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5-chloro-2-[3-(1-ethyl-1H-imidazol-2-yl)piperidine-1-carbonyl]phenol
1-acetyl-N-[(2R,3R)-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]piperidine-4-carboxamide
7-[1-(1,3-benzoxazol-2-yl)piperidin-4-yl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
4-(1-{[8-methyl-2-(piperidine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}piperidin-4-yl)thiomorpholine
methyl N-[1-(4-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}piperidin-1-yl)-1-oxopropan-2-yl]carbamate
ethyl 1-(1,4-dithiepan-6-yl)-4-(2-phenoxyethyl)piperidine-4-carboxylate
6-phenyl-3-(1H-1,2,3,4-tetrazol-5-ylmethyl)-3H,4H-thieno[2,3-d]pyrimidin-4-one
2-{1-[(2-fluorophenyl)methyl]-4-[(1-methyl-1H-indol-3-yl)methyl]piperazin-2-yl}ethan-1-ol
2-(1-{[2-(2,4-dimethoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-4-yl)ethan-1-ol
2-[(2,5-difluorophenyl)methyl]-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
N-(2,3-dimethylpyridin-4-yl)-3-({methyl[1-(pyridin-3-yl)ethyl]amino}methyl)benzamide
4-[1-(2H-1,3-benzodioxol-5-yl)-1H-1,2,4-triazol-5-yl]-1-(pyridin-3-ylmethyl)pyrrolidin-2-one
(3S,9aR)-3-(4-aminobutyl)-8-[4-(trifluoromethyl)benzoyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
5-({[1-(3,4-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]amino}methyl)-2-methoxyphenol
5-(morpholin-4-yl)-2-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-2,3-dihydropyridazin-3-one
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-(4-methyl-1H-imidazole-5-carbonyl)piperidin-3-ol
4-oxo-4-[4-(1H-pyrazol-4-yl)phenyl]butanoic acid
5-{[methyl({5-propylpyrazolo[1,5-a]pyrimidin-7-yl})amino]methyl}pyrimidin-2-amine
methyl (2S,4R)-4-(5-chloro-3-phenyl-1H-indole-2-amido)-1-[(4-methoxy-3-methylphenyl)methyl]pyrrolidine-2-carboxylate
N-[4-(1H-1,2,3,4-tetrazol-1-yl)phenyl]-1-[3-(1H-1,2,3,4-tetrazol-1-yl)propanoyl]piperidine-4-carboxamide
N-[1-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-4-methoxycyclohexane-1-carboxamide
(1S,5R)-6-(cyclopropylmethyl)-3-[2-(3,4-dihydro-2H-1,4-benzoxazin-4-yl)-2-oxoethyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
2-{[3-(2-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}pyridine
2-(ethylamino)-N-{2-[2-(trifluoromethoxy)phenyl]ethyl}pyrimidine-5-carboxamide
(1S,5R)-6-(cyclopropylmethyl)-3-[(2,5-dichlorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
{2-oxo-2-[3-(4-phenylpiperazin-1-yl)piperidin-1-yl]ethyl}urea
1-methyl-5-{[(5-methylfuran-2-yl)methyl]amino}-N-(2-phenylethyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
8-(2-butoxyacetyl)-2-(cyclopropylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
6-chloro-N,N-diethyl-2-(1H-pyrazol-4-yl)quinoline-4-carboxamide
(2R)-N-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]oxolane-2-carboxamide
[2-({4-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]piperazin-1-yl}methyl)phenyl]methanol
N4-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-6-ethyl-5-methylpyrimidine-2,4-diamine
2-[1-(propan-2-yl)piperidin-4-yl]-1-{4-[2-(pyridin-4-yl)ethyl]piperazin-1-yl}ethan-1-one
1-(5-{[4-(3,6-dimethylpyrazin-2-yl)piperazin-1-yl]methyl}-1-methyl-1H-pyrrol-3-yl)ethan-1-one
N,3-dimethyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]-2-phenylbutanamide
1-(3-methoxyphenoxy)-3-({3-methyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}amino)propan-2-ol
5-[3-(benzyloxy)phenyl]pyrazin-2-amine
[(2-butyl-1H-imidazol-4-yl)methyl][(1-cyclopentylpiperidin-4-yl)methyl](oxolan-2-ylmethyl)amine
3-[1-(2,6-dimethylpyrimidine-4-carbonyl)piperidin-3-yl]-N-(4-fluoro-2-methylphenyl)propanamide
1-(4-chloro-3-methylphenoxy)-3-{[6-(methoxymethyl)pyrimidin-4-yl]amino}propan-2-ol
2-{2-ethyl-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}pyridine-3-carboxamide
(2S,4S)-4-(benzylamino)-1-(2,2-diphenylethyl)-N-methylpyrrolidine-2-carboxamide
1-(6-hydroxy-1,4-oxazepan-4-yl)-4-(1H-pyrazol-4-yl)butan-1-one
2-methoxyethyl 4-[4-ethyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carboxylate
2-methyl-6-[3-(pyridin-4-yl)azetidine-1-carbonyl]-2H,3H,5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridin-3-one
1-(azocan-1-yl)-3-(5-methoxy-2-{[methyl(1,2-oxazol-3-ylmethyl)amino]methyl}phenoxy)propan-2-ol
1-(3-ethyl-4-methyl-1H-pyrazole-5-carbonyl)-4-[(methylsulfanyl)methyl]piperidine
1-(cyclopropylmethyl)-N-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]piperidine-2-carboxamide
4-{[4-(pyridin-4-yl)piperidin-1-yl]methyl}-1H-pyrazole-3-carboxylic acid
(4aR,7aS)-N,N-dimethyl-4-[(4-methyl-1H-imidazol-5-yl)methyl]-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide