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ethyl 3-(3-phenylpropyl)-1-(1,3-thiazol-2-ylmethyl)piperidine-3-carboxylate
N-{[5-(furan-2-yl)-1,2-oxazol-3-yl]methyl}-2-(2-oxo-1,3-oxazolidin-3-yl)acetamide
7-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)ethyl]-2-oxa-7-azaspiro[4.5]decan-8-one
N-[(1-ethyl-5-methyl-1H-pyrazol-4-yl)methyl]-N-methyl-3-[(2-methylprop-2-en-1-yl)oxy]benzamide
2-[2-(1-ethylpiperidin-4-yl)-N-methylacetamido]-2-(pyridin-3-yl)acetic acid
5-methyl-N-(1,2,3,4-tetrahydronaphthalen-2-yl)pyrazolo[1,5-a]pyrimidin-7-amine
N-cyclopropyl-5-{[(4-fluorophenyl)carbamoyl]carbonyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
4-{2-[(3-fluorophenyl)methyl]morpholine-4-carbonyl}-1-methyl-1,2-dihydroquinolin-2-one
3-(2-butyl-2,5-dihydro-1H-pyrrole-1-carbonyl)-5-(2,4-difluorophenoxymethyl)-1,2-oxazole
(2R,6R)-4-[2-(3,5-dimethyl-1H-pyrazol-1-yl)acetyl]-10-methoxy-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
N-({7-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-5-(methoxymethyl)furan-2-carboxamide
5-(4-chloro-3-fluorobenzoyl)-2-(3-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
6-[3-(dimethylamino)-2,2-dimethylpropyl]-2-methyl-2H,6H,7H-pyrazolo[4,3-d]pyrimidin-7-one
3-(1,3-benzothiazol-2-yl)-N-[3-(1H-1,2,3-benzotriazol-1-yl)propyl]propanamide
3-[(dimethylamino)methyl]-1-(1H-indole-7-carbonyl)piperidin-3-ol
3-methyl-N-[7-oxo-5-(2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carbonyl)-4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl]benzamide
5-methyl-3-{2-[4-(2-phenylpropyl)-1H-1,2,3-triazol-1-yl]ethyl}-1,2,4-oxadiazole
9-[(2-ethylpyrimidin-5-yl)methyl]-2-[(5-methylpyrazin-2-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
methyl 4-{4-[3-(4H-1,2,4-triazol-4-yl)propanoyl]piperazin-1-yl}benzoate
3-{[(cyclohexylmethyl)amino]methyl}-1-(2,2-dimethylpropyl)-3-hydroxypiperidin-2-one
3-[5-(pyridin-3-ylmethyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]-1-(pyrrolidin-1-yl)propan-1-one
N-(2,3-dihydro-1H-inden-4-yl)-3-(pyridin-3-yl)azetidine-1-carboxamide
5-ethoxy-N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]furan-2-carboxamide
N-(2-methoxyethyl)-3-{1-[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}propanamide
(2S,4R)-4-amino-1-[2-(benzyloxy)ethyl]-N-methylpyrrolidine-2-carboxamide
1-({[1-(2-chlorophenyl)cyclopropyl]carbamoyl}methyl)piperidine-4-carboxamide
N-(3-methoxypropyl)-N-{[6-(2-methylphenyl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}-2-(thiophen-3-yl)acetamide
2-cyclopropyl-4-(3,4-diethoxyphenyl)-1H-imidazole
1-[(1S,5R)-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]-3-(trimethyl-1H-pyrazol-4-yl)propan-1-one
1-[2-(dimethylamino)-4-{[(4-hydroxy-1-methylpiperidin-4-yl)methyl]amino}-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]ethan-1-one
1-[1-(2,2-dimethylpropyl)-5-oxopyrrolidin-3-yl]-3-ethylurea
ethyl 3-[(2-methylphenyl)methyl]-1-(quinoxaline-6-carbonyl)piperidine-3-carboxylate
2-(4-methoxy-3-methylphenyl)-2-{methyl[(trimethyl-1H-pyrazol-4-yl)methyl]amino}acetic acid
{[2-(6-chloro-2H-1,3-benzodioxol-5-yl)-5-methyl-1,3-oxazol-4-yl]methyl}[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl]methylamine
2-(2-{[(butan-2-yl)(thiophen-3-ylmethyl)amino]methyl}phenoxy)acetamide
N-[1-(1-methyl-1H-pyrazol-4-yl)ethyl]-1-[3-(2-methylpyrimidin-4-yl)phenyl]piperidin-4-amine
N-(2-methoxyethyl)-3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)-N-[(4-methylphenyl)methyl]propanamide
N-(2-methoxyethyl)-6-oxo-1-(2-phenylethyl)-N-(propan-2-yl)piperidine-3-carboxamide
2-(azepan-1-yl)-N-{2-[(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)amino]ethyl}acetamide
1-[(4-fluorophenyl)methyl]-4-[(thian-4-yl)amino]pyrrolidin-2-one
1-{2-[(1S,5R)-3-[(4-methyl-1H-imidazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]phenyl}ethan-1-one
N-methyl-N-[1-(5-{[(6-methylpyridin-3-yl)oxy]methyl}-1,2-oxazole-3-carbonyl)pyrrolidin-3-yl]acetamide
2-methyl-4-{4-[4-(thiomorpholin-4-yl)piperidine-1-carbonyl]phenyl}butan-2-ol
2-cyclopropyl-9-[5-(propan-2-yl)-1,3,4-thiadiazol-2-yl]-2,9-diazaspiro[5.5]undecan-3-one
1-{1-[2-(4-methoxyphenyl)acetyl]piperidin-3-yl}-N-(2-methylpropyl)-1H-1,2,3-triazole-4-carboxamide
3-ethyl-6-[6-(methylsulfanyl)-1,2,3,4-tetrahydroisoquinoline-2-carbonyl]-3H-imidazo[4,5-b]pyridin-2-amine
4-(1-acetylpiperidine-4-carbonyl)-1-(4-methylphenyl)piperazin-2-one
2-(4-{[4-(pyridin-3-yl)piperazin-1-yl]methyl}phenoxy)acetic acid
{3-[(2-fluorophenyl)methyl]-1-(2,7,8-trimethylquinoline-4-carbonyl)piperidin-3-yl}methanol
2-[1-({1-[(1,2-dimethyl-1H-imidazol-5-yl)methyl]piperidin-3-yl}methyl)-1H-1,2,3-triazol-4-yl]pyridine