methylpiperidine-2-carbonyl)-4-[3-(trifluoromethyl)phenyl]piperidin-4-ol
2-ethoxy-6-{1-methyl-3-phenyl-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}phenol
1-{1-[5-(propan-2-yl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carbonyl]piperidin-4-yl}-2,3-dihydro-1H-1,3-benzodiazol-2-one
2-ethoxy-4-({3-[4-(piperidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}methyl)phenol
5-acetyl-N-methyl-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
2-(2-methoxy-5-methylphenyl)-2-{4-[(2-methyl-1,3-thiazol-4-yl)methyl]piperazin-1-yl}acetic acid
5-[3-(4-methoxy-3,5-dimethylbenzoyl)piperidine-1-carbonyl]-N-methylpyrimidin-2-amine