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1-methyl-4-{[methyl({[4-(2-methylpropyl)phenyl]methyl})amino]methyl}pyrrolidin-2-one
N-[3-(pyridin-2-yl)propyl]-2-(2,5,7-trimethyl-1H-indol-3-yl)acetamide
1-methanesulfonyl-N-[4-(3-methoxyphenyl)phenyl]piperidine-3-carboxamide
5-{1-[3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole-5-carbonyl]pyrrolidin-2-yl}thiophene-2-carboxamide
1-{1-[6-(morpholin-4-yl)pyrimidin-4-yl]piperidin-4-yl}pyrrolidin-2-one
1-[(2R)-2-(methoxymethyl)pyrrolidin-1-yl]-3-(4-methyl-1,3-thiazol-5-yl)propan-1-one
1-[4-(4-fluorophenyl)benzoyl]-4-methyl-1,4-diazepan-5-one
3-(2-methylphenyl)-5-{2-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]ethyl}-1,2,4-oxadiazole
(4-benzyl-1-{[4-(trifluoromethyl)phenyl]methyl}piperidin-4-yl)methanol
3-[(diethylamino)methyl]-1-[(3,4-difluorophenyl)methyl]-3-hydroxypiperidin-2-one
2-{9-[2-(4-fluorophenoxy)ethyl]-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl}propanoic acid
2-[3-(1H-imidazol-2-yl)piperidine-1-carbonyl]-5,7-dimethylquinolin-8-ol
1-[(1S,5R)-3-benzyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-methyl-2-(morpholin-4-yl)propan-1-one
N-[2-methoxy-1-(pyridin-2-yl)ethyl]-N-methyl-4-(1H-pyrazol-3-yl)benzamide
(1S,5R)-3-(2-hydroxypyridine-3-carbonyl)-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
[(3R,4R)-4-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-1-[5-(1H-imidazol-1-ylmethyl)furan-2-carbonyl]pyrrolidin-3-yl]methanol
methyl 4-(5-{[methyl(oxan-2-ylmethyl)amino]methyl}-1,2,4-oxadiazol-3-yl)benzoate
(3S,4R)-1-[(1-cyclohexyl-1H-imidazol-5-yl)methyl]-4-(2-methylphenyl)pyrrolidine-3-carboxylic acid
2-(1-{[3-(4-chlorophenyl)-1H-pyrazol-4-yl]methyl}piperidin-4-yl)-N-methylacetamide
2-methoxy-4-[3-(4-phenylpiperazin-1-yl)piperidine-1-carbonyl]quinoline
4-(1-{[2-(methoxymethyl)pyrimidin-5-yl]methyl}piperidin-4-yl)thiomorpholine
N-[3-chloro-4-(1H-1,2,4-triazol-1-yl)phenyl]-4,4-difluoropiperidine-1-carboxamide
1-cyclopropyl-5-[4-(2-fluorophenoxy)piperidine-1-carbonyl]piperidin-2-one
N-methyl-N-[(3-phenyl-1H-pyrazol-5-yl)methyl]-2-(1H-pyrazol-1-yl)butanamide
N-[2-(dimethyl-1H-1,2,4-triazol-1-yl)ethyl]-1-phenyl-1H-1,2,3-triazole-4-carboxamide
3-[4-(6-hydroxy-2-methylpyrimidin-4-yl)piperidine-1-carbonyl]-1-phenylpyrrolidin-2-one
N-{1-[1-(3-cyclopentylpropanoyl)piperidin-4-yl]-1H-pyrazol-5-yl}-2-methylbenzamide
2-{3-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}propane-1,3-diol
1-(1-methyl-1H-indole-4-carbonyl)azepan-4-amine
N-methyl-N-[3-(1-methyl-1H-pyrazol-4-yl)propyl]-2-(1,2,3,4-tetrahydroisoquinolin-2-yl)propanamide
3-(2-phenyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-1-[2-(1,3-thiazol-2-yl)piperidin-1-yl]propan-1-one
[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl][(2-ethyl-3-methyl-1H-indol-5-yl)methyl]amine
3-methoxy-N-{[7-(pyrimidin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}propanamide
(1R,2R,6S,7S)-4-(2-phenylquinolin-4-yl)-10-oxa-4-azatricyclo[5.2.1.02,6]decane
(1S,5R)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-[(2-ethyl-1,3-thiazol-4-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
3-(4-fluorophenyl)-4-(1H-imidazol-2-yl)-1-(4-methylphenyl)-1H-pyrazole
N-[(3S,5S)-5-(ethylcarbamoyl)-1-(4-fluorobenzoyl)pyrrolidin-3-yl]-1H-pyrrole-2-carboxamide
4-[4-(quinoxalin-5-ylmethyl)piperazin-1-yl]quinazoline
N-[(2R)-3,4-dihydro-2H-1-benzopyran-2-ylmethyl]-5-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]pyridin-2-amine
7-[2-hydroxy-3-(2-methylphenoxy)propanoyl]-2-methyl-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
methyl[3-(morpholin-4-yl)propyl][(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]amine
N-[(6-chloropyridin-3-yl)methyl]-1-(furan-2-ylmethyl)piperidine-3-carboxamide
2-({[5-(2-methylpropyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}amino)pyridine-3-carbonitrile
9-(2,4-dimethylpyrimidine-5-carbonyl)-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
5-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]-1-(3-phenylpropyl)piperidin-2-one
N-[(3R,4S)-1-(carbamoylmethyl)-4-(propan-2-yl)pyrrolidin-3-yl]-4-phenoxybutanamide
7-[(5-tert-butyl-1,2,4-oxadiazol-3-yl)methyl]-3-methyl-1-oxa-3,7-diazaspiro[4.5]decan-2-one
3-(3-methoxyphenoxy)-1-(2-phenylbenzoyl)azetidine
1-cyclohexyl-N3-(2,2-diphenylethyl)-N5-methyl-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
N-methyl-2-(morpholin-2-yl)-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}acetamide