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7-(6,7-dimethoxy-4-methylquinolin-2-yl)-4-(3-fluorobenzoyl)-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepine
4-hydroxy-N-({1-[(2-methyl-1H-imidazol-1-yl)methyl]cyclopropyl}methyl)-2-(thiophen-2-yl)pyrimidine-5-carboxamide
4-(cyclopropylmethyl)-1-(2-methoxypyridine-4-carbonyl)-3-(propan-2-yl)-1,4-diazepan-5-one
2-[(dimethyl-1,2-oxazol-4-yl)methyl]-8-(4-methyl-1,3-thiazole-5-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
2-[(4-chlorophenyl)methyl]-N,N-dimethyl-3-oxo-2,8-diazaspiro[4.5]decane-8-sulfonamide
3-(2H-1,3-benzodioxol-5-yl)-1-benzyl-4-{[3-(methoxymethyl)pyrrolidin-1-yl]methyl}-1H-pyrazole
2-[3-(3-ethoxyphenyl)-1H-indazol-1-yl]-N-(2-methyl-2H-1,2,3-triazol-4-yl)acetamide
3-benzyl-4-[3-(4,5,6,7-tetrahydro-1H-indazol-3-yl)propanoyl]piperazin-2-one
2,3-dimethyl-5-[3-(1-methyl-1H-imidazol-2-yl)piperidine-1-carbonyl]benzene-1-sulfonamide
2-(5-acetylthiophen-3-yl)-N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}acetamide
2-methyl-1-(1-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}piperidin-4-yl)propan-1-ol
2-(6-methoxy-1H-1,3-benzodiazol-2-yl)-7,7-dimethyl-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
(4aS,7aR)-1-[2-(2-chloro-4-fluorophenyl)acetyl]-4-ethyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-benzyl-N-methyl-2-{[(1,2-oxazol-3-ylmethyl)amino]methyl}-2,3-dihydro-1H-inden-2-amine
5-{[3-(3-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}-1,3-oxazolidin-2-one
4-{[2-(2-fluoro-4-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazin-2-one
5-ethyl-1'-(2-methoxy-4-methylbenzoyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
(5-{[1-(4-methoxy-3-methylphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}furan-2-yl)methanol
methyl 4-({1-[2-(azocan-1-yl)-4-methylpyrimidin-5-yl]ethyl}carbamoyl)butanoate
4-{1-[1-(4-methoxyphenyl)cyclopentanecarbonyl]piperidin-3-yl}pyrimidine
3-[(2E)-3-phenylprop-2-en-1-yl]-3,9-diazaspiro[5.6]dodecan-10-one
2-[(1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]-N,N-diethylacetamide
5-methoxy-9-[6-(1-methyl-1H-imidazol-2-yl)pyridazin-3-yl]-1-oxa-9-azaspiro[5.5]undecane
{[1-(4-chlorophenyl)-1H-pyrazol-4-yl]methyl}({1-[1-(3-fluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl})amine
N-{[1-(1-methylpiperidin-4-yl)piperidin-4-yl]methyl}-N-(pyridin-4-ylmethyl)thiophene-3-carboxamide
1-{1'-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}propan-1-one
4-[(2,4-dimethoxyphenyl)methyl]-3-[2-oxo-2-(pyrrolidin-1-yl)ethyl]piperazin-2-one
N-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-[1-(1H-pyrrole-3-carbonyl)piperidin-4-yl]propanamide
4-[1-(3,4-difluorophenyl)-3-(2-methoxyethyl)-1H-1,2,4-triazol-5-yl]pyridine
1-(4-methoxyphenyl)-5-methyl-4-[3-(prop-2-en-1-yloxy)benzoyl]piperazin-2-one
3-[(3R,4S)-1-(4-fluoro-3-methylbenzoyl)-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propanoic acid
3-[2-(1,3-benzothiazol-2-yl)pyrrolidine-1-carbonyl]-1-methyl-1,2,5,6,7,8-hexahydroquinolin-2-one
7-[(3,4-difluorophenyl)methyl]-2-(4-ethenylbenzoyl)-2,7-diazaspiro[4.5]decane
2,5-dimethyl-N-[(2S)-oxolan-2-ylmethyl]-1-phenyl-1H-pyrrole-3-carboxamide
1-{[2-(morpholin-4-yl)-1,3-thiazol-5-yl]methyl}-N-[4-(propan-2-yl)phenyl]piperidin-3-amine
5-ethyl-N-[1-(pyridin-2-ylmethyl)piperidin-4-yl]pyrimidin-2-amine
N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-2,3,4,9-tetrahydro-1H-carbazole-1-carboxamide
1-[5-(1-phenylcyclopropyl)-1H-1,2,4-triazol-1-yl]butan-2-ol
6-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
2-(3-fluorophenyl)-1-{4-[4-(2-hydroxypropan-2-yl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}ethan-1-one
7-(3-ethyl-1H-indole-2-carbonyl)-N,N-dimethyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
2-[(thiophen-3-ylmethyl)(4,4,4-trifluorobutyl)amino]butan-1-ol
(2S)-N-propyl-N-(pyridin-3-ylmethyl)pyrrolidine-2-carboxamide
5-chloro-N-cyclohexyl-4,6-dimethyl-2-oxo-N-(pyridin-2-ylmethyl)-1,2-dihydropyridine-3-carboxamide
[(2-fluorophenyl)methyl](2-methoxyethyl)(quinoxalin-2-ylmethyl)amine
2-(ethylamino)-N-[(3R,4S)-1-methanesulfonyl-4-(propan-2-yl)pyrrolidin-3-yl]pyrimidine-5-carboxamide
1-[(1-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carbonyl}pyrrolidin-2-yl)methyl]-1H-pyrazole
6-methoxy-N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
N-methyl-4-(4-methylphenyl)-N-[2-(1H-pyrazol-4-yl)ethyl]-5-(pyrimidin-5-yl)pyrimidin-2-amine
(2R,6R)-11-methoxy-4-[(1-propyl-1H-imidazol-2-yl)methyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid