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1-cyclopentyl-4-[5-(1H-imidazol-1-ylmethyl)pyridin-2-yl]-1,4-diazepane
3-(2-ethylphenyl)-5-[(2-methoxyethyl)sulfamoyl]benzoic acid
[4-(6-methoxypyridazin-3-yl)phenyl]methanamine
N-(2-phenyl-5,6,7,8-tetrahydroquinazolin-5-yl)-2H-1,3-benzodioxole-5-carboxamide
2-[3-(diphenylmethyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-N-ethylpropanamide
N-[(3R,5S)-1-benzyl-5-(ethylcarbamoyl)pyrrolidin-3-yl]-2-methyl-1,3-thiazole-4-carboxamide
1-methyl-3-(propan-2-yl)-4-[2-(pyridin-4-yl)pyrimidine-5-carbonyl]piperazin-2-one
4,6-dimethyl-N-{[5-(thiophen-2-yl)-1H-pyrazol-4-yl]methyl}pyrimidin-2-amine
1-[2-(4-methoxyphenyl)ethyl]-3-methyl-8-(pyridin-4-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-(4-{[2-(3,4-difluorophenyl)-2,3,4,5-tetrahydro-1,5-benzothiazepin-5-yl]methyl}phenyl)acetamide
ethyl 5-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl]-1-(2-methoxyethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
(1S,5R)-3-[5-(2-chlorophenyl)furan-2-carbonyl]-6-methyl-3,6-diazabicyclo[3.2.2]nonan-7-one
(2E)-1-(3-{[2-(3,4-dimethoxyphenyl)ethyl](methyl)amino}piperidin-1-yl)-3-(1H-imidazol-4-yl)prop-2-en-1-one
2-methyl-1-{4-[3-(propan-2-yl)-1H-pyrazol-5-yl]piperidin-1-yl}-3-(1H-pyrazol-1-yl)propan-1-one
1-(furan-2-ylmethyl)-1-(2-hydroxyethyl)-3-(1-propyl-1H-1,3-benzodiazol-5-yl)urea
8-methoxy-N-[3-(4-methyl-1,3-thiazol-2-yl)propyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
1-{[3-(3-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}-4-(4-methyl-1,2,5-oxadiazol-3-yl)piperazine
2-{8-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-2,4-dioxo-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decan-3-yl}acetamide
7-benzoyl-N-(pyridin-2-ylmethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
N-methyl-5-{[2-methyl-4-(1H-pyrazol-1-yl)phenyl]methyl}-2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
4-[(2,3-difluorophenyl)methyl]-3-[2-oxo-2-(pyrrolidin-1-yl)ethyl]piperazin-2-one
4-({5-cyclopropanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}carbonyl)-2,3-dihydro-1H-imidazol-2-one
1-butyl-4-[6-methyl-2-(pyridin-3-yl)pyrimidin-4-yl]piperazin-2-one
1-(4-fluorophenyl)-4-[5-(methoxymethyl)thiophene-2-carbonyl]-1,4-diazepane
3-({3-[2-(pyridin-3-yl)pyridin-4-yl]pyrrolidin-1-yl}methyl)phenol
(1R,3S)-7-(1H-indole-6-carbonyl)-3-methoxy-7-azaspiro[3.5]nonan-1-ol
1-(1,3-benzothiazol-6-yl)-3-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-3-methylurea
3-(4-{[methyl(thian-4-yl)amino]methyl}-1H-pyrazol-1-yl)propanoic acid
1-{3-fluoroimidazo[1,2-a]pyridine-2-carbonyl}-4-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-yl}piperidine
N-cyclopropyl-1-[(3-methoxyphenyl)methyl]-5-(3-phenylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
(1S,6R)-3-(1-benzofuran-2-ylmethyl)-3,9-diazabicyclo[4.2.1]nonane
2-(3-methoxyphenoxy)-1-[3-(2-methylphenoxy)azetidin-1-yl]propan-1-one
(2,1,3-benzoxadiazol-5-ylmethyl)(methyl)[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]amine
9-({3-[2-(piperidin-1-yl)ethoxy]phenyl}methyl)-3-oxa-9-azaspiro[5.5]undecane
3-[2-(3-methyl-1,2,4-oxadiazol-5-yl)ethyl]-1H-indole
3-(1-{[5-(1,5-dimethyl-1H-pyrrol-2-yl)-1,3,4-oxadiazol-2-yl]methyl}pyrrolidin-2-yl)-4-methyl-1,2,5-oxadiazole
3-methyl-5-(2H-1,2,3-triazol-2-ylmethyl)-1-[4-(trifluoromethoxy)phenyl]-1H-1,2,4-triazole
1-(1-{imidazo[2,1-b][1,3,4]thiadiazol-6-yl}ethyl)-2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazole
1-methyl-N-(2-phenylethyl)-N-{pyrazolo[1,5-a]pyrimidin-3-ylmethyl}piperidin-4-amine
8-[(4-methoxy-5,6,7,8-tetrahydronaphthalen-1-yl)sulfonyl]-2,8-diazaspiro[4.5]decan-3-one
1-{[3-(4-phenylphenyl)-1H-pyrazol-4-yl]methyl}-4-(pyrrolidin-1-yl)piperidine
2-methyl-N-[1-(4-methyl-4H-1,2,4-triazol-3-yl)ethyl]-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-amine
N-methyl-3-phenyl-N-{[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}-1,2,4-oxadiazol-5-amine
2-{[(2-chlorophenyl)methyl]sulfanyl}-N-(prop-2-yn-1-yl)acetamide
3-{3-hydroxy-5-[2-(piperidin-2-yl)ethyl]phenyl}-1,2-dihydropyridin-2-one
2-[(3R,4R)-3-hydroxy-4-(morpholin-4-yl)piperidin-1-yl]-5,6,7,8-tetrahydroquinoline-3-carbonitrile
4-[2-(dimethylamino)ethyl]-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
(3aR,6aR)-2-acetyl-N-(adamantan-1-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
3-{2-[4-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]-2-oxoethyl}-3,4-dihydroquinazolin-4-one
(3aR,5R,6S,7aS)-2-[4-(ethylamino)pyrimidin-2-yl]-octahydro-1H-isoindole-5,6-diol