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7-acetamido-1-[(4-fluorophenyl)methyl]-N-[1-(1,3-thiazol-5-yl)propan-2-yl]-1H-1,3-benzodiazole-5-carboxamide
N-{1-[(2-chlorophenyl)methyl]-5-oxopyrrolidin-3-yl}but-3-enamide
5-{3-phenyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}-3-(propan-2-yl)-4,5-dihydro-1,2-oxazole
N-[3-(cyclohexylsulfanyl)propyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxamide
(3S,4S)-4-methyl-1-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}piperidine-3,4-diol
3-(4-methylphenyl)-3-phenyl-N-[3-(1H-1,2,4-triazol-1-yl)propyl]propanamide
4-methoxy-2-{[2-(3-methoxyphenyl)-2,3,4,5-tetrahydro-1,5-benzothiazepin-5-yl]methyl}phenol
5-(4-methoxyphenyl)-N-(3-phenylpropyl)-1,2,4-triazin-3-amine
N-methyl-4-[4-(morpholin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]-1,3-thiazol-2-amine
methyl({[5-methyl-2-(3-methylthiophen-2-yl)-1,3-oxazol-4-yl]methyl})(1H-pyrazol-3-ylmethyl)amine
(3,4-dihydro-2H-1,5-benzodioxepin-7-ylmethyl)[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl](2-methoxyethyl)amine
N-ethyl-N-(2-methylprop-2-en-1-yl)-1-(2-methylpropyl)-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
5-(2-{[2-(4-fluorophenoxy)ethyl]amino}ethyl)-1-(thiophen-2-ylmethyl)pyrrolidin-2-one
4-[3-cyclopentyl-1-(1-methylpiperidin-4-yl)-1H-1,2,4-triazol-5-yl]-2,6-dimethylpyrimidine
({4-[(dimethylamino)methyl]phenyl}methyl)(methyl){[2-(morpholin-4-yl)-1,3-thiazol-5-yl]methyl}amine
3-[(thian-4-yl)amino]-2-(thiophen-2-ylmethyl)propan-1-ol
2-[4-(1,3-benzothiazol-2-ylmethyl)-1-[(6-methylpyridin-2-yl)methyl]piperazin-2-yl]ethan-1-ol
(1S,9R)-11-[2-(2-aminoethyl)-5,6-dimethylthieno[2,3-d]pyrimidin-4-yl]-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-6-one
(4S)-1-[(3-chloro-5-fluoro-4-methoxyphenyl)methyl]-4-(methoxymethyl)-3,3-dimethylpiperidin-4-ol
6-[(2-fluorophenyl)methoxy]-1-(2-methylpropyl)-4-(pyridine-3-carbonyl)-1,4-diazepan-2-one
N-[(3-phenylphenyl)methyl]-2-(pyrrolidin-3-yl)acetamide
2-({2-amino-6-[4-(1H-1,2,3-benzotriazol-1-yl)piperidin-1-yl]pyrimidin-4-yl}amino)ethan-1-ol
4-[4-(2-methoxyethoxy)piperidin-1-yl]-1-[4-(1H-pyrazol-1-yl)phenyl]piperidine
ethyl 1-benzyl-5-(4-methyl-1,2,5-oxadiazole-3-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
4-{3-[(3aS,6aS)-1-methyl-octahydropyrrolo[3,4-b]pyrrole-5-carbonyl]phenyl}-2-methylbutan-2-ol
2-{2-[4-(1-methoxyethyl)phenyl]phenyl}ethan-1-amine
4-methoxy-3-(8-methoxyquinolin-5-yl)-N-methylbenzamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-3-(3-hydroxyquinoxalin-2-yl)-N-methylpropanamide
2-(2,5-dioxoimidazolidin-1-yl)-N-{[2-(2-fluorophenoxy)pyridin-3-yl]methyl}acetamide
3-ethoxy-N-[(2S)-oxolan-2-ylmethyl]-4-(prop-2-en-1-yloxy)benzamide
3-(2-{1-ethyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazin-2-yl}-2-oxoethyl)-3,4-dihydroquinazolin-4-one
(2S,4S)-4-amino-N,N-diethyl-1-[2-(2-oxopyrrolidin-1-yl)acetyl]pyrrolidine-2-carboxamide
(1S,5R)-3-(3-phenyl-1,2,4-oxadiazol-5-yl)-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
(2S,4S)-4-amino-1-[3-(1H-pyrrol-1-yl)benzoyl]pyrrolidine-2-carboxylic acid
2-[5-(1-aminoethyl)-4H-1,2,4-triazol-3-yl]-N-(2H-1,3-benzodioxol-5-ylmethyl)-N-(pentan-3-yl)acetamide
3-[(3R,4S)-1-(4-chloro-2-fluorobenzoyl)-4-(morpholin-4-yl)piperidin-3-yl]propan-1-ol
5-[4-(2-methoxyethyl)piperazine-1-carbonyl]-2-(3-phenylpropyl)-1,3-benzoxazole
N-(pentan-3-yl)-N-(2-phenylethyl)-6-(4H-1,2,4-triazol-4-yl)pyridine-3-carboxamide
N-({4-methoxy-3-[(3-methyloxetan-3-yl)methoxy]phenyl}methyl)-1-methyl-4-oxo-N-(oxolan-2-ylmethyl)-1,4-dihydroquinoline-3-carboxamide
4-(3-ethyl-5-methyl-1,2-oxazole-4-carbonyl)-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
2-amino-4-(7-methyl-2,3-dihydro-1,4-benzodioxin-6-yl)-6-(1H-pyrrol-2-yl)pyridine-3-carbonitrile
3-[(1-acetylpiperidin-4-yl)oxy]-4-methoxy-N-methyl-N-(2-phenoxyethyl)benzamide
N-[(4-{2-[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]ethoxy}-3-methoxyphenyl)methyl]-N-[(3S)-2-oxoazepan-3-yl]acetamide
3-[1-(4-chloro-1,5-dimethyl-1H-pyrazole-3-carbonyl)piperidin-3-yl]benzoic acid
N-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}-4-sulfamoylbenzamide
(3S,4S)-4-cyclopropyl-1-[4-(piperidin-1-ylmethyl)benzoyl]pyrrolidine-3-carboxylic acid
(3R,5R)-5-{4-[(2E)-3-phenylprop-2-en-1-yl]piperazine-1-carbonyl}pyrrolidin-3-ol
N-[3-(1H-1,2,4-triazol-1-yl)phenyl]-9-oxa-2-azaspiro[5.5]undecane-2-carboxamide
(2S,4S)-4-amino-N-ethyl-1-[(2-hydroxy-7-methylquinolin-3-yl)methyl]pyrrolidine-2-carboxamide
(4aR,8aR)-7-(4,6-dimethoxypyrimidin-2-yl)-4a-hydroxy-N,N-dimethyl-decahydro-2,7-naphthyridine-2-carboxamide