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N-ethyl-5-{1-[2-(4-methyl-4H-1,2,4-triazol-3-yl)ethyl]-1H-imidazol-2-yl}pyrimidin-2-amine
1-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-3-(3-methoxy-1,5-dimethyl-1H-pyrazol-4-yl)-1-methylurea
N-methyl-N-[(3-methylpyridin-4-yl)methyl]-1-(9H-purin-6-yl)piperidin-4-amine
3-({1-[3-(difluoromethoxy)benzoyl]pyrrolidin-3-yl}methyl)benzamide
5-(1H-pyrazol-1-ylmethyl)-N-{[2-(pyrrolidin-1-yl)-1,3-thiazol-4-yl]methyl}furan-2-carboxamide
(3S,4R)-1-(3,5-dimethylbenzoyl)-4-phenylpyrrolidine-3-carboxylic acid
2-[2-(cyclopropylcarbamoyl)ethyl]-N-(thiophen-2-ylmethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide
N-[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]-1-propanoylpyrrolidine-2-carboxamide
5-[4-(1-acetylpiperidine-3-carbonyl)piperazin-1-yl]-2-methyl-2,3-dihydropyridazin-3-one
1-{1-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]piperidin-3-yl}pyrrolidin-2-one
3-(5-cyclohexyl-1,3,4-oxadiazol-2-yl)-N-[2-(4-hydroxyphenyl)ethyl]propanamide
(1S,5R)-6-(3,5-difluoropyridine-2-carbonyl)-3-(pyridine-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
2-ethoxy-1-[7-(pyrrolidine-1-sulfonyl)-1,2,3,4-tetrahydroisoquinolin-2-yl]ethan-1-one
2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]-N-{5H,6H,7H,8H,9H,10H-cyclohepta[b]indol-2-ylmethyl}acetamide
1-{4-[3-(2-phenylethyl)-4H-1,2,4-triazol-4-yl]phenyl}ethan-1-one
2-(2,6-dimethoxy-4-methylphenyl)-5-[3-(methoxymethyl)piperidine-1-carbonyl]pyridine
N'-{2-[(2-chlorophenyl)formamido]ethyl}-N-(2-ethoxyphenyl)propanediamide
N-[4-(1H-indol-2-yl)phenyl]-1-(pyridine-3-carbonyl)piperidine-4-carboxamide
1-[(8-methoxy-3,4-dihydro-2H-1,5-benzodioxepin-7-yl)methyl]piperidine-3-carbonitrile
6-cyclopentyl-N-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-{[2-(1H-imidazol-1-yl)pyridin-3-yl]methyl}-5-methoxy-3-methyl-1H-indole-2-carboxamide
ethyl 2-({5-[2-amino-3-cyano-6-(1H-pyrrol-2-yl)pyridin-4-yl]pyrimidin-2-yl}amino)acetate
2-[2-(1H-imidazol-1-yl)ethyl]-1-{4H-thieno[3,2-b]pyrrole-5-carbonyl}piperidine
1-[2-fluoro-3-(trifluoromethyl)phenyl]-3-methyl-3-[(1,2,2-trimethylpyrrolidin-3-yl)methyl]urea
N-[2-fluoro-3-(trifluoromethyl)phenyl]-4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperidine-1-carboxamide
1-(4-methoxyphenyl)-5-(2-methyloxolan-2-yl)-3-(1H-1,2,4-triazol-1-ylmethyl)-1H-1,2,4-triazole
3-[(2,3-difluoro-4-methoxyphenyl)methyl]-1-[4-(2-methyl-5-oxopyrrolidin-1-yl)phenyl]urea
2-({[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}sulfamoyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
3-chloro-4-fluoro-N-[2-(5-methyl-1,3,4-thiadiazol-2-yl)ethyl]-1-benzothiophene-2-carboxamide
N-(3-{3-[2-(4-fluorophenyl)ethyl]piperidin-1-yl}-3-oxopropyl)methanesulfonamide
3-(3-fluoropyridin-4-yl)-2-methyl-6-(4H-1,2,4-triazol-4-yl)pyridine
5-{1-[(3E)-pent-3-enoyl]pyrrolidin-2-yl}-N-(1-propyl-1H-1,2,3-triazol-4-yl)thiophene-2-carboxamide
8-cyclopropanecarbonyl-2-[(4,6-dimethylpyrimidin-2-yl)methyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
8-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-1-[2-(4-methoxyphenyl)ethyl]-3-methyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-{[1-(dimethylsulfamoyl)pyrrolidin-3-yl]methyl}benzoic acid
(4aS,7aR)-1-(6-methylpyridine-3-carbonyl)-4-propyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-[4-(morpholin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]-1H-indole
2-{[4-(2-methanesulfonylethyl)piperazin-1-yl]methyl}-1H-1,3-benzodiazole
N-[(3S,7S,8aS)-3-methyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-4-(trifluoromethyl)benzamide
3-[2-(2-{[benzyl(methyl)amino]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl)-2-oxoethyl]-1,3-oxazolidin-2-one
2-methyl-N-{2-[3-(2-methylphenyl)pyrrolidin-1-yl]ethyl}pyrido[2,3-d]pyrimidin-4-amine
N-{[2-(1H-1,2,4-triazol-1-yl)pyridin-3-yl]methyl}-2,8-diazaspiro[4.5]decane-3-carboxamide
3,4-dimethoxy-2-{[3-(4-methoxy-3,5-dimethylbenzoyl)piperidin-1-yl]methyl}pyridine
5-(methoxymethyl)-N-[2-(1-phenyl-1H-pyrazol-4-yl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine
1-(3-chloro-4-methoxyphenyl)-4-(2,3-dihydro-1H-isoindole-2-carbonyl)pyrrolidin-2-one
1-{[4-methoxy-3-(methoxymethyl)phenyl]methyl}-3-(3-methoxybenzoyl)piperidine
2-methoxy-3-[4-(2-methoxybenzoyl)piperazin-1-yl]pyrazine
1-[(3S,4R)-3-[(dimethylsulfamoyl)amino]-4-(propan-2-yl)pyrrolidin-1-yl]-2-(pyridin-2-yl)ethan-1-one
N-(2-methylquinolin-8-yl)-4-(morpholine-4-carbonyl)piperidine-1-carboxamide
3-[({1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}amino)methyl]-1-(2,2-dimethylpropyl)-3-hydroxypiperidin-2-one