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5-[3-(2H-1,3-benzodioxol-5-ylmethyl)-3-methylpiperidine-1-carbonyl]-1,2-dihydropyridin-2-one
3-butyl-1-{2-[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidin-1-yl]-2-oxoethyl}-4-ethyl-4,5-dihydro-1H-1,2,4-triazol-5-one
1-(2-cyclohexylacetyl)-N-(4-fluorophenyl)piperazine-2-carboxamide
N-(2-methoxyethyl)-2-[2-(1H-pyrazol-1-yl)acetyl]-1,2,3,4-tetrahydroisoquinoline-6-sulfonamide
3-fluoro-5-{4-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyridine
2-[4-(naphthalen-1-ylmethyl)-1-[1-(propan-2-yl)piperidin-4-yl]piperazin-2-yl]ethan-1-ol
4-{4-ethyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}-1-[(4-methyl-1,3-thiazol-5-yl)methyl]piperidine
3-(5-{2,8-diazaspiro[4.5]decan-2-ylmethyl}thiophen-2-yl)prop-2-yn-1-ol
5-[1-(5-chlorothiophene-2-carbonyl)pyrrolidin-2-yl]-N-cyclopropylthiophene-2-carboxamide
1-(4-methoxyphenyl)-3-methyl-4-[4-(1H-pyrazol-4-yl)butanoyl]piperazin-2-one
N-ethyl-2-{4-[(1-phenyl-1H-pyrazol-5-yl)methyl]piperazin-1-yl}acetamide
(2E)-N-(2-{4-methyl-5-[(2-methylpropyl)sulfanyl]-4H-1,2,4-triazol-3-yl}ethyl)-3-(thiophen-2-yl)prop-2-enamide
7-methoxy-3-{1-[2-(piperazin-1-yl)ethyl]-1H-1,2,3-triazole-4-carbonyl}-2,3,4,5-tetrahydro-1H-3-benzazepine
methyl 3-(2-methoxyacetamido)-5-[(2-methylbutyl)amino]-1-(3-phenylpropyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
5-methoxy-4-oxo-N-(thiolan-3-yl)-1,4-dihydropyridine-2-carboxamide
N-[(1,2-dimethyl-1H-1,3-benzodiazol-5-yl)methyl]-3-(3-methoxyphenyl)-1H-pyrazole-4-carboxamide
6-[2-methoxy-5-(pyrrolidin-1-ylmethyl)phenoxy]pyridine-2-carbonitrile
1-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-4-(6-methyl-2H-1,3-benzodioxol-5-yl)-1H-1,2,3-triazole
2-amino-6-(1,3-dimethyl-1H-pyrazol-4-yl)-4-(2,2-dimethyloxan-4-yl)pyridine-3-carbonitrile
(3R,4S)-4-[4-(1-benzofuran-2-ylmethyl)-1,4-diazepan-1-yl]oxolan-3-ol
(3S,4R)-1-[3-(3-hydroxy-3-methylbut-1-yn-1-yl)benzoyl]-4-(3-methylthiophen-2-yl)piperidin-3-ol
3-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-5-methyl-3H,4H-thieno[2,3-d]pyrimidin-4-one
3-{5-[1-(4-chlorophenyl)cyclobutyl]-1,3,4-oxadiazol-2-yl}-1-(2-methylpiperidin-1-yl)propan-1-one
3-[(tert-butylamino)methyl]-1-[(3,4-difluorophenyl)methyl]-3-hydroxypiperidin-2-one
N-methyl-N-[2-(oxan-2-yl)ethyl]-4-oxo-3,4-dihydroquinazoline-2-carboxamide
N-methyl-N'-(5-methyl-1,2-oxazol-3-yl)-N-{[1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}ethanediamide
4-{[2-(azepan-1-yl)ethyl](methyl)amino}-N-(2-hydroxyethyl)pyridine-2-carboxamide
5-{[benzyl(methyl)amino]methyl}-N-methyl-N-[1-(thiophen-2-yl)ethyl]-1,2-oxazole-3-carboxamide
(3S,4S)-1-[4-(methoxymethyl)-5-methyl-1,2-oxazole-3-carbonyl]-4-(naphthalen-2-yl)piperidin-3-ol
4-(cyclohex-3-en-1-ylmethyl)-1-(3-methoxyphenyl)piperazin-2-one
1,5-dimethyl-4-{[3-(2-methylphenoxy)azetidin-1-yl]methyl}-2-phenyl-2,3-dihydro-1H-pyrazol-3-one
2-amino-6-(4-{[1-methyl-6-(propan-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]amino}piperidin-1-yl)-3,4-dihydropyrimidin-4-one
4-[(1S,5R)-3-[(dimethyl-1,2-oxazol-4-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-N-methylpyridin-2-amine
N-[3-(3-chlorophenyl)phenyl]-1-(pyrazine-2-carbonyl)piperidine-4-carboxamide
N-ethyl-N-(pyridin-4-ylmethyl)-2,8-diazaspiro[4.5]decane-3-carboxamide
2-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-N-methylpyridine-4-carboxamide
3-[({2-methyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}amino)methyl]-1λ6-thiolane-1,1-dione
6-methoxy-N-methyl-2-oxo-N-(quinolin-3-ylmethyl)-1,2,3,4-tetrahydroquinoline-4-carboxamide
3-[2-({5-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}amino)ethyl]-1,3-oxazinan-2-one
1-(4-{4-[(1S,6R)-3,9-diazabicyclo[4.2.1]nonane-3-carbonyl]-2-methoxyphenoxy}piperidin-1-yl)ethan-1-one
[1-(1H-imidazol-1-yl)propan-2-yl]({[1-(piperidin-1-yl)cyclohexyl]methyl})amine
5-(1-benzyl-1H-pyrazol-4-yl)-3-(oxan-4-yl)-1H-1,2,4-triazole
2-amino-4-(5-cyano-1-methyl-1H-pyrrol-3-yl)-6-(4-hydroxy-2-methylphenyl)pyridine-3-carbonitrile
6-(2-chlorophenyl)-N-(2-methoxyethyl)-7-methyl-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
2-(2-aminoethyl)-N-[3-(3-fluorophenyl)phenyl]morpholine-4-carboxamide
3-{5-[(4-chlorophenyl)methyl]-1,3,4-thiadiazol-2-yl}-1-[2-(pyridin-2-yl)ethyl]urea
(1S,4S)-2-[4-(piperazine-1-sulfonyl)benzoyl]-2,5-diazabicyclo[2.2.1]heptane
dimethyl({[4-(3,5,7-trimethyl-1H-indole-2-carbonyl)-1,4-oxazepan-6-yl]methyl})amine
9-(5-fluoro-1-methyl-1H-indole-2-carbonyl)-1-oxa-9-azaspiro[5.5]undecan-5-ol
4-({3-[6-methyl-2-(pyrrolidin-1-yl)pyrimidin-4-yl]phenyl}methyl)morpholine