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N-methyl-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-2-{[2-(pyrrolidin-1-yl)ethyl]sulfanyl}acetamide
3-chloro-N-cyclopentyl-4-({1-[(methylcarbamoyl)methyl]piperidin-4-yl}oxy)benzamide
N-[(2-methylphenyl)methyl]-3-(4-methylpiperazine-1-carbonyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
2-(2-fluoro-5-methoxyphenyl)-2-{methyl[(3-methyl-1,2-oxazol-5-yl)methyl]amino}acetic acid
(1R,2S,9R)-11-(1H-indole-2-carbonyl)-7,11-diazatricyclo[7.3.1.02,7]tridecan-6-one
6-[(diethylamino)methyl]-N-methyl-N-[(2-methyl-1,3-thiazol-4-yl)methyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
(3R)-3,4,4-trimethyl-1-{4-[(4-methylpiperazin-1-yl)methyl]benzoyl}pyrrolidin-3-ol
4-(3-{[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]formamido}propyl)-1,2,5-oxadiazole-3-carboxylic acid
N-(4-{[(3R,4R)-3-(azepan-1-ylmethyl)-4-(hydroxymethyl)pyrrolidin-1-yl]methyl}phenyl)acetamide
4-[2-(2-hydroxyphenyl)-6-methylpyrimidin-4-yl]-1λ6-thiomorpholine-1,1-dione
[(2S,6S)-4-(3-methyl-1-propyl-1H-pyrazole-4-carbonyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(9),10,12-trien-6-yl]methanol
1-methyl-8-[(2-methyl-1H-indol-3-yl)methyl]-3-[3-(pyridin-4-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
6-amino-N-[1-(morpholine-4-carbonyl)piperidin-4-yl]pyridine-3-carboxamide
4-[(2,3-difluorophenyl)methyl]-1,3λ6,4-oxathiazinane-3,3-dione
4-[(3R,4R)-4-[4-(2-cyclohexylpyrimidin-5-yl)-1H-1,2,3-triazol-1-yl]oxolan-3-yl]morpholine
(3R,4S)-1-(2-methyl-1,3-benzothiazole-5-carbonyl)-4-(5-methylfuran-2-yl)pyrrolidin-3-amine
methyl 3-methyl-4-({[3-(morpholin-4-yl)propyl]carbamoyl}amino)benzoate
7-[(4-fluorophenyl)methyl]-2-(3-methoxypropanoyl)-2,7-diazaspiro[4.5]decan-6-one
N-[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]-N-methylthian-4-amine
2-(3-fluorophenoxymethyl)-N-methyl-N-[(1-methylpyrrolidin-3-yl)methyl]-1,3-oxazole-4-carboxamide
2-cyclopropyl-4-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}quinoline
5-amino-N-[3-(3,4-diethoxyphenyl)propyl]-1H-pyrazole-3-carboxamide
(3R,4R)-4-ethyl-1-[2-(methylamino)pyridine-4-carbonyl]piperidine-3,4-diol
methyl 5-[2-(2-oxo-2,3-dihydro-1,3-benzoxazol-3-yl)ethyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylate
N-methyl-4-phenoxy-N-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}butanamide
(3S,5S)-1-[(3-methylphenyl)methyl]-5-[(6-methylpyridin-3-yl)carbamoyl]piperidine-3-carboxylic acid
6-methoxy-1-[(1S,5R)-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]hexan-1-one
N-[2-(morpholin-4-yl)ethyl]-4-[4-(4-phenylazepan-1-yl)piperidin-1-yl]benzamide
2-[2-(4-{2-methylimidazo[1,2-a]pyridine-6-carbonyl}piperazin-1-yl)ethoxy]ethan-1-ol
1-{[2-(4-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-(3-methoxypropyl)piperidine
(1R,9aR)-1-{[methyl(quinolin-2-ylmethyl)amino]methyl}-octahydro-1H-quinolizin-1-ol
N-cyclopentyl-3-{methyl[1-(pyridin-4-yl)ethyl]sulfamoyl}benzamide
N-(pyridin-3-ylmethyl)-3-{[1-(thian-4-yl)piperidin-4-yl]oxy}benzamide
N-(4-chloro-2-methylphenyl)-1-methyl-10-oxo-1,4,9-triazaspiro[5.6]dodecane-4-carboxamide
N-{1,9-dioxaspiro[5.5]undecan-4-yl}-2-(quinazolin-4-yloxy)acetamide
2-(methoxymethyl)-5-{[3-(2-methylphenyl)piperidin-1-yl]methyl}pyrimidine
N-(1H-pyrazol-3-ylmethyl)-3,4-dihydro-2H-1-benzopyran-3-carboxamide
N-benzyl-4-(6-methyl-3-oxo-2,3-dihydropyridazin-4-yl)benzene-1-sulfonamide
4,6-dimethyl-2-{3-oxo-2-[2-(pyridin-2-yl)ethyl]-2,9-diazaspiro[5.5]undecan-9-yl}pyridine-3-carbonitrile
1-{3-[2-(4-methoxyphenyl)ethyl]piperidin-1-yl}-2-[(5-methyl-1,3,4-oxadiazol-2-yl)sulfanyl]ethan-1-one
4-amino-1-(cyclohexylmethyl)pyrrolidin-2-one
N-[(7S,8aS)-2-methyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-2-(1-methyl-1H-indol-3-yl)acetamide
2-(2,2-dimethyloxan-4-yl)-1-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}-1H-imidazole
3-{5-[3-(6-oxo-1,6-dihydropyridazin-3-yl)propanoyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanoic acid
4-({3-[3-(2-methylpiperidin-1-yl)azetidine-1-carbonyl]-1,2-oxazol-5-yl}methyl)morpholine
2-(4-chloro-3-methyl-1H-pyrazol-1-yl)-1-[4-(3-methylpyridin-2-yl)piperazin-1-yl]ethan-1-one
N-[3-(cyclopentyloxy)propyl]-6-(4H-1,2,4-triazol-4-yl)pyridine-3-carboxamide
5-[2-(4-hydroxy-1,2,3,4-tetrahydroisoquinolin-2-yl)-2-oxoethyl]-2,6-dimethyl-3,4-dihydropyrimidin-4-one
4-{[3-(4-chlorobenzoyl)piperidin-1-yl]methyl}-2-ethoxyphenol
5-(1H-indol-1-ylmethyl)-N-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]-1H-pyrazole-3-carboxamide