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8-(1H-1,3-benzodiazol-2-ylmethyl)-3-[(3-methoxyphenyl)methyl]-1-(3-methylbutyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-{3-[2-(4-fluorophenyl)ethyl]piperidin-1-yl}ethan-1-one
2-{imidazo[1,2-a]pyridin-2-yl}-7-phenyl-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
N-{3-[2-(3,4-dichlorophenyl)morpholin-4-yl]-3-oxopropyl}acetamide
3-(3-fluorophenyl)-N-{[3-(oxolan-3-ylmethoxy)phenyl]methyl}-N-(pyridin-2-ylmethyl)benzamide
N-[(3R,4R)-1-[(2,3-dimethoxyphenyl)methyl]-3-hydroxypiperidin-4-yl]pyridine-2-carboxamide
2-{1-[(4-methoxy-3-methylphenyl)methyl]-4-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]piperazin-2-yl}ethan-1-ol
1-[2-(2-chlorophenyl)ethyl]-N-[(2,3-dimethoxyphenyl)methyl]-2-(methoxymethyl)-6-methyl-4-oxo-1,4-dihydropyridine-3-carboxamide
1-[(4-fluorophenyl)methyl]-5-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazole
N-({1-[(3-methyl-1H-pyrazol-5-yl)methyl]pyrrolidin-3-yl}methyl)-1-phenylcyclopropane-1-carboxamide
N-[(2,2-dimethyl-2,3-dihydro-1-benzofuran-5-yl)methyl]-5-[(4-hydroxypiperidin-1-yl)methyl]-1,2-oxazole-3-carboxamide
1-cyclopentyl-4-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]piperidine
methyl 1-{5-[(2E)-but-2-en-1-yl]-1,3,4-oxadiazole-2-carbonyl}-3-phenylpyrrolidine-3-carboxylate
2-(4-fluorophenyl)-N-methyl-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}benzamide
N'-cyclopentyl-N-[1-(1H-pyrazol-1-yl)propan-2-yl]butanediamide
6-(3-oxo-2,3-dihydro-1H-indene-1-carbonyl)-N-[(4-phenyloxan-4-yl)methyl]-6-azaspiro[2.5]octane-1-carboxamide
N-[(3S,4R)-4-(5-methylfuran-2-yl)-1-{[3-(5-methylfuran-2-yl)phenyl]methyl}pyrrolidin-3-yl]acetamide
methyl 6-[(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-3-hydroxypiperidin-1-yl]pyrazine-2-carboxylate
3-bromo-5-[(4-methylpiperazin-1-yl)sulfonyl]benzoic acid
N-({5-cyclohexyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-2-[(cyclopropylmethyl)sulfanyl]acetamide
2-[(1-benzyl-1H-imidazol-5-yl)methyl]-7-methyl-2,7-diazaspiro[4.5]decan-6-one
2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-(2-ethoxyethyl)-1,3-oxazole-4-carboxamide
2-methoxy-3-{4-[1-(piperidin-1-yl)ethyl]phenyl}pyrazine
(1S,5R)-3-(2-{3-oxo-2H,3H,4H-pyrido[3,2-b][1,4]oxazin-4-yl}acetyl)-6-propyl-3,6-diazabicyclo[3.2.2]nonan-7-one
1-[(3S,4S)-3,4-dihydroxy-4-methylpiperidin-1-yl]-2-(1,3-thiazol-5-yl)ethan-1-one
2-{2-[(6-methoxypyrimidin-4-yl)amino]ethyl}-6-phenyl-2,3,4,5-tetrahydropyridazin-3-one
(3S,4S)-4-cyclopropyl-1-[4-(pyrrolidine-1-carbonyl)pyridin-2-yl]pyrrolidine-3-carboxylic acid
(3aS,6aR)-3-[2-(3-chlorophenyl)ethyl]-5-[6-(dimethylamino)pyrimidin-4-yl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
1-[(3-fluorophenyl)methyl]-4-(1-methyl-5-phenyl-1H-pyrrole-2-carbonyl)piperazine
(4aR,7aS)-1-methyl-4-(5-methyl-2-phenylfuran-3-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-(3-{[3-(2-chlorophenoxy)azetidin-1-yl]methyl}phenoxy)ethan-1-ol
N-{2-[4-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)morpholin-2-yl]ethyl}propanamide
[(1R,3S,3aS,6aR)-3-[3-chloro-4-(prop-2-en-1-yloxy)phenyl]-1-ethyl-5-methyl-octahydropyrrolo[3,4-c]pyrrol-1-yl]methanol
(4aS,7aR)-1-{[6-(dimethylamino)pyridin-3-yl]methyl}-4-(2-methoxyethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-{[1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}-4-phenylpyrrolidin-2-one
3-(benzylsulfanyl)-1-(3-hydroxy-3,4,4-trimethylpyrrolidin-1-yl)propan-1-one
1-[3-(cyclohexyloxy)-2-hydroxypropyl]-3-(2-ethyl-1H-1,3-benzodiazol-6-yl)urea
N,N-dimethyl-2-[(1S,5R)-6-{[2-(propylamino)pyrimidin-5-yl]methyl}-3,6-diazabicyclo[3.2.2]nonan-3-yl]acetamide
9-(1-methyl-1H-pyrazole-4-carbonyl)-2-[2-(pyridin-3-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
1-{3-[2-(4-fluorophenyl)morpholin-4-yl]-3-oxopropyl}azepan-2-one
N-{[1-(1H-1,3-benzodiazol-2-ylmethyl)pyrrolidin-3-yl]methyl}propane-1-sulfonamide
N-[3-(isoquinolin-1-yl)phenyl]acetamide
N-[(1-ethylpyrrolidin-2-yl)methyl]-3-{1-[2-(pyridin-3-yl)acetyl]piperidin-4-yl}propanamide
methyl 6-[3-(2-fluorophenyl)benzoyl]-2-(methylsulfamoyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
2-(3,5-dimethoxyphenyl)-1-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}ethan-1-one
2-amino-4-[2-(2-hydroxyethoxy)phenyl]-6-(2-methoxyphenyl)pyridine-3-carbonitrile
4-[(3-chloro-4,5-dimethoxyphenyl)methyl]-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
1-[(3,4-dimethoxypyridin-2-yl)methyl]-1,2,3,4-tetrahydroquinolin-2-one
(2S)-3-methyl-2-({6-methyl-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-yl}amino)butanamide
2-(1-{[1-(9H-purin-6-yl)piperidin-3-yl]methyl}-1H-1,2,3-triazol-4-yl)propan-2-ol