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(2S)-1-(1-methyl-1H-pyrrole-2-carbonyl)-N-[3-(3-methylphenyl)phenyl]pyrrolidine-2-carboxamide
5-[(3S,4S)-1-butyl-4-hydroxypyrrolidin-3-yl]-N,N-dimethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-methyl-3-[3-(4-phenoxybenzoyl)piperidin-1-yl]propanamide
1-{3,5-diazatricyclo[9.4.0.02,7]pentadeca-1(11),2(7),3,5,12,14-hexaen-4-yl}-N-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-5-methyl-1H-pyrazole-4-carboxamide
3-[(2R,3R,6R)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]-6-methyl-1,2-dihydropyridin-2-one
2-(1H-indol-3-yl)-1-[3-(5-methyl-2-{[2-(morpholin-4-yl)ethyl]sulfanyl}pyrimidin-4-yl)piperidin-1-yl]ethan-1-one
N-[(7R,8aS)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-6-methoxy-1-methyl-1H-indole-2-carboxamide
1-(7-{[4-(propan-2-yl)phenyl]methyl}-2,7-diazaspiro[4.5]decan-2-yl)-3-(pyrazin-2-yl)propan-1-one
3-chloro-N-cyclopentyl-4-[(1-methanesulfonylpiperidin-4-yl)oxy]benzamide
3-[5-(1-ethyl-3-methyl-1H-pyrazol-4-yl)-1,2,4-oxadiazol-3-yl]-6-methylpyridazine
1-{1-[1-(difluoromethyl)-1H-pyrazole-5-carbonyl]-4-phenylpiperidin-4-yl}ethan-1-one
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-ethyl-3-(piperidin-3-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
N-cyclopropyl-2-{[5-(phenoxymethyl)-1H-pyrazol-3-yl]formamido}acetamide
7-[2-(2-fluorophenyl)acetamido]-N-(thiophen-2-yl)-1,2,3,4-tetrahydroisoquinoline-2-carboxamide
8-methoxy-N-methyl-N-{[3-(thiophen-2-yl)-1H-pyrazol-5-yl]methyl}-3,4-dihydro-2H-1-benzopyran-3-carboxamide
3-amino-1-[9-hydroxy-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-methylpropan-1-one
4-[(2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazol-1-yl)methyl]phenol
3-methyl-7-(7-methyl-2,3-dihydro-1,4-benzodioxine-6-carbonyl)-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
1-({methyl[3-(3-methylphenoxy)propyl]carbamoyl}methyl)piperidine-4-carboxamide
3,3-dimethyl-1-(3-methyl-1-propyl-1H-pyrazole-4-carbonyl)-4-(morpholin-4-ylmethyl)piperidin-4-ol
(3S)-3-({5-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}amino)azepan-2-one
N-{[7-(4,6-dimethylpyrimidin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-5-phenoxyfuran-2-carboxamide
1-{2-[(4S)-4-hydroxy-4-(methoxymethyl)-3,3-dimethylpiperidin-1-yl]-2-oxoethyl}azepan-2-one
1-[(2R,3R,6R)-3-(3-hydroxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-3-(2-methyl-1H-imidazol-1-yl)propan-1-one
(3ar,6ar)-N-{[2-(1H-1,2,4-triazol-1-yl)phenyl]methyl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
2-(3-chloro-6-oxo-1,6-dihydropyridazin-1-yl)-N-{1-[(3-methoxyphenyl)methyl]piperidin-3-yl}acetamide
1-{1-[1-(4-chlorophenyl)cyclopropanecarbonyl]piperidin-4-yl}-2-(oxolan-2-yl)-1H-1,3-benzodiazole
5-(3-fluorophenoxymethyl)-3-[3-(2-methylpropyl)pyrrolidine-1-carbonyl]-1H-pyrazole
5-{[3-(2,3-dimethoxyphenyl)pyrrolidin-1-yl]methyl}-2-methoxypyridine
8-(4-fluoro-2-methylbenzenesulfonyl)-2,8-diazaspiro[4.5]decan-3-one
3-methyl-6-{5-[1-(oxan-4-yl)piperidin-4-yl]-1,2,4-oxadiazol-3-yl}pyridazine
1-methyl-1'-{[1,2,3,4]tetrazolo[1,5-a]pyridine-6-carbonyl}-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
1-cyclopropyl-N-{[3-(2-methoxyethoxy)phenyl]methyl}-5-oxopyrrolidine-3-carboxamide
1-(1H-1,3-benzodiazol-2-ylmethyl)-3-(hydroxymethyl)piperidin-3-ol
4-{4-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-6-methylpyrimidine
2-[(4aR,7aS)-4-[(2,4-difluorophenyl)methyl]-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]acetic acid
(3S,4S)-4-cyclopropyl-1-[ethyl(methyl)sulfamoyl]pyrrolidine-3-carboxylic acid
methyl 4-{[3-(3,4-difluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}benzoate
5-methyl-2-({[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]methyl}sulfanyl)-1H-1,3-benzodiazole
N-[1-(1-{[3-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]acetamide
(4aS,7aR)-1-{[3-(2,5-dimethylphenyl)-1H-pyrazol-4-yl]methyl}-4-methyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
9-(3-fluoro-4-hydroxybenzoyl)-2-methyl-2,9-diazaspiro[5.5]undecan-3-one
N-{[1-(3-methoxypropyl)pyrrolidin-3-yl]methyl}-6-(propan-2-yl)pyrimidin-4-amine
N-[(1,1-dioxo-1λ6-thiolan-3-yl)methyl]-2-(thiophen-3-yl)acetamide
8-{[2,5-dimethoxy-4-(methylsulfanyl)phenyl]methyl}-2,8-diazaspiro[4.5]decan-3-one
2-amino-6-(4-hydroxy-2-methylphenyl)-4-(2-methoxypyrimidin-5-yl)pyridine-3-carbonitrile
N-({6-methylimidazo[1,2-a]pyridin-2-yl}methyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
N-[3-hydroxy-1-(4-methylphenyl)propyl]-2-(1H-1,2,4-triazol-3-yl)benzamide
1-(1,4-dioxan-2-ylmethyl)-3-(3-methyl-1,2,4-thiadiazol-5-yl)urea
1-{[3-(2,5-dimethylphenyl)-1H-pyrazol-4-yl]methyl}-4-[2-(methylsulfanyl)ethyl]piperazine