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6-ethyl-1-methyl-N-[2-(3-phenyl-1,2,4-oxadiazol-5-yl)ethyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
5-(3-chloro-4-methoxyphenyl)pyrazin-2-amine
5-methyl-N-(oxolan-2-ylmethyl)-6-(piperidine-1-carbonyl)thieno[2,3-d]pyrimidin-4-amine
1-(oxolane-3-carbonyl)-4-[4-(pyrrolidin-1-ylmethyl)-1H-1,2,3-triazol-1-yl]piperidine
6-methyl-N-[1-(4-methyl-1H-imidazol-2-yl)propyl]-2-oxo-1,2-dihydropyridine-4-carboxamide
1-[(2-methoxyphenyl)methyl]-N3-[(5-methylfuran-2-yl)methyl]-N5-[3-(methylsulfanyl)propyl]-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
N-{2-[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]ethyl}-2-(pyridin-4-yl)pyrimidine-5-carboxamide
N-[(3R,4S)-1-(1-acetylpiperidin-4-yl)-4-cyclopropylpyrrolidin-3-yl]-2-(methylsulfanyl)acetamide
3-[(3R,4S)-1-(1-methyl-1H-indole-3-carbonyl)-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propan-1-ol
2-methyl-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
N4-(1-cycloheptyl-5-oxopyrrolidin-3-yl)-N1,N1-dimethylpiperidine-1,4-dicarboxamide
8-chloro-2-(furan-2-yl)-4-(thiomorpholine-4-carbonyl)quinoline
[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl](methyl)[(4-methyl-1H-imidazol-2-yl)methyl]amine
(1S,5R)-3-(3-methylthiophene-2-carbonyl)-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1'-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}-3H-spiro[2-benzofuran-1,4'-piperidine]-3-one
6-[3-(4-phenyl-1H-pyrazol-5-yl)piperidin-1-yl]pyridine-3-carboxylic acid
1-{4-[(furan-2-ylmethyl)sulfanyl]phenyl}-3-[1-(1-methyl-1H-imidazol-2-yl)butyl]urea
6-[4-(pyridin-2-ylmethyl)piperazin-1-yl]-9H-purine
(2-ethoxy-5-{[(1H-indol-4-ylmethyl)amino]methyl}phenyl)methyl acetate
4-[(dipropylamino)methyl]-N-methyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]benzamide
3-{4-[(2-fluoro-4-methoxyphenyl)methyl]-3-(2-hydroxyethyl)piperazine-1-carbonyl}phenol
methyl 3-[(2E)-3-(4-fluorophenyl)prop-2-enamido]-6-{[methyl(propan-2-yl)amino]methyl}thieno[2,3-b]pyridine-2-carboxylate
(1R,7S)-N-methyl-4-oxo-3-(pentan-3-yl)-N-(1H-pyrazol-3-ylmethyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
5-(2H-1,3-benzodioxol-5-ylmethyl)-3-cyclopropyl-1-(4-methanesulfonylphenyl)-1H-1,2,4-triazole
1-[(1R,3S)-1,3-dihydroxy-7-azaspiro[3.5]nonan-7-yl]-3-(1-methyl-1H-pyrazol-4-yl)propan-1-one
N-[(3S,5S,9S)-2,8-dioxo-1,7-diazatricyclo[7.3.0.03,7]dodecan-5-yl]-4-methoxybenzamide
5-(2-methylpropyl)-1'-(pyridine-3-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
1-(3-cyanophenyl)-3-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}-3-methylurea
5-(2,6-dimethoxyphenyl)-N-methyl-N-[(7-methyl-1H-1,3-benzodiazol-2-yl)methyl]-1,2,4-triazin-3-amine
9-(2-fluoro-4-methylbenzoyl)-2-(3-methoxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
1-[(5-chloro-3-methoxy-2-propoxyphenyl)methyl]-4-(pyrrolidin-3-yl)piperazine
8-(1-ethyl-1H-pyrazole-3-carbonyl)-2-[2-(1H-imidazol-4-yl)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
methyl({[5-methyl-2-(2-methylphenyl)-1,3-oxazol-4-yl]methyl})[1-(thiophen-2-yl)ethyl]amine
1-[(3R,4S)-4-hydroxy-3,4-dimethylpiperidin-1-yl]-2-[2-(trifluoromethyl)phenyl]ethan-1-one
{[2-(morpholin-4-yl)pyridin-3-yl]methyl}[(trimethylpyrazin-2-yl)methyl]amine
N,5-dimethyl-N-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}-1-(pyridin-2-yl)-1H-pyrazole-4-carboxamide
4-{3-[(2-methyl-1H-imidazol-1-yl)methyl]piperidine-1-carbonyl}-N-[(3-methylthiophen-2-yl)methyl]aniline
1-[1-(2H-1,3-benzodioxol-5-ylmethyl)piperidin-4-yl]-N-cyclopropylpiperidine-3-carboxamide
2-(2,5-dimethoxyphenyl)-1-[4-(2,6-dimethylpyridin-4-yl)piperazin-1-yl]ethan-1-one
[1-(2-chloro-5-fluorobenzoyl)-3-ethylpiperidin-3-yl]methanol
methyl(2-methylpropyl){2-[4-(piperidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]ethyl}amine
(3S,4R)-1-[3-(cyclopentylcarbamoyl)propanoyl]-4-(pyridin-3-yl)pyrrolidine-3-carboxylic acid
9-[(dimethyl-1H-1,2,4-triazol-5-yl)methyl]-2-[2-(pyridin-2-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
3-[(1S,4S)-2-azabicyclo[2.2.1]heptan-2-yl]-N-(2-methylphenyl)-3-oxopropanamide
6-{2-[4-(2-methoxyethyl)phenoxymethyl]phenyl}-2-methyl-2,3-dihydropyridazin-3-one
5-amino-3-[2-(prop-2-en-1-yloxy)phenyl]-1,6-diazatricyclo[6.2.2.02,7]dodeca-2,4,6-triene-4-carbonitrile
3-({[(3-methylthiophen-2-yl)methyl](pyridin-2-ylmethyl)amino}methyl)phenol
3-[1-(1-acetylpiperidin-4-yl)piperidin-4-yl]-N-(2,4-dimethoxyphenyl)propanamide
methyl 6-{8-cyclopropyl-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl}pyridine-3-carboxylate
[2-(2H-1,3-benzodioxol-5-ylmethyl)propyl]({[2-(morpholin-4-yl)pyridin-3-yl]methyl})amine