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(2R,6R)-4-{[6-(dimethylamino)pyridin-3-yl]methyl}-11-methoxy-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
6-[(1R,5R)-6-benzyl-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]-2-methyl-2,3-dihydropyridazin-3-one
1-(2-phenylethyl)-3,8-bis(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-[3-(methylsulfanyl)propyl]-N-(6-phenoxypyridin-3-yl)piperidine-2-carboxamide
3-[(1S,5R)-3-(pyrazin-2-yl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-4,5,6,7-tetrahydro-1,2-benzoxazole
1-[(3R,4S)-3-amino-4-(3-methoxyphenyl)pyrrolidin-1-yl]-3-phenoxypropan-1-one
1-[(1R,5R)-6-[(4-chloro-3-fluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
2-ethyl-9-[(1-methyl-1H-imidazol-2-yl)methyl]-4-phenyl-2,9-diazaspiro[5.5]undecan-3-one
2-(2-aminoethyl)-N-methyl-N-{[2-(1H-pyrazol-1-yl)phenyl]methyl}quinazolin-4-amine
2-(3-phenylpropyl)-4-(pyridine-3-carbonyl)morpholine
1-(4-{2-[(9aS)-octahydro-1H-pyrrolo[1,2-a][1,4]diazepin-2-yl]-2-oxoethoxy}phenyl)propan-1-one
N-(4-fluorophenyl)-1-(2-methylfuran-3-carbonyl)piperidin-3-amine
2,5-dioxo-6-{[2-(pyrrolidin-1-yl)-1,3-thiazol-4-yl]methyl}-1,2,5,6-tetrahydro-1,6-naphthyridine-3-carbonitrile
5-{3-[(2-methylphenyl)methoxy]azetidine-1-carbonyl}-N-phenylpyrimidin-2-amine
2-[4-(piperidine-1-carbonyl)piperidin-1-yl]pyridine-4-carboxamide
N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-4-(1H-1,2,4-triazol-1-yl)butanamide
3-[4-(2,6-difluorophenyl)-1H-pyrazol-5-yl]-1-[(2-fluoro-4-methoxyphenyl)methyl]piperidine
dimethyl({[(3S,4R)-4-(propan-2-yl)-1-(2,4,5-trimethylbenzoyl)pyrrolidin-3-yl]sulfamoyl})amine
(3R,5S)-N3-(4-fluorophenyl)-1-[(4-hydroxyphenyl)methyl]-N5-[(2-methoxyphenyl)methyl]piperidine-3,5-dicarboxamide
1-(1H-imidazol-2-ylmethyl)-N-methyl-N-(2-phenylethyl)piperidin-3-amine
(3S,4R)-1-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-4-(pyridin-4-yl)pyrrolidine-3-carboxylic acid
2-[(2,6-dichlorophenyl)methyl]-4-hydroxy-N-[(2S)-1-methoxypropan-2-yl]pyrimidine-5-carboxamide
2-(1-cyclopentyl-1H-imidazol-2-yl)benzoic acid
2-methyl-N-({2-[(6-methylpyridin-3-yl)oxy]pyridin-3-yl}methyl)-3-(pyrrolidin-1-yl)propanamide
[(3-methoxyphenyl)methyl]({[2-(morpholine-4-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl})amine
3-(oxolan-3-yl)-5-(2-propyl-1,3-thiazol-4-yl)-1,2,4-oxadiazole
1-[(1R,3S)-1-hydroxy-3-methoxy-7-azaspiro[3.5]nonan-7-yl]-3-(4H-1,2,4-triazol-4-yl)propan-1-one
3-(1-propyl-1H-1,2,3-triazol-4-yl)-1-[3-(1,2,3,4-tetrahydroquinolin-1-yl)propyl]urea
5-{[3-(2,3-dimethoxyphenyl)pyrrolidin-1-yl]methyl}-2-(pyridin-2-yl)pyrimidine
2-(4-methoxypiperidin-1-yl)-5-{4-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}pyridine
2-propyl-1-{pyrazolo[1,5-a]pyrimidin-3-yl}-1H-imidazole
6-methoxy-N-[3-(4-methylpiperazin-1-yl)propyl]-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
N-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-6-cyclopropyl-3-methyl-[1,2]oxazolo[5,4-b]pyridine-4-carboxamide
1-[3-(3-hydroxypiperidin-1-yl)propyl]-3-[2-(4-methoxyphenyl)phenyl]urea
(4aS,8aS)-2-[(4-phenoxyphenyl)methyl]-decahydro-2,7-naphthyridin-4a-ol
4-({3-[3-(1H-imidazol-1-yl)propoxy]phenyl}methyl)-2-methyl-1-(propan-2-yl)piperazine
methyl 6-{[butyl(methyl)amino]methyl}-3-(1,3-dimethyl-1H-pyrazole-5-amido)thieno[2,3-b]pyridine-2-carboxylate
2-[1-(1-{furo[3,2-c]pyridin-4-yl}piperidin-4-yl)-1H-1,2,3-triazol-4-yl]propan-2-ol
3-benzyl-4-(2-methoxyquinoline-4-carbonyl)piperazin-2-one
2-methyl-4-phenyl-9-[3-(pyridin-3-yl)propanoyl]-2,9-diazaspiro[5.5]undecan-3-one
[3-(2-methoxyethyl)-1-[(6-methyl-2H-1,3-benzodioxol-5-yl)methyl]piperidin-3-yl]methanol
9-[3-(4-fluorophenoxy)propyl]-2-(prop-2-en-1-yl)-2,9-diazaspiro[5.5]undecan-3-one
3-[(3R,4S)-1-{[5-(3-fluorophenyl)-1,3,4-oxadiazol-2-yl]methyl}-4-(morpholin-4-yl)piperidin-3-yl]propan-1-ol
(2R)-2-cyclohexyl-2-hydroxy-N-({2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}methyl)acetamide
N-[(3R,4S)-4-cyclopropyl-1-[(1-methyl-1H-imidazol-5-yl)methyl]pyrrolidin-3-yl]-2-methanesulfonamidoacetamide
4-{[5-(piperidin-1-ylmethyl)thiophen-2-yl]methyl}thiomorpholine
2-{[1-(3-methoxyphenyl)propan-2-yl]amino}-N,N-dimethylethane-1-sulfonamide
N,4-dimethyl-3-(2-oxoimidazolidin-1-yl)-N-[1-(2-phenylethyl)piperidin-3-yl]benzamide
1-ethyl-4-{3-[2-(6-methylpyridin-2-yl)-1H-imidazol-1-yl]propyl}piperazine
N-(3,4-dimethoxyphenyl)-1-(quinoxalin-2-yl)piperidin-3-amine