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1-[(3R,4R)-4-cyclopropyl-4-hydroxy-3-methylpiperidin-1-yl]-2-(4-methylphenoxy)ethan-1-one
(1R,7S)-3-cycloheptyl-6-(4-ethyl-3-oxopiperazine-1-carbonyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-4-one
5-{[2-(3-methoxypropyl)-3-oxo-2,8-diazaspiro[4.5]decan-8-yl]methyl}-N,N-dimethylfuran-2-carboxamide
N-[5-(1H-indol-4-yl)pyridin-2-yl]methanesulfonamide
1-{[2-(cyclopentylmethyl)-1H-imidazol-4-yl]methyl}-3-(piperidin-1-ylmethyl)pyrrolidin-3-ol
5-[(4-hydroxypiperidin-1-yl)methyl]-N-[1-(1-methyl-1H-pyrazol-5-yl)propyl]-1,2-oxazole-3-carboxamide
N-[(7R,8aS)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-2-methoxypyridine-4-carboxamide
5-[(1S,5R)-3-[(dimethyl-1,2-oxazol-4-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-1,2-dihydropyridin-2-one
(4aS,7aR)-1-(2,3-dihydro-1-benzofuran-5-carbonyl)-4-methanesulfonyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-chloro-4-({1-[(5-chlorothiophen-2-yl)methyl]piperidin-4-yl}oxy)-N-(2-methoxyethyl)benzamide
S-(4-fluoro-3-methylphenyl)-2-[3-(1H-imidazol-2-yl)piperidin-1-yl]-2-oxoethane-1-sulfonamido
1-(1H-imidazol-2-ylmethyl)-8-[5-(trifluoromethyl)pyridin-2-yl]-1,8-diazaspiro[4.5]decane
1-[4-(dimethylamino)-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-2-(3-hydroxyphenyl)ethan-1-one
4-cyclopentyl-N-(2-fluoro-5-methylphenyl)-1,4-diazepane-1-carboxamide
9-[3-(1H-1,2,3-benzotriazol-1-yl)propanoyl]-1-methyl-1,4,9-triazaspiro[5.5]undecan-5-one
1-cyclopentyl-3-{pyrazolo[1,5-a]pyridin-3-ylmethyl}urea
2-{2-[1-(6-cyanopyridine-3-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}acetamide
(3R,4R)-4-ethyl-1-{4H,5H,6H,7H-pyrazolo[1,5-a]pyridine-3-carbonyl}piperidine-3,4-diol
2-[({5-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)(thiophen-2-ylmethyl)amino]ethan-1-ol
(3aS,6aS)-5-[(3-chloro-4-propoxyphenyl)methyl]-1-methyl-octahydropyrrolo[3,4-b]pyrrole
2-[(4-methoxyphenyl)methyl]-4-(2,2,2-trifluoroethanesulfonyl)morpholine
N-[1-(2,5-difluorophenyl)cyclopropyl]-1-methyl-6-oxo-1,6-dihydropyridine-3-carboxamide
N-(2-{4-methyl-5H,6H,7H-cyclopenta[d]pyrimidin-2-yl}ethyl)-7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carboxamide
N-methyl-2-oxo-6-phenyl-N-{2-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}-1,2-dihydropyridine-3-carboxamide
6-(2-benzyl-1,3-thiazole-4-carbonyl)-1H,2H,3H,4H,5H,6H,7H,8H-pyrazolo[3,4-d]azepin-3-one
1-[4-(3-hydroxy-3-methylbut-1-yn-1-yl)benzoyl]-4-(pyridin-2-yl)piperidin-4-ol
1-(3-{[3-(hydroxymethyl)-3-[(3-methoxyphenyl)methyl]piperidin-1-yl]methyl}phenyl)ethan-1-one
1-(2-methoxyphenyl)-5-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-3-(2-methylpropyl)-1H-1,2,4-triazole
3-(dimethyl-1,2-oxazol-4-yl)-1-[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)pyrrolidin-1-yl]propan-1-one
6-{1-[5-(methoxymethyl)thiophene-2-carbonyl]piperidin-3-yl}pyrimidin-4-ol
1-(4-acetyl-1,4-diazepan-1-yl)-3-(3-chlorophenyl)-3-(3-hydroxyphenyl)propan-1-one
2-[(6-methoxypyrimidin-4-yl)amino]-1-phenylethan-1-ol
1-[3-(2-amino-6-methylpyrimidin-4-yl)phenyl]ethan-1-one
3-[5-(1-carbamoylethyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]-N-(2-hydroxyethyl)propanamide
(1S,4S)-2-(2-chlorophenyl)-5-[(3,4-difluorophenyl)methyl]-2,5-diazabicyclo[2.2.1]heptan-3-one
1-{1'-[(2,3-difluoro-4-methylphenyl)methyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}ethan-1-one
1-(3-{4-amino-1H-pyrazolo[3,4-d]pyrimidin-3-yl}phenyl)ethan-1-one
3-[(3-propyl-1,2,4-oxadiazol-5-yl)methoxy]pyridine-2-carbonitrile
1-(2-aminoethyl)-N-{1-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}-1H-1,2,3-triazole-4-carboxamide
2-(methylsulfanyl)-N-[(3R,4S)-1-(oxan-4-ylmethyl)-4-phenylpyrrolidin-3-yl]acetamide
2-methoxy-5-{[({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)(2-methylpropyl)amino]methyl}phenol
3-{4-[(1-ethyl-1H-imidazol-2-yl)methyl]piperazin-1-yl}-1,2-dihydropyrazin-2-one
N-(1-hydroxybutan-2-yl)-N-[(5-methylthiophen-2-yl)methyl]-2-{5H,6H,7H-[1,3]thiazolo[3,2-a]pyrimidin-3-yl}acetamide
1-{1,9-dioxaspiro[5.5]undecan-4-yl}-4-(4-fluorophenyl)piperidin-4-ol
1-(1-cyclopropanecarbonylpiperidin-4-yl)-N-ethyl-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide
N-{[2-(1H-imidazol-1-yl)phenyl]methyl}-2-[4-(pyrimidin-2-yl)piperazin-1-yl]acetamide
2-(2-aminoethyl)-N-methyl-N-{2-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}quinazolin-4-amine
(1R,2R,6S,7S)-4-{dimethyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}-10-oxa-4-azatricyclo[5.2.1.02,6]decane
2-methyl-6-[1-(1,2,3,4-tetrahydronaphthalene-2-carbonyl)piperidin-4-yl]pyrimidin-4-ol
methyl 6-[(4-ethylphenyl)methyl]-2-[(prop-2-en-1-yl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate