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4-oxo-2-{[2-(trifluoromethyl)morpholin-4-yl]methyl}-1,4-dihydroquinoline-6-carboxamide
1-(3-{5-[(dimethylamino)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-2-phenoxyethan-1-one
2-{3-[2-(4-methylpiperidin-1-yl)-2-oxoethyl]morpholine-4-carbonyl}-1,4-dihydroquinolin-4-one
2-{4-[(2-methylphenyl)methyl]piperazine-1-carbonyl}thiophene-3-sulfonamide
2-(1-methyl-1H-imidazol-2-yl)-1-({3-[1-(4-methylphenyl)cyclopentyl]-1,2,4-oxadiazol-5-yl}methyl)piperidine
1-(2-{4-[1-(dimethylamino)ethyl]piperidin-1-yl}-2-oxoethyl)-4-methyl-1,2-dihydroquinolin-2-one
2-{2-[2-(pyridin-3-yl)-1,3-thiazol-4-yl]ethyl}-2,9-diazaspiro[5.5]undecan-3-one
6-methyl-2-(2-phenylethyl)-1-(pyridin-4-ylmethyl)-3-{1,3,3-trimethyl-6-azabicyclo[3.2.1]octane-6-carbonyl}-1,4-dihydropyridin-4-one
5-methyl-2-(methylamino)-N-{[1-(pyridin-4-ylmethyl)pyrrolidin-3-yl]methyl}benzamide
N4-[(2,5-dimethylphenyl)methyl]-1H-pyrazolo[3,4-d]pyrimidine-4,6-diamine
3,3-dimethyl-1-[(5-{[1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl)methyl]urea
4-[2-(2,5-dimethoxyphenyl)-1H-imidazol-1-yl]-2-methyl-4,5,6,7-tetrahydro-1,3-benzothiazole
4-[(2-ethylpyrimidin-4-yl)methyl]-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
3-{[(5-tert-butyl-2-hydroxyphenyl)methyl](ethyl)amino}-1λ6-thiolane-1,1-dione
1-{4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-hydroxy-2-(4-methoxyphenyl)ethan-1-one
[5-(1-{[3-(cyclopentyloxy)phenyl]methyl}piperidin-4-yl)-4-methyl-4H-1,2,4-triazol-3-yl]methanol
N-[(3R,4S)-4-cyclopropyl-1-methanesulfonylpyrrolidin-3-yl]-2-methyl-1H-pyrrole-3-carboxamide
3-(1H-indole-6-carbonyl)-7-methoxy-2,3,4,5-tetrahydro-1H-3-benzazepine
4-{4-ethyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}-1-(1,3-thiazol-2-ylmethyl)piperidine
1-(2-methylpropyl)-N-[2-(propan-2-yloxy)ethyl]-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
(4aR,7aS)-1-cyclobutanecarbonyl-4-(2-hydroxypyridine-3-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-(3-methoxyphenyl)-6-methylpyridine
2-ethyl-5-{4-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidine-1-carbonyl}pyrimidine
N-(2,1,3-benzoxadiazol-5-ylmethyl)-N-methyl-6-oxo-1-[3-(2-oxopyrrolidin-1-yl)propyl]piperidine-3-carboxamide
N-{2-[7-(9H-fluoren-2-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}-1-methylpiperidine-3-carboxamide
1-({[1-(4-methylpyridin-2-yl)propyl]carbamoyl}methyl)piperidine-4-carboxamide
4-{[3-ethyl-4-(propan-2-yl)piperazin-1-yl]methyl}-1,5-dimethyl-1H-pyrrole-2-carbonitrile
N-[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]-2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]acetamide
3-[2-oxo-2-(2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethyl]-4-{[3-(trifluoromethyl)phenyl]methyl}piperazin-2-one
2-(azepan-1-yl)-2-(2,5-dimethoxyphenyl)acetic acid
[(3R,4R)-4-[(dimethylamino)methyl]-1-[(8-fluoroquinolin-2-yl)methyl]pyrrolidin-3-yl]methanol
ethyl 4-{6-[4-(1H-indol-3-yl)butan-2-yl]-6-azaspiro[2.5]octane-1-carbonyl}piperazine-1-carboxylate
2-(2,6-dimethoxypyridine-3-carbonyl)-7-[(3-methoxyphenyl)methyl]-2,7-diazaspiro[4.5]decane
3-hydroxy-1-[(3-methoxyphenyl)methyl]-3-{[4-(prop-2-en-1-yl)piperazin-1-yl]methyl}piperidin-2-one
2-methoxy-4-({4-methyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}methyl)phenol
1-[(2,2-dimethyloxan-4-yl)methyl]-4-(4-ethyl-1H-pyrazol-5-yl)piperidine
2-methyl-N-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}-1,3-thiazole-4-carboxamide
1-{2-amino-3-ethyl-3H-imidazo[4,5-b]pyridine-6-carbonyl}-4-phenylpiperidin-4-ol
3-(4-{3,9-diazaspiro[5.5]undecan-3-ylmethyl}phenyl)prop-2-yn-1-ol
3-({3-[(1-methylpiperidin-4-yl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-2,3-dihydro-1H-isoindol-1-one
2-chloro-3-({cyclopentyl[(3-methylthiophen-2-yl)methyl]amino}methyl)-9-methyl-4H-pyrido[1,2-a]pyrimidin-4-one
4-[5-({3-[2-(methylsulfanyl)benzoyl]piperidin-1-yl}methyl)-1,3-thiazol-2-yl]morpholine
2-({[2-(2-fluoro-4-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)amino)-N-methylacetamide
1-[(2,6-difluorophenyl)methyl]-N-methyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-1H-1,2,3-triazole-4-carboxamide
1-(cyclohexylmethyl)-N-cyclopropyl-4-oxo-5-(4-phenylpiperazine-1-carbonyl)-1,4-dihydropyridine-3-carboxamide
4-[(4-methoxypyridin-2-yl)methyl]-1-methyl-2,3,4,5-tetrahydro-1H-1,4-benzodiazepine-2,5-dione
(3S,4R)-1-[3-(2-oxoazepan-1-yl)propanoyl]-4-(pyridin-3-yl)pyrrolidine-3-carboxylic acid
2-[3-(2-methoxyphenoxy)azetidin-1-yl]-4-(pyridin-3-yl)pyrimidine
[4-(oxan-2-ylmethyl)-1-(quinoxalin-2-yl)piperidin-4-yl]methanol
5-(2-chloro-4-methoxyphenoxymethyl)-N-(oxolan-2-ylmethyl)-1,2-oxazole-3-carboxamide