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1-(2-methoxyacetyl)-4-[2-(piperidin-1-yl)ethyl]-1,4-diazepane-6-carboxylic acid
4-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(1H-pyrrole-3-carbonyl)piperidine
(3aR,6aR)-2-methyl-N-{[1-(phenoxymethyl)cyclopropyl]methyl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
[1-(2-chlorophenyl)ethyl]({[2-(3-methylphenyl)pyrimidin-5-yl]methyl})amine
3-[4-(benzyloxy)piperidine-1-carbonyl]-2-methyl-4,5,6,7-tetrahydro-1-benzofuran-4-one
(4aS,8aR)-1-(2-aminoethyl)-6-{5-[(dimethylamino)methyl]furan-2-carbonyl}-decahydro-1,6-naphthyridin-2-one
(2S)-N-{5H,6H,7H,8H,9H,10H,11H-cycloocta[b]indol-2-ylmethyl}-3-hydroxy-2-(methylamino)propanamide
4-[5-(1-benzyl-1H-imidazol-5-yl)-1H,4H-pyrazolo[3,4-d]imidazol-1-yl]-1-methylpiperidine
3-(3-{3-[2-(dimethylamino)-6-methylpyrimidin-4-yl]phenyl}-1H-pyrazol-1-yl)propan-1-ol
1-(3-chloropyridin-2-yl)-4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazine
1-[(3S,4R)-4-ethoxyoxolan-3-yl]-4-phenyl-5-{pyrazolo[1,5-a]pyrimidin-3-yl}-1H-imidazole
N-({5-[6-(4-fluorophenyl)pyridazin-3-yl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)acetamide
1-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-5-oxopyrrolidine-3-carboxylic acid
N-[2-(3-fluorophenyl)ethyl]-2-[1-(naphthalen-2-ylmethyl)-3-oxopiperazin-2-yl]acetamide
3-[(3R,4S)-1-(4-chloro-1-methyl-1H-pyrrole-2-carbonyl)-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propan-1-ol
N-(dimethyl-1,2-oxazol-4-yl)-4-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)benzamide
2-methoxy-N-{[1-(2-methylpropyl)pyrrolidin-3-yl]methyl}pyrimidine-5-carboxamide
N-ethyl-5-[7-methoxy-4-(pyrrolidine-1-carbonyl)quinolin-2-yl]pyrimidin-2-amine
1-[(5-methylfuran-2-yl)methyl]-4-(naphthalen-2-yloxy)piperidine-4-carboxylic acid
(3R,5S)-N-[2-(4,6-dimethylpyrimidin-2-yl)ethyl]-5-(pyrrolidine-1-carbonyl)piperidine-3-carboxamide
6-chloro-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]imidazo[1,2-a]pyridine-2-carboxamide
(1R,3S)-7-[2-(1,1,2,2-tetrafluoroethoxy)benzoyl]-7-azaspiro[3.5]nonane-1,3-diol
5-[4-(propan-2-yl)piperazin-1-yl]-1-propyl-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazole
2-(dimethylamino)-8-[3-(1H-pyrazol-1-ylmethyl)phenyl]-4H,5H,6H,7H,8H-[1,3]thiazolo[4,5-c]azepin-6-one
3-{[4-(pyrimidin-2-yl)-1,4-diazepan-1-yl]methyl}-1,2,5,6,7,8-hexahydroquinolin-2-one
1-[(2,3-difluorophenyl)methyl]-3-hydroxy-3-[(3-hydroxyazetidin-1-yl)methyl]piperidin-2-one
methyl({1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}methyl)(3-phenylpropyl)amine
1-[(1-{pyrazolo[1,5-a]pyridine-7-carbonyl}pyrrolidin-2-yl)methyl]-1H-pyrazole
4-phenyl-N-{1-[1-(1,2,3,4-tetrahydronaphthalen-2-yl)piperidin-4-yl]-1H-pyrazol-5-yl}butanamide
1-[2-(1H-1,2,3,4-tetrazol-5-yl)benzoyl]-4-(thian-4-yl)piperazine
(3R,4R)-1-(1-benzothiophene-2-carbonyl)-3-methyl-4-(oxan-4-yl)piperidin-4-ol
N-[(2-methoxyphenyl)methyl]-2-[4-(pyrazine-2-carbonyl)morpholin-3-yl]acetamide
N-{2-[2-(1H-imidazol-1-yl)acetyl]-1,2,3,4-tetrahydroisoquinolin-7-yl}-3-(4-methylphenyl)propanamide
4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-1-{[5-methyl-2-(3-methylthiophen-2-yl)-1,3-oxazol-4-yl]methyl}piperidine
3-{1-[(2-butyl-1H-imidazol-4-yl)methyl]piperidin-4-yl}-N-[(4-fluorophenyl)methyl]propanamide
4-(4-methoxy-3-methylbenzoyl)-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
N-[(3R,4R)-3-hydroxypiperidin-4-yl]-2-{[(2-methylphenyl)methyl]sulfanyl}acetamide
(2,1,3-benzoxadiazol-4-ylmethyl)(methyl){[3-(pyridin-2-yl)-1,2-oxazol-5-yl]methyl}amine
[(3R,4R)-4-(azepan-1-ylmethyl)-1-(4-chloro-1H-pyrazole-3-carbonyl)pyrrolidin-3-yl]methanol
N-[2-(4-methyl-1H-pyrazol-1-yl)ethyl]-7-(oxolan-3-ylmethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
5-{1-methyl-10-oxo-1,4,9-triazaspiro[5.6]dodecane-4-carbonyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
(3S,4R)-1-[(1R,5S,6S)-3-azabicyclo[3.1.0]hexan-6-ylmethyl]-4-(2-methylphenyl)pyrrolidine-3-carboxylic acid
3-(3-fluorophenyl)-5-(4-methoxybenzoyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
methyl 3-(5-methylthiophene-2-amido)-6-(morpholin-4-ylmethyl)thieno[2,3-b]pyridine-2-carboxylate
{[1-(2,4-difluorophenyl)-3-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]amine
3-(4-methyl-1H-imidazol-5-yl)-4-[(3-methylphenyl)methyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
(3S,4R)-4-phenyl-1-(quinoxaline-5-carbonyl)pyrrolidine-3-carboxylic acid
3-[2-fluoro-3-(trifluoromethyl)phenyl]-1-[1-(oxolan-2-ylmethyl)piperidin-4-yl]urea
(3aS,6aS)-2-acetyl-5-[(3-methylphenyl)methanesulfonyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-[(2,4-dimethoxyphenyl)methyl]-4-propylpyrimidine-5-carboxamide