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N-(quinolin-4-ylmethyl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]cyclopropanamine
2-(3-{[2-(hydroxymethyl)piperidin-1-yl]methyl}phenoxy)acetamide
5-(1H-imidazol-1-ylmethyl)-N-[(5-methyl-1H-1,3-benzodiazol-2-yl)methyl]furan-2-carboxamide
3-(6-methoxynaphthalene-2-carbonyl)-1-[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]piperidine
N-[(3R,4S)-4-cyclopropyl-1-(piperidine-1-carbonyl)pyrrolidin-3-yl]-2-(pyridin-2-yl)acetamide
(4-methoxy-4-methylpentan-2-yl)({[4-(1H-1,2,4-triazol-1-yl)phenyl]methyl})amine
3-(azepane-1-carbonyl)-N-[2-(morpholin-4-yl)ethyl]-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
(2S,3R)-2-[({[2-(4-chlorophenyl)ethyl]carbamoyl}methyl)amino]-3-hydroxybutanamide
7-[(2-fluoro-5-methoxyphenyl)methyl]-2-(2-methylfuran-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
N-[(3R,4S)-1-(carbamoylmethyl)-4-cyclopropylpyrrolidin-3-yl]-2-(2-chloro-6-fluorophenyl)acetamide
1-[3-(3-fluorophenyl)-1H-pyrazole-4-carbonyl]-4-(pyrimidin-2-yl)-1,4-diazepane
2-methoxy-1-[4-(3-phenylpiperazine-1-carbonyl)piperidin-1-yl]ethan-1-one
N-(3-carbamoyl-4-fluorophenyl)-4-[(2-methyl-1H-imidazol-1-yl)methyl]piperidine-1-carboxamide
3-[(3-cyclohexyl-1,2,4-oxadiazol-5-yl)methyl]-1λ6-thiolane-1,1-dione
4-{[2-(2-fluoro-5-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazine-1-sulfonamide
5-[2,2-bis(prop-2-en-1-yl)pyrrolidine-1-carbonyl]-3,4-dihydropyrimidin-4-one
(1S,6R)-9-(5-fluoro-1-methyl-1H-indole-2-carbonyl)-3,9-diazabicyclo[4.2.1]nonane
4-benzyl-1-[(3,5-difluorophenyl)methyl]-3-(piperidin-4-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[3-(1H-imidazol-1-yl)propyl]-1-{2-methylthieno[2,3-d]pyrimidin-4-yl}piperidin-4-amine
N-[2-(piperidin-1-yl)ethyl]-1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
1-{4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepane-1-carbonyl}cyclopropane-1-carboxamide
N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-2-(pyridin-3-yl)pyrimidine-5-carboxamide
2-cyclopentyl-N-[2-(4-methyl-5-{[2-(morpholin-4-yl)ethyl]sulfanyl}-4H-1,2,4-triazol-3-yl)ethyl]acetamide
3-{1-methyl-3-phenyl-1,8-diazaspiro[4.5]decan-8-yl}propanoic acid
N-[3-(morpholin-4-yl)propyl]-3-propyl-1H-pyrazole-5-carboxamide
4-{5-[2-methyl-5-(propan-2-yl)furan-3-carbonyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carbonyl}morpholine
1-(4-{5-[(dimethylamino)methyl]-4-ethyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-4,4,4-trifluorobutan-1-one
(2E)-1-(3-{2-[(2-methoxyethyl)sulfanyl]-5-(3-methoxyphenyl)pyrimidin-4-yl}piperidin-1-yl)-3-(thiophen-2-yl)prop-2-en-1-one
4-[1-(2-methoxyethyl)-6-oxopiperidine-3-carbonyl]-1-(4-methylphenyl)piperazin-2-one
(2R,3R)-3-{2-azaspiro[4.4]nonan-2-yl}-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
N-[2-(dimethylamino)-5,6,7,8-tetrahydroquinazolin-5-yl]-2-(1H-1,2,4-triazol-1-yl)acetamide
2-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)-N-(pentan-3-yl)-N-(2-phenylethyl)acetamide
5-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}-N,N-dimethylpyridin-2-amine
1-[6-ethyl-2-(morpholin-4-yl)pyrimidin-4-yl]-N-(1H-pyrazol-3-ylmethyl)piperidin-4-amine
2-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-(5-fluoropyridin-3-yl)acetamide
1-(1-cyclopentanecarbonylpiperidine-4-carbonyl)-4-(pyridin-4-yl)piperazine
4-({2-benzyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl}methyl)-3,5-dimethyl-1-(propan-2-yl)-1H-pyrazole
N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}-2-(pyridin-2-yl)acetamide
(2S,4R)-4-amino-1-(3-{[(4-fluorophenyl)methyl]amino}benzoyl)-N-methylpyrrolidine-2-carboxamide
N-methyl-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-1,3-benzothiazole-2-carboxamide
dimethyl(3-{2-[1-(pyridin-4-yl)piperidin-4-yl]-1H-imidazol-1-yl}propyl)amine
2-{1-cyclohexyl-5-[(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)methyl]-1H-1,2,4-triazol-3-yl}acetamide
(1s,4s)-4-({methyl[2-(morpholin-4-yl)propyl]amino}methyl)cyclohexan-1-amine
5-oxo-1-{[2-(1H-pyrazol-1-yl)phenyl]methyl}pyrrolidine-3-carboxylic acid
2-{1-[(3,5-dimethoxyphenyl)methyl]-4-{[5-(2-methylpropyl)-1H-pyrazol-3-yl]methyl}piperazin-2-yl}ethan-1-ol
1-{[6-(2-ethylphenyl)pyridin-3-yl]methyl}-4-methylpiperazine
2-{1-[(4-ethoxyphenyl)methyl]-4-(pentan-3-yl)piperazin-2-yl}ethan-1-ol
N'-(3,5-dimethylphenyl)-N-[2-(2-oxo-1,3-oxazinan-3-yl)ethyl]propanediamide
(3S,4S)-1-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-4-(piperidin-1-yl)pyrrolidin-3-ol
3-amino-1-[(5-cyclopropyl-1-methyl-1H-pyrazol-4-yl)methyl]pyrrolidine-3-carboxylic acid