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N-(2-{4-[(2-fluorophenyl)methyl]morpholin-2-yl}ethyl)-2,2-dimethylpropanamide
N-[(4-chlorophenyl)(pyridin-4-yl)methyl]-1-[4-(morpholine-4-carbonyl)phenyl]piperidin-4-amine
methyl 4-[2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)acetyl]piperazine-1-carboxylate
4-methyl-2-(propan-2-yl)-6-(1H-pyrazol-3-yl)pyrimidine
(3S,4R)-4-(3-fluorophenyl)-1-(1-methyl-1H-pyrrole-2-carbonyl)pyrrolidine-3-carboxylic acid
4-(1-benzothiophene-5-carbonyl)-1,4-oxazepan-6-ol
1-[4-({methyl[1-(pyrimidin-4-yl)ethyl]amino}methyl)thiophen-2-yl]ethan-1-one
6-(3-carbamoylpiperidin-1-yl)-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}pyridine-3-carboxamide
1-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-N-(oxan-3-ylmethyl)piperidin-4-amine
4-{5-[(dimethylamino)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}-N-[(4-methylphenyl)methyl]piperidine-1-carboxamide
N-[3-(5-methyl-2H-1,2,3,4-tetrazol-2-yl)adamantan-1-yl]furan-3-carboxamide
4-(1-benzofuran-5-ylmethyl)-1-[(3-methoxyphenyl)methyl]piperazin-2-one
methyl 3-{6-[(3-methoxyphenyl)methoxy]-2-oxo-4-[3-(pyridin-4-yl)propanoyl]-1,4-diazepan-1-yl}propanoate
2-[4-(1-{3,5-diazatricyclo[9.4.0.02,7]pentadeca-1(11),2(7),3,5,12,14-hexaen-4-yl}-5-methyl-1H-pyrazole-4-carbonyl)piperazin-1-yl]phenol
1-[4-(4-fluoropiperidin-1-yl)-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]ethan-1-one
2-[2-({3-[2-(4-fluorophenyl)ethyl]piperidin-1-yl}methyl)phenoxy]ethan-1-ol
6-chloro-2-{[3-(2-hydroxyethyl)-4-methylpiperazin-1-yl]methyl}-1,4-dihydroquinolin-4-one
11-[(3-chloro-4-ethoxyphenyl)methyl]-7-methyl-3,7,11-triazaspiro[5.6]dodecane
9-(6-ethylpyrimidin-4-yl)-3-oxa-9-azaspiro[5.5]undecane
1-[3-(methylsulfanyl)propyl]-8-(quinoxalin-2-yl)-1,8-diazaspiro[4.5]decane
methyl 5-[(oxan-4-yl)amino]-3-(oxolane-2-amido)-1-(2-phenylethyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N-[(3-ethyl-1,2-oxazol-5-yl)methyl]-1-(2-methoxyphenyl)-N-methyl-1H-pyrazole-4-carboxamide
N-cyclohexyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxamide
2-(1,1-dioxo-1λ6-thian-4-yl)-N-methyl-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]acetamide
6-[({6-cyclopentyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)methyl]-2-methylpyrimidin-4-ol
1-(furan-2-ylmethyl)-N-{2-[2-(propan-2-yl)-1,3-thiazol-4-yl]ethyl}piperidine-4-carboxamide
N-{1-[4-(3-methoxypropyl)-4H-1,2,4-triazol-3-yl]ethyl}-N'-(2-methylphenyl)propanediamide
2-({[1-(1H-pyrazole-4-carbonyl)piperidin-4-yl]oxy}methyl)pyridine
2-ethoxy-4-{5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepin-8-ylmethyl}phenol
N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-3-(dimethylamino)-2-methylpropanamide
(1R,2R,4R)-N-(isoquinolin-5-ylmethyl)-N-methylbicyclo[2.2.1]hept-5-ene-2-carboxamide
5-[(1R,5R)-6-(cyclobutylmethyl)-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]-1H-1,2,3-benzotriazole
1-(2-methoxyacetyl)-N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}piperidine-4-carboxamide
4-[(2E)-3,7-dimethylocta-2,6-dien-1-yl]-1-methyl-2,3,4,5-tetrahydro-1H-1,4-benzodiazepine-2,5-dione
N-{1-[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]ethyl}-2-(pyridin-3-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-amine
[(3R,4R)-4-({[2-(dimethylamino)ethyl](methyl)amino}methyl)-1-(3-methoxy-4-methylbenzoyl)pyrrolidin-3-yl]methanol
3,5-dimethyl-1-[1-(thiophen-3-ylmethyl)pyrrolidin-3-yl]-1H-pyrazole
N-[(2S)-oxolan-2-ylmethyl]-5-[4-(2-phenylethyl)piperidine-1-carbonyl]pyridin-2-amine
3-methyl-N-{2-[({2-[(2-methylprop-2-en-1-yl)oxy]phenyl}methyl)amino]ethyl}pyridin-2-amine
1-(4-methylpiperidin-1-yl)-3-[(3S,4R)-4-(morpholin-4-yl)-1-(pyridin-4-ylmethyl)piperidin-3-yl]propan-1-one
1-(cyclopropylmethyl)-4-(3-methoxypyridine-2-carbonyl)-2-(propan-2-yl)-1,4-diazepane
4-chloro-1-ethyl-N-{[2-(2-fluorophenoxy)pyridin-3-yl]methyl}-1H-pyrazole-5-carboxamide
5-{[benzyl(methyl)amino]methyl}-N-[2-(pyrazin-2-yl)ethyl]-1,2-oxazole-3-carboxamide
N-[2-methoxy-2-(thiophen-2-yl)ethyl]-2,3-dihydro-1H-inden-2-amine
4-methyl-6-(4-{[4-(oxolan-2-yl)butyl]amino}piperidin-1-yl)pyrimidin-2-amine
3,3-diphenyl-1-(1,3-thiazol-4-ylmethyl)piperidine
3-(3,5-dimethylphenyl)-N-[2-(N-methylmethanesulfonamido)ethyl]propanamide
1'-(2-ethyl-4-methyl-1,3-oxazole-5-carbonyl)-5-propyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
3-({3-[(2H-1,3-benzodioxol-5-yl)amino]piperidin-1-yl}methyl)-4H-chromen-4-one
N-[(1-ethylpyrrolidin-2-yl)methyl]-3-[1-(4-methyl-1,3-oxazole-5-carbonyl)piperidin-4-yl]propanamide