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4-{imidazo[1,2-a]pyrimidine-2-carbonyl}-2-(3-phenylpropyl)morpholine
4-[(2-chlorophenyl)methyl]-1-[(1-phenyl-1H-pyrazol-4-yl)methyl]-1,4-diazepan-5-one
(1S,5R)-3-[(4-methoxyphenyl)methyl]-6-(3-methyl-1,2-oxazole-5-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
N-[cyclopropyl(4-methylpyridin-2-yl)methyl]-5-[(4-methylpiperazin-1-yl)methyl]furan-2-carboxamide
4-{1,8-dioxa-4,11-diazaspiro[5.6]dodecane-4-sulfonyl}benzonitrile
(4aS,8aS)-2-[7-(pyridine-3-carbonyl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl]-decahydroisoquinoline
4-{[4-methyl-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}-1-(2,4,5-trimethylbenzoyl)piperidine
9-(2-methylpyrimidine-5-carbonyl)-2-[2-(pyridin-2-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
N-{[1-methyl-2-(methylsulfanyl)-1H-imidazol-5-yl]methyl}-4-sulfamoylbenzamide
4-(3-hydroxy-3-methylbutyl)-N-{[1-(hydroxymethyl)cyclobutyl]methyl}-N-methylbenzamide
1-{7-[(2-fluoro-5-methoxyphenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}-2-(methylsulfanyl)ethan-1-one
2-(4-benzyl-2-oxopyrrolidin-1-yl)-N-methyl-N-{[3-(methylsulfanyl)phenyl]methyl}acetamide
5-{6-[(pyridin-2-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}pyridin-2-amine
ethyl 4-(3-phenylpropyl)-1-(1,2,5-thiadiazole-3-carbonyl)piperidine-4-carboxylate
N-(2,4-dimethyl-6-oxo-1,6-dihydropyridin-3-yl)-4-[(3-methylpiperidin-1-yl)methyl]benzamide
N,N-bis(furan-2-ylmethyl)-1-(oxan-4-yl)piperidine-3-carboxamide
1-(furan-2-ylmethyl)-N-{2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]ethyl}piperidine-4-carboxamide
ethyl 4-{3-[(cyclopentylamino)methyl]-6-methylquinolin-2-yl}piperazine-1-carboxylate
3-(2,3-dimethoxyphenyl)-1-{2-methylpyrido[2,3-d]pyrimidin-4-yl}pyrrolidine
3-cyclopropyl-1-[3-(pyridin-2-yl)phenyl]-3-[(trimethyl-1H-pyrazol-4-yl)methyl]urea
3-{[(2S,5R)-5-({ethyl[(1-methyl-1H-pyrazol-4-yl)methyl]amino}methyl)oxolan-2-yl]methyl}benzonitrile
1-(2-{4-phenyl-5-[1-(propan-2-yl)-1H-pyrazol-4-yl]-1H-imidazol-1-yl}ethyl)pyrrolidin-2-one
methyl({[5-(oxan-2-yl)furan-2-yl]methyl}){[3-(1H-1,2,3,4-tetrazol-5-yl)phenyl]methyl}amine
[(3R,4R)-1-(2,5-difluorobenzoyl)-4-{[4-(hydroxymethyl)piperidin-1-yl]methyl}pyrrolidin-3-yl]methanol
3-[5-(1H-indol-3-ylmethyl)-1,3,4-oxadiazol-2-yl]-1-[2-(1,3-thiazol-2-yl)piperidin-1-yl]propan-1-one
N-{[2-(2,3-dihydro-1,4-benzodioxin-6-yl)phenyl]methyl}propanamide
4-{1-[1-(3-ethyl-1,2,4-oxadiazol-5-yl)ethyl]-1H-imidazol-2-yl}-N-methylbenzene-1-sulfonamide
N-[2-(5-methylfuran-2-yl)ethyl]-2-[2-(propan-2-yl)-1H-imidazol-1-yl]propanamide
1-[(1-phenylcyclopentyl)methyl]-5-{2-[(pyridin-3-ylmethyl)amino]ethyl}pyrrolidin-2-one
2-{1-[3-(propan-2-yl)-1,2-oxazole-5-carbonyl]piperidine-3-carbonyl}pyridine
2-(dimethylamino)-N-(2-methoxy-2-methylpropyl)-2-(2-methylphenyl)acetamide
N-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]-1-(propan-2-yl)piperidine-4-carboxamide
4-[2-(6-methylpyridin-2-yl)-1H-imidazol-1-yl]-1-(propan-2-yl)pyrrolidin-2-one
1-[(5-methyl-1H-pyrazol-3-yl)methyl]-3-(1,3,6-trimethyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)urea
N-[(4-chlorophenyl)methyl]-3-[(4S)-4-hydroxy-3,3,4-trimethylpiperidin-1-yl]propanamide
5-[1-(2,3-dihydro-1-benzofuran-5-ylmethyl)piperidin-4-yl]-5-propyl-3-[2-(pyridin-2-yl)ethyl]imidazolidine-2,4-dione
N-[1-(pyridin-2-ylmethyl)piperidin-3-yl]quinoxalin-2-amine
methyl[(3-methylpyridin-2-yl)methyl]{[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}amine
3-[3-(furan-2-yl)-1H-1,2,4-triazol-5-yl]-1-methyl-1-[(5-phenyl-1H-pyrazol-4-yl)methyl]urea
N-[2-(3-methylphenyl)ethyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
2-{3-[(3,4-dimethoxyphenyl)methyl]-5-(oxolan-3-yl)-1H-1,2,4-triazol-1-yl}ethan-1-ol
(4aS,7aR)-1-(1H-imidazol-2-ylmethyl)-4-(pyrimidin-2-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
ethyl 5-(1-{[(1,4-dimethyl-1H-pyrazol-5-yl)carbamoyl]methyl}-1H-pyrazol-4-yl)thiophene-2-carboxylate
5-(2-chloro-4-fluorophenoxymethyl)-N-[(1-hydroxycyclohexyl)methyl]-1,2-oxazole-3-carboxamide
N3-[2-(3-fluorophenyl)ethyl]-4-oxo-1-(oxolan-2-ylmethyl)-N5-(2-phenylethyl)-1,4-dihydropyridine-3,5-dicarboxamide
1-[(3-benzyl-1H-1,2,4-triazol-5-yl)methyl]-4-phenylpyrrolidin-2-one
4-{[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]sulfamoyl}-N-propylbenzamide
N-(1-{[3-(2,5-dimethylphenyl)-1H-pyrazol-4-yl]methyl}piperidin-4-yl)methanesulfonamide
5-{[benzyl(methyl)amino]methyl}-N-[2-(morpholin-4-yl)propyl]-1,2-oxazole-3-carboxamide
N-(5-ethyl-1-methyl-1H-1,2,4-triazol-3-yl)-4-(3-phenyl-1,2,4-oxadiazol-5-yl)piperidine-1-carboxamide