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4-[(4-methoxyphenyl)methyl]-3-(pyridin-3-ylmethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
5-({[1-(1H-imidazol-1-yl)propan-2-yl]amino}methyl)-1,3-dimethyl-2,3-dihydro-1H-1,3-benzodiazol-2-one
N-{2-[2-(4-methanesulfonylphenyl)-1H-imidazol-1-yl]ethyl}-3-methylpyridin-4-amine
6-butyl-2-[3-({methyl[1-(pyridin-3-yl)ethyl]amino}methyl)phenyl]-3,4-dihydropyrimidin-4-one
3-cyclopropyl-1-methyl-5-[2-(prop-2-en-1-yloxy)phenyl]-1H,4H-pyrazolo[3,4-d]imidazole
3-({1-[1-(methoxymethyl)cyclobutanecarbonyl]pyrrolidin-3-yl}methyl)benzoic acid
3-{1-[5-(2-methylpropyl)-1,2-oxazole-3-carbonyl]piperidin-4-yl}-1-(morpholin-4-yl)propan-1-one
4-{3-[3-(3,5-dimethyl-1H-pyrazol-1-yl)azetidine-1-carbonyl]phenyl}-4H-1,2,4-triazole
butyl N-[(3S,5S)-1-methyl-5-(morpholine-4-carbonyl)pyrrolidin-3-yl]carbamate
N-methyl-N-{[3-(methylsulfanyl)phenyl]methyl}-2-(2-oxoazepan-1-yl)acetamide
2-{[3-(hydroxymethyl)-3-(3-methoxypropyl)piperidin-1-yl]sulfonyl}benzonitrile
(4S)-4-hydroxy-4-(methoxymethyl)-3,3-dimethyl-N-(4-phenoxyphenyl)piperidine-1-carboxamide
4-{[2-(3-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}morpholine
N-[(3R)-4-hydroxy-3-methylbutyl]-4-[(2-methylprop-2-en-1-yl)oxy]benzamide
(3R,4S)-1-[4-chloro-1-methyl-3-(trifluoromethyl)-1H-pyrazole-5-carbonyl]-3,4-dimethylpiperidin-4-ol
1-[4-(1H-imidazol-1-yl)benzoyl]-4-[(3-methylphenyl)methyl]piperazine
[(3,5-dimethoxyphenyl)methyl]({[1-(2-methoxyethyl)piperidin-4-yl]methyl})(oxolan-2-ylmethyl)amine
[1-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)-3-(3-methoxypropyl)piperidin-3-yl]methanol
1-[1-(difluoromethyl)-1H-pyrazole-5-carbonyl]-3-(3-methylphenoxymethyl)piperidine
2-{5-[6-(1-hydroxyethyl)pyridin-2-yl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-1-yl}ethan-1-ol
4-[5-methoxy-2-(pyrrolidine-1-carbonyl)phenoxy]-1-[3-(1H-pyrazol-1-yl)propyl]piperidine
2-(2-methoxyethyl)-8-{5-[(methylsulfanyl)methyl]pyridin-2-yl}-2,8-diazaspiro[5.5]undecan-3-one
4-(1H-pyrazol-4-yl)-N-{2-[(2S)-pyrrolidin-2-yl]ethyl}butanamide
4-({2-[3-(dimethylamino)-2-hydroxypropoxy]-5-methoxyphenyl}methyl)-N,N-dimethylpiperazine-1-carboxamide
2-[1-(2-methoxyethyl)-1H-imidazol-5-yl]-7,7-dimethyl-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
6-cyano-N-[3-(furan-2-yl)propyl]pyridine-3-carboxamide
(5S)-5-{3-oxo-3-[4-(4H-1,2,4-triazol-3-yl)piperidin-1-yl]propyl}imidazolidine-2,4-dione
(1R,2R,6S,7S)-4-(1-ethyl-1H-pyrazole-3-carbonyl)-4-azatricyclo[5.2.1.02,6]decane
N2,N2-dimethyl-N4-[1-phenyl-2-(1H-pyrazol-1-yl)ethyl]-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-2,4-diamine
1-(2-{1-[2-amino-6-(morpholin-4-yl)pyrimidin-4-yl]piperidin-4-yl}ethyl)pyrrolidin-2-one
(2S,4S)-4-{[(2-methoxynaphthalen-1-yl)methyl]amino}-1-[(2E)-3-phenylprop-2-en-1-yl]-N-(pyridin-3-ylmethyl)pyrrolidine-2-carboxamide
1-(butan-2-yl)-N3-[3-(dimethylamino)-2,2-dimethylpropyl]-N5-(furan-2-ylmethyl)-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
2-{3-[(3,4-dimethoxyphenyl)methyl]-5-(1-methyl-1H-pyrazol-4-yl)-1H-1,2,4-triazol-1-yl}acetic acid
3-(3-methoxyphenyl)-N-[3-(4-methyl-1H-pyrazol-1-yl)propyl]-1H-pyrazole-5-carboxamide
2-[({5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}(methyl)amino)methyl]-3,4-dihydroquinazolin-4-one
1-benzoyl-3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine
2-[4-(1,2,3,4-tetrahydroisoquinolin-5-yl)phenoxy]acetamide
4-(7-{[ethyl(pyridin-4-ylmethyl)amino]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carbonyl)-1-(prop-2-en-1-yl)pyrrolidin-2-one
2-(2H-1,2,3-benzotriazol-2-yl)-N-[(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)methyl]acetamide
N-[(3R,5S)-5-(diethylcarbamoyl)-1-(furan-3-carbonyl)pyrrolidin-3-yl]-1H-pyrrole-3-carboxamide
8-(2-methanesulfonylacetyl)-2-(2-phenylethyl)-2,8-diazaspiro[5.5]undecan-3-one
2-(5-ethyl-1-benzofuran-3-yl)-1-[(2R)-2-(methoxymethyl)pyrrolidin-1-yl]ethan-1-one
1-[3-(2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazol-1-yl)phenyl]imidazolidin-2-one
methyl[(5-{[(2-methylphenyl)methyl]sulfanyl}-4-(oxolan-2-ylmethyl)-4H-1,2,4-triazol-3-yl)methyl]{[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}amine
1-(1-{[2-(cyclopentylmethyl)-1H-imidazol-4-yl]methyl}piperidin-4-yl)-3-methylbutan-1-ol
5-({3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)-1H-indole
methyl[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]{[5-methyl-2-(3-methylthiophen-2-yl)-1,3-oxazol-4-yl]methyl}amine
2-(2-{4-[2-(dimethylamino)ethoxy]piperidin-1-yl}pyrimidin-4-yl)pyridine-4-carboxylic acid
1-[2-(4-fluorobenzenesulfonyl)ethyl]-2-(4-methylphenyl)-1H-imidazole
2-[(5-methylpyrazin-2-yl)methyl]-8-(pyridine-2-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one