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4-ethyl-2-methyl-5-[2-methyl-4-(pyrrolidin-1-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]-1,3-thiazole
1-cyclohexyl-4-(1H-imidazol-4-ylmethyl)piperazin-2-one
N-[2-(1H-1,3-benzodiazol-2-yl)ethyl]-1-(methoxymethyl)cyclobutane-1-carboxamide
1-{2-[(5-ethyl-2-methylpyrimidin-4-yl)amino]ethyl}piperidin-4-ol
N-{2-[3-(hydroxymethyl)piperidin-1-yl]ethyl}-2,3-dimethyl-1H-indole-7-carboxamide
(3R,4R)-3-methyl-1-[2-(3-methylphenyl)benzoyl]-4-(oxan-4-yl)piperidin-4-ol
(1S,5R)-3-(2-methylquinolin-4-yl)-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
(1R,3S)-3-[2-(dimethylamino)ethoxy]-7-[6-(dimethylamino)pyrazin-2-yl]-7-azaspiro[3.5]nonan-1-ol
1-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carbonyl}-4-(3-phenyl-1,2,4-oxadiazol-5-yl)piperidine
3-ethyl-1-{2-[4-(2-oxoimidazolidin-1-yl)phenyl]acetyl}piperidine-3-carboxylic acid
3-{2-[3-(2-ethylphenoxy)azetidin-1-yl]-2-oxoethyl}-1λ6-thiolane-1,1-dione
5-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-N-methyl-N-[1-(thiophen-2-yl)ethyl]-1H-pyrazole-3-carboxamide
3-methoxy-5-methyl-N-(propan-2-yl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]thiophene-2-carboxamide
2-ethyl-5-[4-methoxy-3-(4H-1,2,4-triazol-4-yl)phenyl]-1,3,4-oxadiazole
methyl({2-phenylimidazo[1,2-a]pyrimidin-3-yl}methyl)[1-(pyridin-2-yl)propan-2-yl]amine
3-(1H-1,3-benzodiazol-1-yl)-1-{3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}propan-1-one
9-(5-ethyl-1H-pyrrole-2-carbonyl)-2-(3-hydroxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
(3R,4S)-4-(propan-2-yl)-1-(5-propyl-1,3,4-thiadiazol-2-yl)pyrrolidin-3-amine
2,3,5,6-tetramethyl-N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}benzamide
4-{1-[2-(1H-imidazol-1-yl)ethyl]-1H-imidazol-2-yl}pyridine
N-[(3-benzyl-1,2,4-oxadiazol-5-yl)methyl]-1-(4-fluorophenyl)cyclopropane-1-carboxamide
2-(4-acetylphenoxy)-1-[(3S,4R)-3-(dimethylamino)-4-propylpyrrolidin-1-yl]ethan-1-one
(7-{1-[(4-methoxyphenyl)methyl]-1H-pyrazol-4-yl}-2,3-dihydro-1-benzofuran-2-yl)methanamine
2-benzyl-9-[3-(pyridin-3-yl)propyl]-2,9-diazaspiro[5.5]undecan-3-one
N4,N4,5-trimethyl-N2-[1-(pyridin-3-yl)propan-2-yl]pyrimidine-2,4-diamine
N-(2-methylpropyl)-1-[1-(6-methylpyridazin-3-yl)piperidin-4-yl]-1H-1,2,3-triazole-4-carboxamide
N-(1-benzyl-3-methyl-1H-pyrazol-5-yl)-4-(2-oxo-1,3-oxazolidin-3-yl)piperidine-1-carboxamide
5-[4-(2-methoxyphenyl)-3,3-dimethylpiperazine-1-carbonyl]-2-(pyridin-3-yl)pyrimidine
1-(2,3-dihydro-1H-inden-2-yl)-4-{6-methylpyrazolo[1,5-a]pyrimidine-3-carbonyl}-1,4-diazepane
3-(4-fluorophenyl)-4-{1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-ylmethyl}-1H-pyrazole
N-[(4,6-dimethylpyrimidin-2-yl)methyl]-2-(2-methyl-1,3-thiazol-4-yl)acetamide
1-{3-[(dimethylamino)methyl]-3-hydroxypyrrolidin-1-yl}-3-[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]propan-1-one
(3R,4S)-1-[1-(4-methoxyphenyl)cyclopentanecarbonyl]-4-(5-methylfuran-2-yl)pyrrolidin-3-amine
1-{[3-(2-fluorophenyl)-1-methyl-1H-pyrazol-4-yl]methyl}-4-(pyridin-3-ylmethyl)piperazine
1-{2-methoxy-4-[({2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}amino)methyl]phenoxy}-3-[methyl(propan-2-yl)amino]propan-2-ol
(1R,5R)-3-(3-methylbenzoyl)-6-propyl-3,6-diazabicyclo[3.2.2]nonane
N-benzyl-1-[3-(3-methoxyphenyl)-1H-pyrazole-4-carbonyl]-N-methylpiperidin-3-amine
1-{2-[(3S,4R)-3-hydroxy-4-(3-methylthiophen-2-yl)piperidin-1-yl]-2-oxoethyl}-1,2,3,6-tetrahydropyridazine-3,6-dione
2-cyclohexyl-5-{[2-(4-fluorophenyl)azetidin-1-yl]methyl}pyrimidine
10-methoxy-5-(oxolane-2-carbonyl)-3,4,5,6-tetrahydro-2H-1,5-benzoxazocine
3-(2-{1-[2-(methylamino)-1,3-thiazole-4-carbonyl]piperidin-2-yl}ethyl)phenol
N-[1-(3-phenylpropyl)piperidin-3-yl]pyridine-3-sulfonamide
5-(1H-1,3-benzodiazol-1-ylmethyl)-N-{[1-(propan-2-yl)-1H-imidazol-2-yl]methyl}-1H-pyrazole-3-carboxamide
1-(5-propylpyrimidin-4-yl)-N-[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]piperidin-4-amine
5-{4-[(3-fluorophenyl)methyl]piperazine-1-carbonyl}isoquinoline
5-{2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-ylmethyl}-2-(thiophen-2-yl)pyrimidine
(3R,4R)-4-(2-ethyl-4-methyl-1H-imidazol-5-yl)-1-methyl-N-(pyridin-3-yl)pyrrolidine-3-carboxamide
(3S,4R)-1-[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]-4-(2-methoxyphenyl)pyrrolidine-3-carboxylic acid
N-[2-(5-methyl-4-{[methyl({[1-(pyridin-3-yl)-1H-pyrrol-2-yl]methyl})amino]methyl}-1,3-oxazol-2-yl)phenyl]thiophene-3-carboxamide
1-[(4aR,8aS)-1-{5,7-dimethylpyrazolo[1,5-a]pyrimidine-2-carbonyl}-decahydro-1,6-naphthyridin-6-yl]-2-(3-fluorophenyl)ethan-1-one