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N-benzyl{[2-(2-fluorophenoxy)pyridin-3-yl]amino}sulfonamide
[(5-methylfuran-2-yl)methyl][(2-phenoxypyridin-3-yl)methyl]amine
N-[2-(2-fluorophenyl)ethyl]-5-[4-hydroxy-1-(thiophen-3-ylmethyl)piperidin-4-yl]-1-benzofuran-2-carboxamide
1-(3-methoxyphenyl)-6-methyl-4-(1-methyl-1H-pyrazole-5-carbonyl)piperazin-2-one
5-[6-amino-5-cyano-4-(pyridin-3-yl)pyridin-2-yl]-2,4-dimethyl-1H-pyrrole-3-carboxylic acid
4-[(3,5-dimethoxyphenyl)methyl]-7-(pyridin-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
8-methanesulfonyl-2-[(2E)-3-phenylprop-2-en-1-yl]-2,8-diazaspiro[4.5]decan-3-one
2-{methyl[(5-methyl-1,2-oxazol-3-yl)methyl]amino}-1-phenylethan-1-ol
(2S)-2-({2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-1,3-oxazol-4-yl}formamido)-4-methylpentanamide
5-chloro-2-{2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}-1,2,3,4-tetrahydroisoquinoline
1-ethyl-N-methyl-3-(2-methylpropyl)-N-[2-(pyridin-2-yl)ethyl]-1H-pyrazole-5-carboxamide
2-{2-[2-(dimethylamino)-1,3-thiazol-5-yl]-1H-imidazol-1-yl}-3-phenylpropanoic acid
8-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-2-propyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
1-[2-(3-fluorophenyl)ethyl]-N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-6-oxopiperidine-3-carboxamide
(2E)-N-[1-(2-phenylethyl)piperidin-3-yl]-3-(pyridin-4-yl)prop-2-enamide
6-ethyl-N-{[3-(pyrrolidin-1-ylmethyl)phenyl]methyl}pyrimidin-4-amine
1-(3-ethyl-1,2-oxazole-5-carbonyl)-4-phenylpiperidine-4-carbonitrile
N-(1-cyclopropylethyl)-2-[(2,6-dichlorophenyl)methyl]-4-hydroxypyrimidine-5-carboxamide
(3S,4R)-N-(2,4-difluorophenyl)-3-(dimethylamino)-4-(propan-2-yl)pyrrolidine-1-carboxamide
2-methoxy-N-{1-[1-(2-methylfuran-3-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}benzamide
(1S,5R)-N-(3-cyanophenyl)-3-methyl-3,6-diazabicyclo[3.2.2]nonane-6-carboxamide
4-{[2-(1H-imidazol-4-yl)-1H-imidazol-1-yl]methyl}-1H-indole
1-(2-methoxyphenyl)-N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}-1H-pyrazole-4-carboxamide
1-tert-butyl-4-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-2-one
4-(5-{[3-(hydroxymethyl)-1-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}-1,2,4-oxadiazol-3-yl)benzoic acid
(2R,3R)-3-({[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}amino)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
methyl 1-[3-(2-hydroxyphenyl)-3-(3-hydroxyphenyl)propanoyl]piperidine-4-carboxylate
2-(1H-imidazol-2-yl)-N-[1-methyl-4-(propan-2-yloxy)-1H-indazol-3-yl]benzamide
5-[1-(1H-imidazol-2-ylmethyl)pyrrolidin-2-yl]-N-methyl-N-[(3-methyl-1,2-oxazol-5-yl)methyl]thiophene-2-carboxamide
4-methoxy-N-(2-methoxyethyl)-2-({1-[3-(methylsulfanyl)propyl]piperidin-4-yl}oxy)benzamide
1-(cyclohex-3-en-1-ylmethyl)-4-(1H-pyrazol-1-yl)piperidine-4-carboxylic acid
2-(1H-pyrazol-1-yl)-1-[4-(thiophen-2-ylmethyl)piperazin-1-yl]butan-1-one
N-[2-(1H-imidazol-1-yl)ethyl]-N-methyl-1-(6-methyl-2-phenylpyrimidin-4-yl)piperidin-4-amine
ethyl 4-[3-({[2-(1H-indol-3-yl)ethyl]amino}methyl)-6H,7H,8H-cyclopenta[g]quinolin-2-yl]piperazine-1-carboxylate
methyl 2-({4-[1-(2,5-dimethylfuran-3-carbonyl)piperidin-3-yl]-5-(4-fluorophenyl)pyrimidin-2-yl}sulfanyl)acetate
N-{[1-(3-methylphenyl)-1H-imidazol-2-yl]methyl}-1-(pyridin-2-yl)-4,5,6,7-tetrahydro-1H-indazol-4-amine
1-[2-(cyclopropylmethyl)-3-oxo-2,9-diazaspiro[5.5]undecan-9-yl]-4-phenylbutane-1,2-dione
(3R,4R)-4-(azepan-1-yl)-1-[(3,4,5-trimethoxyphenyl)methyl]piperidin-3-ol
4-{4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine-1-carbonyl}benzonitrile
3-methoxy-2-(quinolin-8-yl)pyridin-4-amine
3-({methyl[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]amino}methyl)quinolin-7-ol
9-[2-(4,5-dimethyl-1H-imidazol-1-yl)acetyl]-2-[3-(dimethylamino)propyl]-2,9-diazaspiro[5.5]undecan-3-one
3-[(dimethylamino)methyl]-1-[(4-methanesulfonylphenyl)methyl]piperidin-3-ol
2-(2H-1,2,3-benzotriazol-2-yl)-1-{4-[(3-methylphenyl)methyl]piperazin-1-yl}ethan-1-one
6-methyl-5-{4-[1-(pyrrolidin-1-yl)ethyl]phenyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
4-hydroxy-2-(3-methylphenyl)-N-[4-(pyridin-2-yl)butyl]pyrimidine-5-carboxamide
4-(butan-2-yl)-3-(3-methoxyphenyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
3-fluoro-2-{1-[(4-fluorophenyl)methyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl}pyridine
2-cyclopropyl-8-[2-methyl-5-(propan-2-yl)furan-3-carbonyl]-2,8-diazaspiro[5.5]undecan-3-one
N-(1-hydroxybutan-2-yl)-4-[(5-methyl-1H-1,2,3,4-tetrazol-1-yl)methyl]-N-(thiophen-3-ylmethyl)benzamide