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methyl 3-(2-phenylacetamido)-5-[(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylformamido)methyl]benzoate
N,N-diethyl-1-(1-{2-[2-(3-methoxyphenyl)ethyl]-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl}piperidine-3-carbonyl)piperidine-3-carboxamide
8-(4-hydroxy-3-methylbenzoyl)-2-(3-methoxypropyl)-2,8-diazaspiro[4.5]decan-3-one
3-[2-(propan-2-yl)-1H-1,3-benzodiazol-5-yl]-1-{3-[(pyridin-3-yl)amino]propyl}urea
4-tert-butyl-6-{4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-1,2-dihydropyrimidin-2-one
N-ethyl-N-({1-[2-(3-fluorophenyl)ethyl]piperidin-3-yl}methyl)-2-(4-methoxyphenyl)acetamide
[(3R,4R)-1-{[1-(4-chlorophenyl)-1H-pyrazol-4-yl]methyl}-4-(pyrrolidin-1-ylmethyl)pyrrolidin-3-yl]methanol
4-[1-(5-chloro-2-methoxyphenyl)-3-cyclopropyl-1H-1,2,4-triazol-5-yl]pyridazine
1-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}-2-(2-methoxyphenyl)pyrrolidine
1-(4-{1-[(3-methyl-1H-pyrazol-5-yl)methyl]-4-phenyl-1H-imidazol-5-yl}phenyl)ethan-1-one
methyl (2S)-2-phenyl-2-({1-[3-(pyridine-4-amido)phenyl]piperidin-4-yl}amino)acetate
[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl](methyl)[1-(4-methylpyridin-2-yl)propan-2-yl]amine
3-(1,1-dioxo-1λ6-thiolan-3-yl)-3-(2-hydroxyethyl)-1-[3-(1,3-oxazol-5-yl)phenyl]urea
1-{[4-(3,5-dimethoxyphenyl)phenyl]methyl}piperazine
N-[3-(dimethyl-1,2-oxazol-4-yl)propyl]-6-(4-ethylpiperazin-1-yl)pyridine-3-carboxamide
5-methyl-4-[1-(1-methyl-1H-pyrazole-5-carbonyl)piperidin-3-yl]-2-[(oxolan-2-ylmethyl)sulfanyl]pyrimidine
2-{5-[1-(2-methoxyethyl)pyrrolidin-3-yl]-3-methyl-1H-1,2,4-triazol-1-yl}pyridine
3-(3-hydroxy-3-methylbutyl)-N-(isoquinolin-5-ylmethyl)-N-methylbenzamide
4-hydroxy-N-(2-methoxyethyl)-N-(1,3-thiazol-2-ylmethyl)-2-(thiophen-2-yl)pyrimidine-5-carboxamide
3-butyl-1-methyl-4-(3,5,7-trimethyl-1H-indole-2-carbonyl)piperazin-2-one
1-(2-ethoxyethyl)-3-(3-methylbutyl)-2-oxo-1H,2H,3H-imidazo[4,5-b]pyridine-6-carboxylic acid
N-[2-(4-methyl-1H-1,2,3-triazol-1-yl)ethyl]-5-phenyl-1,2-oxazole-3-carboxamide
2-benzyl-9-(4-hydroxy-1-methylpiperidine-4-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
N-[1-(3-fluoro-4-hydroxyphenyl)ethyl]-2-(methylamino)pyridine-3-carboxamide
N-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-5-(3,4-dimethylphenoxymethyl)-1,2-oxazole-3-carboxamide
N-ethyl-3-fluoro-N-({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)benzamide
1-(1,3-benzoxazol-2-yl)-N-{[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}piperidin-4-amine
[2-(2-{[2-(4-fluorophenyl)morpholin-4-yl]methyl}-6-methoxyphenoxy)ethyl]dimethylamine
1-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]-4-(pyrrolidine-1-sulfonyl)piperazine
2-({[5-methyl-2-(thiophen-2-yl)-1,3-oxazol-4-yl]methyl}(thiophen-2-ylmethyl)amino)ethan-1-ol
1-[1-(4-methoxypyrimidin-2-yl)piperidin-3-yl]pyrrolidin-2-one
1-(2-{2-[2-(4-hydroxyphenyl)ethyl]piperidin-1-yl}-2-oxoethyl)imidazolidine-2,4-dione
(2S,4S)-1-[(4-chlorophenyl)methyl]-4-{[(3,4-difluorophenyl)methyl]amino}-N-(2-methoxyethyl)pyrrolidine-2-carboxamide
methyl 2-{[2-(2,3-difluorophenoxymethyl)-1,3-oxazol-4-yl]formamido}acetate
2-{5-[5-(hydroxymethyl)furan-2-yl]-1-(2-methyl-1,3-benzothiazol-6-yl)-1H-1,2,4-triazol-3-yl}acetamide
1-[3-(methylsulfanyl)butyl]-4-(4H-1,2,4-triazol-3-yl)piperidine
2-[1-(2,3-dihydro-1H-inden-2-yl)-5-(1,1-dioxo-1λ6-thiolan-3-yl)-1H-1,2,4-triazol-3-yl]acetamide
ethyl 2-({5-[2-amino-3-cyano-6-(1H-pyrrol-3-yl)pyridin-4-yl]pyrimidin-2-yl}(methyl)amino)acetate
N-(1-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)-1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
7-oxo-2-(2-phenylacetamido)-N-[2,2,2-trifluoro-1-(furan-2-yl)ethyl]-4,5,6,7-tetrahydro-1,3-benzothiazole-5-carboxamide
1-{2,7-dimethylpyrazolo[1,5-a]pyrimidine-5-carbonyl}-2-(4-fluorophenyl)piperidine
5-methyl-N-{2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}pyrazolo[1,5-a]pyrimidin-7-amine
2-{2-[(3S,4S)-3,4-dihydroxypiperidin-1-yl]-2-oxoethyl}-3-(thiophen-2-yl)cyclopent-2-en-1-one
N-[2-(5-chloro-4-methyl-1,3-thiazol-2-yl)ethyl]-1-(furan-2-ylmethyl)piperidine-3-carboxamide
2-{methyl[2-(4-methyl-1,3-thiazol-5-yl)ethyl]amino}acetic acid
N-[3-(phenylsulfanyl)propyl]oxane-2-carboxamide
1-[(1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-(3-methyl-1,2-oxazol-5-yl)ethan-1-one
methyl (1R,3S,3aR,6aS)-3-[5-methoxy-2-(1H-pyrazol-1-yl)phenyl]-5-methyl-4,6-dioxo-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
2-methyl-6-{2-methyl-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-1-yl}pyridine
5-amino-1-[2-(6-methoxynaphthalen-2-yl)morpholin-4-yl]pentan-1-one