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3-[(2R,3R,6R)-5-(furan-2-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-3-yl]phenol
N-[(2,5-dimethoxyphenyl)methyl]-5-{[(6-methylpyridin-3-yl)oxy]methyl}-1,2-oxazole-3-carboxamide
2-({3-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}methyl)benzonitrile
4-chloro-1-ethyl-N-(propan-2-yl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]-1H-pyrazole-5-carboxamide
4-[(1-acetylpiperidin-4-yl)oxy]-N-(3-cyclopentylpropyl)-3-methoxybenzamide
N-cyclopentyl-1-ethyl-7-methyl-4-oxo-N-propyl-1,4-dihydro-1,8-naphthyridine-3-carboxamide
N-benzyl-N-methyl-3-{[(1-methylpiperidin-4-yl)amino]methyl}pyridin-2-amine
(2S)-4-methyl-2-[4-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)-1H-1,2,3-triazol-1-yl]pentanamide
(3R,4R)-4-(azepan-1-yl)-1-[1-(4-methoxyphenyl)piperidin-4-yl]piperidin-3-ol
1-{[(2S,4S)-4-fluoro-1-{5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridine-3-carbonyl}pyrrolidin-2-yl]methyl}-3,3-dimethylurea
7-methoxy-N-[3-(1,2,3,4-tetrahydroquinolin-1-yl)propyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
2,6-dimethyl-4-(3-{1-[(1-methyl-1H-imidazol-5-yl)methyl]-1H-pyrazol-3-yl}phenyl)pyridine
5-({2-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}methyl)-2-(pyridin-2-yl)pyrimidine
N-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}-5-propyl-1,2-oxazole-3-carboxamide
N-[2-(3,5-difluorophenyl)ethyl]-2-(3-oxo-2,3-dihydro-1H-indazol-2-yl)acetamide
2-[(1R,3S)-1-hydroxy-3-methoxy-7-azaspiro[3.5]nonan-7-yl]-1-(6-methyl-1,2,3,4-tetrahydroquinolin-1-yl)ethan-1-one
1-(3-{2-[2-(1H-imidazol-1-yl)ethyl]piperidine-1-carbonyl}phenyl)imidazolidin-2-one
1-(2-phenylpropyl)-4-(pyridin-2-ylmethyl)-1,4-diazepane
1-(1-benzoxepine-4-carbonyl)-N-(4-fluorophenyl)piperidin-3-amine
N-{[4-(5-methyl-1,2,4-oxadiazol-3-yl)phenyl]methyl}-1,9-dioxaspiro[5.5]undecan-4-amine
5-(piperidin-1-yl)-2-[2-(1H-1,2,4-triazol-1-yl)ethyl]-2,3-dihydropyridazin-3-one
8-{[2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl}-1-oxa-8-azaspiro[4.6]undecane
4-[({[2-(dimethylamino)-5,6,7-trimethoxyquinolin-3-yl]methyl}amino)methyl]benzene-1-sulfonamide
3-{4-[(3-fluorophenyl)methyl]piperazine-1-carbonyl}-2,6-dimethyl-1,4-dihydropyridin-4-one
4-{1-[(6-methoxy-2H-1,3-benzodioxol-5-yl)methyl]piperidin-4-yl}pyrimidine
[(6-chloropyridin-3-yl)methyl][(4-fluorophenyl)methyl](oxolan-2-ylmethyl)amine
1-methyl-N-[2-(1-phenyl-1H-pyrazol-4-yl)ethyl]-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
3-{[2-(3,4-dichlorophenyl)morpholin-4-yl]methyl}-1,2,4-oxadiazole-5-carboxamide
1-(diphenylmethyl)-N-methyl-N-[(1-methylpiperidin-2-yl)methyl]-1H-1,2,3-triazole-4-carboxamide
3-(azocan-1-yl)-N-{[4-(5-methyl-1,2,4-oxadiazol-3-yl)phenyl]methyl}propanamide
N2-[2-methoxy-1-(1-methyl-1H-pyrazol-5-yl)ethyl]-N4,N4,5-trimethylpyrimidine-2,4-diamine
N-(1-{[5-methyl-2-(3-phenoxyphenyl)-1,3-oxazol-4-yl]methyl}piperidin-4-yl)acetamide
N-(2-hydroxy-3-phenylpropyl)-2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]acetamide
4-[(5-{1-[(2,4-dimethylphenyl)methyl]piperidin-4-yl}-4-methyl-4H-1,2,4-triazol-3-yl)methyl]morpholine
3-(3-methylbut-2-en-1-yl)-1-(4-propylpyrimidine-5-carbonyl)piperidine-3-carboxylic acid
N-({1-[(4-ethyl-4H-1,2,4-triazol-3-yl)methyl]piperidin-3-yl}methyl)-4-phenylbenzamide
4-{4-[(2,5-dimethoxyphenyl)methyl]piperazin-1-yl}-2-(oxolan-2-ylmethyl)-2,3-dihydro-1H-isoindole-1,3-dione
N-benzyl-N-butyl-1-cyclopentyl-4-oxo-5-(piperidine-1-carbonyl)-1,4-dihydropyridine-3-carboxamide
2-(2,3-dihydro-1,4-benzodioxin-6-yl)-N,N-dimethylpyridine-3-carboxamide
3-(1H-imidazol-1-ylmethyl)-N-[3-(1H-imidazol-5-yl)phenyl]piperidine-1-carboxamide
3-({2-[1-(dimethyl-1,3-thiazole-5-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}methyl)pyridine
2-{3-hydroxy-5-[2-(piperidin-2-yl)ethyl]phenyl}pyridin-3-ol
N-[3-(3-methoxyphenyl)phenyl]-1-(2-methoxypyridine-3-carbonyl)piperidine-2-carboxamide
N-methyl-1-{6-methylthieno[2,3-d]pyrimidin-4-yl}-N-[3-(1H-pyrazol-1-yl)propyl]piperidin-4-amine
4-(cyclopropylmethyl)-3-(propan-2-yl)-1-[1-(1H-pyrazol-1-ylmethyl)cyclopropanecarbonyl]-1,4-diazepan-5-one
3-[3-(dimethylamino)propyl]-1-(3-methylbutyl)-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxylic acid
N-(2-{7-[3-(1H-indol-3-yl)propanoyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)cyclohexanecarboxamide
5-[3-(4-fluorophenoxymethyl)piperidine-1-carbonyl]quinoxaline
N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
2-methyl-N-[2-(2-methylpropanesulfonyl)ethyl]-1,2,3,4-tetrahydroisoquinoline-3-carboxamide