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5-[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]-N-methyl-N-[(1-methylpyrrolidin-2-yl)methyl]pyridin-2-amine
N-(1-hydroxybutan-2-yl)-N-(pyridin-3-ylmethyl)-1H-pyrrole-2-carboxamide
4-({2-[1-(2-ethylbenzoyl)piperidin-4-yl]-1H-imidazol-1-yl}methyl)pyridine
N-[2-(1H-imidazol-4-yl)ethyl]-3-(propan-2-yl)-1,2-oxazole-5-carboxamide
2-(dimethyl-1,2-oxazole-4-carbonyl)-N-(5-methyl-1,2-oxazol-3-yl)-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
N-[(4-hydroxyazepan-4-yl)methyl]-3-(trimethyl-1H-pyrazol-1-yl)propanamide
4-{4-ethyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}-1-(3-methylbutyl)piperidine
2-(2-{1-[1-(2-methoxyphenyl)-1H-pyrazole-4-carbonyl]piperidin-2-yl}ethyl)pyridine
N-methyl-N-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}-2-{5H,6H,7H-[1,3]thiazolo[3,2-a]pyrimidin-3-yl}acetamide
2-tert-butyl-8-{2,7-dimethylpyrazolo[1,5-a]pyrimidine-5-carbonyl}-1,3,8-triazaspiro[4.5]dec-1-en-4-one
1-[7-(2-methoxyacetamido)-1-(2-phenylethyl)-1H-1,3-benzodiazole-5-carbonyl]piperidine-3-carboxamide
1-({4-methyl-5-[1-(pyridazin-3-yl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)azepane
1-(3,4-dimethylphenyl)-3-methyl-5-[(oxolan-2-ylmethoxy)methyl]-1H-1,2,4-triazole
(4aR,7aS)-1-(2-hydroxyethyl)-4-[3-(2-methylphenyl)propanoyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-(1,2-oxazol-3-ylmethyl)-1-(pyridin-2-yl)-4,5,6,7-tetrahydro-1H-indazol-4-amine
8-(2-amino-4-methyl-1,3-thiazole-5-carbonyl)-2-(2-methoxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
1-[4-(5-tert-butyl-1,3,4-oxadiazol-2-yl)-1,4-diazepan-1-yl]-2,2,2-trifluoroethan-1-one
4-[(1R,5R)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]benzene-1-sulfonamide
2-[(3-fluorophenyl)methyl]-4-[4-(2-methylpropyl)piperazin-1-yl]-2,3-dihydro-1H-isoindole-1,3-dione
N-({1-[(5-ethylfuran-2-yl)methyl]piperidin-3-yl}methyl)-6-oxo-1,6-dihydropyridine-3-carboxamide
N-[2-(5-methoxy-1H-1,3-benzodiazol-2-yl)ethyl]-N,2,5-trimethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
(1R,2R,6S,7S)-N-(6-cyanopyridin-3-yl)-4-azatricyclo[5.2.1.02,6]decane-4-carboxamide
1-(7-chloro-4-methylquinolin-2-yl)-N-(1-methoxypropan-2-yl)piperidine-4-carboxamide
2-{4-[(3-fluorophenyl)methyl]-1-[(3-methoxyphenyl)methyl]piperazin-2-yl}ethan-1-ol
7-chloro-N-(3,4-diethyl-1-methyl-1H-pyrazol-5-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carboxamide
(2S)-2-amino-N-({5-cyclohexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-3-hydroxypropanamide
1-amino-N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)cyclopropane-1-carboxamide
(3S,4S)-1-(2,1,3-benzothiadiazol-4-ylmethyl)-4-(4-fluorophenyl)piperidin-3-ol
N-[3-(1H-indol-2-yl)phenyl]-1-(3,3,3-trifluoropropanoyl)piperidine-3-carboxamide
3-{[(1-carbamoyl-1-methylethyl)carbamoyl]methyl}-N,N,4-trimethyl-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
{1-[(2E)-2-methyl-3-phenylprop-2-en-1-yl]pyrrolidin-3-yl}methanamine
N-[(3S,4R)-1-(dimethylsulfamoyl)-4-(4-methoxyphenyl)pyrrolidin-3-yl]acetamide
N-[2-methoxy-1-(pyridin-2-yl)ethyl]-N,1-dimethyl-2-oxo-1,2,5,6,7,8-hexahydroquinoline-3-carboxamide
N-[(5-chloro-1H-1,3-benzodiazol-2-yl)methyl]-5-(4-methoxyphenyl)-N-methyl-1,2,4-triazin-3-amine
N-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine
2-(2-fluoro-6-methoxyphenyl)-4,6-dimethylpyridine-3-carbonitrile
3-(2-methyl-2H-1,2,3-benzotriazol-4-yl)-1-[1-(thian-4-yl)piperidin-4-yl]urea
{[5-(2-ethoxypyridin-3-yl)-1,2,4-oxadiazol-3-yl]methyl}dimethylamine
3,5-dimethyl-2-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}-1H-indole
[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl](4,4,4-trifluorobutan-2-yl)amine
N-[2-(4-ethyl-3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-2,5-dimethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
(3S,4R)-4-(4-methoxyphenyl)-N,N-dimethyl-1-{[2-(methylsulfanyl)phenyl]methyl}pyrrolidin-3-amine
4-[(1,1-dioxo-1λ6-thiomorpholin-4-yl)methyl]-N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}benzamide
N-cyclopropyl-1-{1-[(4-methoxynaphthalen-1-yl)methyl]piperidin-4-yl}-1H-1,2,3-triazole-4-carboxamide
N-(2-methylphenyl)-3-{[2-(pyrrolidine-1-sulfonyl)ethyl]amino}propanamide
3-{1-[2-(pyridin-3-yl)pyrimidine-5-carbonyl]piperidin-4-yl}benzonitrile
2-(ethoxymethyl)-N-methyl-N-{[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
(3S,4S)-1-[(1-ethyl-3-methyl-1H-pyrazol-5-yl)sulfonyl]-4-(pyridin-2-yl)pyrrolidine-3-carboxylic acid
3-(2,3-dihydro-1,4-benzodioxin-6-yl)-5-(pyrrolidine-1-sulfonyl)benzoic acid
1-[(2-methyl-1,3-thiazol-5-yl)methyl]-3-[3-(trifluoromethyl)benzoyl]piperidine